Search Count: 11
![]() |
Structure Of Tead2 Bound To G8025
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2026-07-08 Classification: TRANSCRIPTION/INHIBITOR Ligands: A1CA7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-08
Ligands: A1CA7
![]() |
Structure Of Tead2 Bound To G2181
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2026-07-08 Classification: TRANSCRIPTION/INHIBITOR Ligands: A1CA6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-08
Ligands: A1CA6
![]() |
Crystal Structure Of Human Cyclic Gmp-Amp Synthase In Complex With Amppnp And Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2025-04-02 Classification: TRANSFERASE Ligands: A1AU3, GOL, MG, ANP, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-04-02
Ligands: A1AU3, GOL, MG, ANP, ZN
![]() |
Crystal Structure Of Human Cyclic Gmp-Amp Synthase In Complex With Amppnp And Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.47 Å Release Date: 2025-04-02 Classification: TRANSFERASE Ligands: MG, ZN, ANP, GOL, JUJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-04-02
Ligands: MG, ZN, ANP, GOL, JUJ
![]() |
Crystal Structure Of Human Cyclic Gmp-Amp Synthase (Cgas) In Complex With Compound 5; 3-((2-((3-Chloro-4-Fluorophenyl)Amino)-2-Oxoethyl)Carbamoyl)Picolinic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.53 Å Release Date: 2025-01-01 Classification: TRANSFERASE Ligands: ANP, A1BJH, ZN, MN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-01
Ligands: ANP, A1BJH, ZN, MN
![]() |
Crystal Structure Of Human Cyclic Gmp-Amp Synthase (Cgas) In Complex With Compound 36; (S)-(6,7-Dichloro-1-Methyl-1,3,4,5-Tetrahydro-2H-Pyrido[4,3-B]Indol-2-Yl)(5-(2-Hydroxyethoxy)Pyrimidin-2-Yl)Methanone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.25 Å Release Date: 2025-01-01 Classification: TRANSFERASE Ligands: ZN, A1BJA, ANP, MN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-01
Ligands: ZN, A1BJA, ANP, MN
![]() |
Crystal Structure Of Human Cyclic Gmp-Amp Synthase (Cgas) In Complex With Compound 23; (S)-1-(6,7-Dichloro-1-Methyl-1,3,4,5-Tetrahydro-2H-Pyrido[4,3-B]Indol-2-Yl)-2-Methoxyethan-1-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2025-01-01 Classification: TRANSFERASE Ligands: ZN, A1BJD, ANP, MN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-01
Ligands: ZN, A1BJD, ANP, MN
![]() |
Crystal Structure Of Selective Ire1A Inhibitor 29 At The Enzyme Active Site
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.43 Å Release Date: 2024-05-29 Classification: TRANSFERASE/INHIBITOR Ligands: EDO, XOE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-05-29
Ligands: EDO, XOE
![]() |
Crystal Structure Of Ire1A In Complex With G-6904
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2021-04-21 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: N8S, EPE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-04-21
Ligands: N8S, EPE
![]() |
Crystal Structure Of Ire1 In Complex With G-3053
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2021-04-21 Classification: TRANSFERASE/INHIBITOR Ligands: N97 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-04-21
Ligands: N97
![]() |
Crystal Structure Of Ire1A In Complex With G-4100
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.54 Å Release Date: 2021-04-21 Classification: TRANSFERASE/TRANSFERASE INHIBITOR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-04-21
