Search Count: 15
 |
Trka With (6~{R})-3-Methylsulfanyl-6-Phenyl-1-(1~{H}-Pyrazol-3-Yl)-6,7-Dihydro-5~{H}-Thieno[3,4-C]Pyridin-4-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.33 Å Release Date: 2017-08-09 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 69C, CL, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-08-09
Ligands: 69C, CL, ACT
 |
Discovery Of Mli-2, An Orally Available And Selective Lrrk2 Inhibitor That Reduces Brain Kinase Activity
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:1.69 Å Release Date: 2017-03-15 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 81Y, SO4 |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2017-03-15
Ligands: 81Y, SO4
 |
Trka Jm-Kinase With 1-(9{H}-Fluoren-9-Yl)-3-(2-Methyl-4-Phenyl-Pyrimidin-5-Yl)Urea
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.87 Å Release Date: 2016-12-28 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6UE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-12-28
Ligands: 6UE
 |
Trka Jm-Kinase With {N}-(2-Pyridylmethyl)-2-[2-(2-Thienyl)Indol-1-Yl]Acetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.04 Å Release Date: 2016-12-28 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6UF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-12-28
Ligands: 6UF
 |
Trka Jm-Kinase With 2-Fluoro-{N}-[2-(4-Fluorophenyl)-6-Methyl-3-Pyridyl]-4-(Trifluoromethyl)Benzamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.24 Å Release Date: 2016-12-28 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6UG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-12-28
Ligands: 6UG
 |
Trka Jm-Kinase With 1-(5-Methyl-3-Phenyl-1,2-Oxazol-4-Yl)-3-[[2-(Trifluoromethyl)Phenyl]Methyl]Urea
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.01 Å Release Date: 2016-12-28 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6UH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-12-28
Ligands: 6UH
 |
Trka Jm-Kinase With 1-(2-Methyl-4-Phenyl-Pyrimidin-5-Yl)-3-(1-Naphthyl)Urea
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.12 Å Release Date: 2016-12-28 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6UJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-12-28
Ligands: 6UJ
 |
Trka Jm-Kinase With 1-(2-Methyl-4-Phenyl-Pyrimidin-5-Yl)-3-[[2-(Trifluoromethyl)Phenyl]Methyl]Urea
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.14 Å Release Date: 2016-12-28 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6UK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-12-28
Ligands: 6UK
 |
Trka Jm-Kinase With 1-(2-Methyl-4-Phenyl-Pyrimidin-5-Yl)-3-(2-Pyridyl)Urea
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.67 Å Release Date: 2016-12-28 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6UM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-12-28
Ligands: 6UM
 |
Identification Of Lxrbeta Selective Agonists For The Treatment Of Alzheimer'S Disease
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2016-04-06 Classification: SIGNALING PROTEIN Ligands: 668, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-06
Ligands: 668, PEG
 |
Identification Of Lxrbeta Selective Agonists For The Treatment Of Alzheimer'S Disease
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2016-04-06 Classification: SIGNALING PROTEIN Ligands: 668, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-06
Ligands: 668, SO4
 |
The Structure Of Trka Kinase Bound To The Inhibitor N-(3-Cyclopropyl-1-Phenyl-1H-Pyrazol-5-Yl)-2-{4-[3-Methoxy-4-(4-Methyl-1H-Imidazol-1-Yl)Phenyl]-1H-1,2,3-Triazol-1-Yl}Acetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2014-06-18 Classification: Transferase/Transferase inhibitor Ligands: 31V, GOL, CL, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-06-18
Ligands: 31V, GOL, CL, ACT
 |
The Structure Of Trka Kinase Bound To The Inhibitor 1-Cyclopropyl-1-[3-(1,3-Thiazol-2-Yl)Benzyl]-3-[4-(Trifluoromethoxy)Phenyl]Urea
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2014-06-18 Classification: Transferase/Transferase inhibitor Ligands: 31W, CL, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-06-18
Ligands: 31W, CL, ACT
 |
The Structure Of Trka Kinase Bound To The Inhibitor 4-Naphthalen-1-Yl-1-[(5-Phenyl-1,2,4-Oxadiazol-3-Yl)Methyl]-1H-Pyrrolo[3,2-C]Pyridine-2-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2014-06-18 Classification: Transferase/Transferase inhibitor Ligands: 31X, CL, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-06-18
Ligands: 31X, CL, ACT
 |
The Structure Of Trka Kinase Bound To The Inhibitor N~4~-(4-Morpholin-4-Ylphenyl)-N~6~-(Pyridin-3-Ylmethyl)Pyrido[3,2-D]Pyrimidine-4,6-Diamine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2014-06-18 Classification: Transferase/Transferase inhibitor Ligands: 31Y, CL, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-06-18
Ligands: 31Y, CL, ACT