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Search Count: 28

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9ETQ image
Crystal Structure Of Parp1 Catalytic Domain Bound To Azd5305 (Saruparib)

9ETR image
Crystal Structure Of Parp1 Catalytic Domain Bound To Azd9574

7ONR image
Parp1 Catalytic Domain In Complex With 8-Chloroquinazolinone-Based Inhibitor (Compound 9)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.05 Å Release Date: 2021-09-15
Classification: TRANSFERASE
Ligands: VKW, SO4

7ONS image
Parp1 Catalytic Domain In Complex With Isoquinolone-Based Inhibitor (Compound 16)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.97 Å Release Date: 2021-09-15
Classification: TRANSFERASE
Ligands: VKT, SO4

7ONT image
Parp1 Catalytic Domain In Complex With A Selective Pyridine Carboxamide-Based Inhibitor (Compound 22)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.85 Å Release Date: 2021-09-15
Classification: TRANSFERASE
Ligands: VKQ, SO4

6QB3 image
Apo Mcl1 In A Complex With A Scfv

6QB4 image
Mcl1-Scfv Complex With An Indole Acid Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.38 Å Release Date: 2019-11-06
Classification: APOPTOSIS
Ligands: HVN

6QB6 image
Mcl1 In Complex With A Fab

6QB9 image
Structure Of An Anti-Mcl1 Scfv
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.85 Å Release Date: 2019-11-06
Classification: APOPTOSIS
Ligands: TLA

6QBC image
Structure Of Anti-Mcl1 Fab

6QF9 image
Structure Of An Anti-Mcl1 Scfv

6QFC image
Structure Of An Anti-Mcl1 Scfv
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.96 Å Release Date: 2019-11-06
Classification: APOPTOSIS
Ligands: DMS

5FSO image
Mth1 Substrate Recognition: Complex With A Methylaminopyrimidinedione.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.67 Å Release Date: 2017-01-18
Classification: HYDROLASE
Ligands: ACT, S76, DMS

5FSK image
Mth1 Substrate Recognition: Complex With 8-Oxo-Dgtp.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.56 Å Release Date: 2016-07-20
Classification: HYDROLASE
Ligands: H6Y, ACT

5FSL image
Mth1 Substrate Recognition: Complex With A Methylaminopurinone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.24 Å Release Date: 2016-07-20
Classification: HYDROLASE
Ligands: UAN, SO4

5FSM image
Mth1 Substrate Recognition: Complex With A Methylbenzimidazolyl Acetamide.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.67 Å Release Date: 2016-07-20
Classification: HYDROLASE
Ligands: ACT, N91, DMS

5FSN image
Mth1 Substrate Recognition: Complex With A Aminomethylpyrimidinyl Oxypropanol.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.69 Å Release Date: 2016-07-20
Classification: HYDROLASE
Ligands: 6Q3, ACT, DMS

5FSI image
Mth1 Substrate Recognition: Complex With 8-Oxo-Dgtp.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.63 Å Release Date: 2016-07-11
Classification: HYDROLASE
Ligands: 8DG

5ANS image
Potent And Selective Inhibitors Of Mth1 Probe Its Role In Cancer Cell Survival
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.60 Å Release Date: 2016-03-02
Classification: HYDROLASE
Ligands: RX8

5ANT image
Potent And Selective Inhibitors Of Mth1 Probe Its Role In Cancer Cell Survival
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.00 Å Release Date: 2016-03-02
Classification: HYDROLASE
Ligands: RJE
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