Search Count: 28
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Crystal Structure Of Parp1 Catalytic Domain Bound To Azd5305 (Saruparib)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.59 Å Release Date: 2024-12-04 Classification: TRANSFERASE Ligands: A1H63, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-04
Ligands: A1H63, SO4
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Crystal Structure Of Parp1 Catalytic Domain Bound To Azd9574
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.82 Å Release Date: 2024-12-04 Classification: TRANSFERASE Ligands: A1H64, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-04
Ligands: A1H64, SO4
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Parp1 Catalytic Domain In Complex With 8-Chloroquinazolinone-Based Inhibitor (Compound 9)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2021-09-15 Classification: TRANSFERASE Ligands: VKW, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-15
Ligands: VKW, SO4
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Parp1 Catalytic Domain In Complex With Isoquinolone-Based Inhibitor (Compound 16)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2021-09-15 Classification: TRANSFERASE Ligands: VKT, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-15
Ligands: VKT, SO4
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Parp1 Catalytic Domain In Complex With A Selective Pyridine Carboxamide-Based Inhibitor (Compound 22)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2021-09-15 Classification: TRANSFERASE Ligands: VKQ, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-15
Ligands: VKQ, SO4
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Apo Mcl1 In A Complex With A Scfv
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2019-11-06 Classification: APOPTOSIS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-06
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Mcl1-Scfv Complex With An Indole Acid Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.38 Å Release Date: 2019-11-06 Classification: APOPTOSIS Ligands: HVN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-06
Ligands: HVN
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Mcl1 In Complex With A Fab
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.24 Å Release Date: 2019-11-06 Classification: APOPTOSIS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-06
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Structure Of An Anti-Mcl1 Scfv
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2019-11-06 Classification: APOPTOSIS Ligands: TLA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-06
Ligands: TLA
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Structure Of Anti-Mcl1 Fab
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.56 Å Release Date: 2019-11-06 Classification: APOPTOSIS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-06
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Structure Of An Anti-Mcl1 Scfv
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.43 Å Release Date: 2019-11-06 Classification: APOPTOSIS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-06
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Structure Of An Anti-Mcl1 Scfv
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.96 Å Release Date: 2019-11-06 Classification: APOPTOSIS Ligands: DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-06
Ligands: DMS
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Mth1 Substrate Recognition: Complex With A Methylaminopyrimidinedione.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.67 Å Release Date: 2017-01-18 Classification: HYDROLASE Ligands: ACT, S76, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-01-18
Ligands: ACT, S76, DMS
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Mth1 Substrate Recognition: Complex With 8-Oxo-Dgtp.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.56 Å Release Date: 2016-07-20 Classification: HYDROLASE Ligands: H6Y, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-07-20
Ligands: H6Y, ACT
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Mth1 Substrate Recognition: Complex With A Methylaminopurinone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.24 Å Release Date: 2016-07-20 Classification: HYDROLASE Ligands: UAN, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-07-20
Ligands: UAN, SO4
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Mth1 Substrate Recognition: Complex With A Methylbenzimidazolyl Acetamide.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.67 Å Release Date: 2016-07-20 Classification: HYDROLASE Ligands: ACT, N91, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-07-20
Ligands: ACT, N91, DMS
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Mth1 Substrate Recognition: Complex With A Aminomethylpyrimidinyl Oxypropanol.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.69 Å Release Date: 2016-07-20 Classification: HYDROLASE Ligands: 6Q3, ACT, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-07-20
Ligands: 6Q3, ACT, DMS
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Mth1 Substrate Recognition: Complex With 8-Oxo-Dgtp.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.63 Å Release Date: 2016-07-11 Classification: HYDROLASE Ligands: 8DG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-07-11
Ligands: 8DG
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Potent And Selective Inhibitors Of Mth1 Probe Its Role In Cancer Cell Survival
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2016-03-02 Classification: HYDROLASE Ligands: RX8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-03-02
Ligands: RX8
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Potent And Selective Inhibitors Of Mth1 Probe Its Role In Cancer Cell Survival
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2016-03-02 Classification: HYDROLASE Ligands: RJE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-03-02
Ligands: RJE
