Search Count: 16
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Co-Crystal Structure Of Human Smyd3 With Isoxazole Amides Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.59 Å Release Date: 2020-01-15 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, MG, GOL, SAH, LUP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-15
Ligands: ZN, MG, GOL, SAH, LUP
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Co-Crystal Structure Of Human Smyd3 With Isoxazole Amides Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2020-01-15 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, MG, EDO, SAM, L0J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-15
Ligands: ZN, MG, EDO, SAM, L0J
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Co-Crystal Structure Of Human Smyd3 With Isoxazole Amides Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.19 Å Release Date: 2020-01-15 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, MG, SAM, O41 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-15
Ligands: ZN, MG, SAM, O41
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Co-Crystal Structure Of Human Smyd3 With Isoxazole Amides Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.24 Å Release Date: 2020-01-15 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, MG, GOL, SAM, O6A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-15
Ligands: ZN, MG, GOL, SAM, O6A
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X-Ray Structure Of Polypeptide Deformylase Bound To A Acylprolinamide Inhibitor
Organism: Streptococcus pneumoniae
Method: X-RAY DIFFRACTION Resolution:1.78 Å Release Date: 2012-05-30 Classification: hydrolase/hydrolase inhibitor Ligands: NI, 0S5 |
Organism: Streptococcus pneumoniae
Method: X-RAY DIFFRACTION
Release Date: 2012-05-30
Ligands: NI, 0S5
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Phosphoinositide-Dependent Kinase-1 (Pdk1) With Lead Compound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2011-06-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GOL, SO4, JMZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-06-22
Ligands: GOL, SO4, JMZ
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Phosphoinositide-Dependent Kinase-1 (Pdk1) With Fragment8
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.75 Å Release Date: 2011-05-25 Classification: TRANSFERASE Ligands: GOL, JNZ, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-05-25
Ligands: GOL, JNZ, SO4
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Phosphoinositide-Dependent Kinase-1 (Pdk1) With Fragment11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2011-05-25 Classification: TRANSFERASE Ligands: GOL, SO4, JOZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-05-25
Ligands: GOL, SO4, JOZ
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Phosphoinositide-Dependent Kinase-1 (Pdk1) With Fragment17
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2011-05-25 Classification: TRANSFERASE Ligands: GOL, SO4, JPZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-05-25
Ligands: GOL, SO4, JPZ
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Phosphoinositide-Dependent Kinase-1 (Pdk1) Kinase Domain With 6-(3-Amino-1H-Indazol-6-Yl)-N4-Ethyl-2,4-Pyrimidinediamine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2011-03-09 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GOL, SO4, 3Q0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-09
Ligands: GOL, SO4, 3Q0
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Phosphoinositide-Dependent Kinase-1 (Pdk1) Kinase Domain With 6-[2-Amino-6-(4-Morpholinyl)-4-Pyrimidinyl]-1H-Indazol-3-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.49 Å Release Date: 2011-03-09 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GOL, SO4, 3Q1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-09
Ligands: GOL, SO4, 3Q1
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Phosphoinositide-Dependent Kinase-1 (Pdk1) Kinase Domain With 6-{2-Amino-6-[(3R)-3-Methyl-4-Morpholinyl]-4-Pyrimidinyl}-1H-Indazol-3-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2011-03-09 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GOL, SO4, 3Q2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-09
Ligands: GOL, SO4, 3Q2
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Phosphoinositide-Dependent Kinase-1 (Pdk1) Kinase Domain With 4-[2-Amino-6-(3-Amino-1H-Indazol-6-Yl)-4-Pyrimidinyl]-N-Phenyl-2-Morpholinecarboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2011-03-09 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GOL, SO4, 3Q3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-09
Ligands: GOL, SO4, 3Q3
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Phosphoinositide-Dependent Kinase-1 (Pdk1) Kinase Domain With (2R,5S)-1-[2-Amino-6-(3-Amino-1H-Indazol-6-Yl)-4-Pyrimidinyl]-6-Methyl-N-Phenyl-3-Piperidinecarboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2011-03-09 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GOL, SO4, 3Q4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-09
Ligands: GOL, SO4, 3Q4
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Phosphoinositide-Dependent Kinase-1 (Pdk1) Kinase Domain With 1,1-Dimethylethyl {(3R,6S)-1-[2-Amino-6-(3-Amino-1H-Indazol-6-Yl)-4-Pyrimidinyl]-6-Methyl-3-Piperidinyl}Carbamate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2011-03-09 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3Q5, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-09
Ligands: 3Q5, SO4, GOL
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Phosphoinositide-Dependent Kinase-1 (Pdk1) Kinase Domain With 1,1-Dimethylethyl{(3R,5R)-1-[2-Amino-6-(3-Amino-1H-Indazol-6-Yl)-4-Pyrimidinyl]-5-Methyl-3-Piperidinyl}Carbamate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2011-03-09 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3Q6, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-09
Ligands: 3Q6, SO4