Search Count: 27
![]() |
Co-Crystal Structure Of P. Aeruginosa Lpxc-50067 Complex
Organism: Pseudomonas aeruginosa pao1
Method: X-RAY DIFFRACTION Resolution:1.84 Å Release Date: 2019-07-17 Classification: HYDROLASE/INHIBITOR Ligands: MG, JWM |
Organism: Pseudomonas aeruginosa pao1
Method: X-RAY DIFFRACTION
Release Date: 2019-07-17
Ligands: MG, JWM
![]() |
Co-Crystal Structure Of P. Aeruginosa Lpxc-50228 Complex
Organism: Pseudomonas aeruginosa (strain atcc 15692 / dsm 22644 / cip 104116 / jcm 14847 / lmg 12228 / 1c / prs 101 / pao1)
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2019-07-17 Classification: HYDROLASE/INHIBITOR Ligands: JWP, MG |
![]() |
Co-Crystal Structure Of P. Aeruginosa Lpxc-50432 Complex
Organism: Pseudomonas aeruginosa
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2019-07-17 Classification: HYDROLASE/INHIBITOR Ligands: MG, JWV, GOL |
Organism: Pseudomonas aeruginosa
Method: X-RAY DIFFRACTION
Release Date: 2019-07-17
Ligands: MG, JWV, GOL
![]() |
Co-Crystal Structure Of P. Aeruginosa Lpxc-Achn975 Complex
Organism: Pseudomonas aeruginosa
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2019-07-17 Classification: HYDROLASE/INHIBITOR Ligands: ZN, A5F |
Organism: Pseudomonas aeruginosa
Method: X-RAY DIFFRACTION
Release Date: 2019-07-17
Ligands: ZN, A5F
![]() |
Map4K4 In Complex With Inhibitor Gne-495
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.89 Å Release Date: 2015-09-02 Classification: Transferase/Transferase Inhibitor Ligands: MG, MES, 4P4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-02
Ligands: MG, MES, 4P4
![]() |
Lactate Dehydrogenase In Complex With Inhibitor Compound 31
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.11 Å Release Date: 2014-12-24 Classification: OXIDOREDUCTASE Ligands: NAI, EPE, W31, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-24
Ligands: NAI, EPE, W31, SO4
![]() |
Lactate Dehydrogenase In Complex With Inhibitor Compound 13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.19 Å Release Date: 2014-12-24 Classification: OXIDOREDUCTASE Ligands: EPE, NAI, W13, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-24
Ligands: EPE, NAI, W13, SO4
![]() |
Mitogen-Activated Protein Kinase Kinase (Mek1) Bound To G805
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.81 Å Release Date: 2014-09-24 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: MG, 3EW, ANP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-09-24
Ligands: MG, 3EW, ANP
![]() |
Mek 1 Kinase Bound To G799
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2014-09-24 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: ANP, 3EX, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-09-24
Ligands: ANP, 3EX, MG
![]() |
Mek1 Kinase Bound To Small Molecule Inhibitor G659
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2014-09-24 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: MG, 3EY, ANP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-09-24
Ligands: MG, 3EY, ANP
![]() |
Map4K4 In Complex With Inhibitor (Compound 6)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.18 Å Release Date: 2014-09-03 Classification: Transferase/Transferase inhibitor Ligands: 3D8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-09-03
Ligands: 3D8
![]() |
Map4K4 In Complex With Inhibitor (Compound 16)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.43 Å Release Date: 2014-09-03 Classification: Transferase/Transferase inhibitor Ligands: MES, NA, 3D9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-09-03
Ligands: MES, NA, 3D9
![]() |
Map4K4 In Complex With Inhibitor (Compound 25)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.58 Å Release Date: 2014-09-03 Classification: Transferase/Transferase inhibitor Ligands: MG, 3DC, MES |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-09-03
Ligands: MG, 3DC, MES
![]() |
Lactate Dehydrogenase A In Complex With Substituted 3-Hydroxy-2-Mercaptocyclohex-2-Enone Compound 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.14 Å Release Date: 2014-07-16 Classification: oxidoreductase/oxidoreductase inhibitor Ligands: NAI, EPE, 36V, 2OP, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-16
Ligands: NAI, EPE, 36V, 2OP, SO4
![]() |
Lactate Dehydrogenase A In Complex With Substituted 3-Hydroxy-2-Mercaptocyclohex-2-Enone Compound 104
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2014-07-16 Classification: oxidoreductase/oxidoreductase inhibitor Ligands: NAI, EPE, SO4, 36U, LAC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-16
Ligands: NAI, EPE, SO4, 36U, LAC
![]() |
Map4K4 In Complex With Inhibitor (Compound 22), 6-(3-Chlorophenyl)Quinazolin-4-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2014-04-23 Classification: transferase/transferase inhibitor Ligands: MES, NA, 2QV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-23
Ligands: MES, NA, 2QV
![]() |
Map4K4 In Complex With Inhibitor (Compound 29), 6-(2-Fluoropyridin-4-Yl)Pyrido[3,2-D]Pyrimidin-4-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.27 Å Release Date: 2014-04-23 Classification: transferase/transferase inhibitor Ligands: MG, MES, 2QU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-23
Ligands: MG, MES, 2QU
![]() |
Map4K4 In Complex With Inhibitor (Compound 31), N-[3-(4-Aminoquinazolin-6-Yl)-5-Fluorophenyl]-2-(Pyrrolidin-1-Yl)Acetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.19 Å Release Date: 2014-04-23 Classification: transferase/transferase inhibitor Ligands: MES, MG, 2QT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-23
Ligands: MES, MG, 2QT
![]() |
Back Pocket Flexibility Provides Group-Ii Pak Selectivity For Type 1 Kinase Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2014-02-12 Classification: transferase/transferase inhibitor Ligands: 7KC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-02-12
Ligands: 7KC
![]() |
Back Pocket Flexibility Provides Group-Ii Pak Selectivity For Type 1 Kinase Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2014-02-12 Classification: transferase/transferase inhibitor Ligands: 2OL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-02-12
Ligands: 2OL
