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Search Count: 11

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8SWE image
Fgfr2 Kinase Domain Bound To Reversible Inhibitor Cmpd 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.24 Å Release Date: 2024-02-14
Classification: ONCOPROTEIN
Ligands: GOL, GSH, WXQ

8U1F image
Fgfr2 Kinase Domain Bound To Irreversible Inhibitor Cmpd 10

8TS7 image
Human Pi3K P85Alpha/P110Alpha

8TS8 image
P85Alpha/P110Alpha Heterodimer H1047R Mutant

8TS9 image
Human Pi3K P85Alpha/P110Alpha H1047R Bound To Compound 1

8TSA image
Human Pi3K P85Alpha/P110Alpha H1047R Bound To Compound 2

8TSB image
Human Pi3K P85Alpha/P110Alpha Bound To Compound 2

8TSC image
Human Pi3K P85Alpha/P110Alpha H1047R Bound To Compound 3

8TSD image
Human Pi3K P85Alpha/P110Alpha Bound To Rly-2608


8STG image
Discovery And Clinical Validation Of Rly-4008, The First Highly Selective Fgfr2 Inhibitor With Activity Across Fgfr2 Alterations And Resistance Mutations
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