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Search Count: 10

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8TWY image
Structure Of P110 Alpha Bound To (S)-1-(4-((2-(4-(4-(2-Amino-4-(Difluoromethyl)Pyrimidin-5-Yl)-6-(3-Methylmorpholino)-1,3,5- Triazin-2-Yl)Piperazin-1-Yl)-2-Oxoethoxy)Methyl)Piperidin-1-Yl)Prop-2-En-1-One (Compound 9)

6OAC image
Pqr530 [(S)-4-(Difluoromethyl)-5-(4-(3-Methylmorpholino)-6-Morpholino-1,3,5-Triazin-2-Yl)Pyridin-2-Amine] Bound To The Pi3Ka Catalytic Subunit P110Alpha
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:3.15 Å Release Date: 2019-06-26
Classification: TRANSFERASE
Ligands: M1J

6GY0 image
Mpi3Kd In Complex With Az3
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Resolution:2.55 Å Release Date: 2019-02-06
Classification: TRANSFERASE
Ligands: FGE

5OQ4 image
Pqr309 - A Potent, Brain-Penetrant, Orally Bioavailable, Pan-Class I Pi3K/Mtor Inhibitor As Clinical Candidate In Oncology
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.70 Å Release Date: 2017-09-06
Classification: TRANSFERASE
Ligands: A3W, SO4

5M8D image
Tubulin Mtd265-R1 Complex

5JHA image
Structure Of Phosphoinositide 3-Kinase Gamma (Pi3K) Bound To The Potent Inhibitor Pikin2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.51 Å Release Date: 2017-03-15
Classification: TRANSFERASE
Ligands: 6K7, SO4

5JHB image
Structure Of Phosphoinositide 3-Kinase Gamma (Pi3K) Bound To The Potent Inhibitor Pikin3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.48 Å Release Date: 2017-03-15
Classification: TRANSFERASE
Ligands: 6K5, SO4



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