Search Count: 19
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Structure Of Vsd4-Nav1.7-Navpas Channel Chimera Bound To The Hybrid Inhibitor Gne-1305
Organism: Homo sapiens, Periplaneta americana
Method: ELECTRON MICROSCOPY Release Date: 2023-04-12 Classification: MEMBRANE PROTEIN/INHIBITOR Ligands: NAG, PEE, Y01, X7L |
Organism: Homo sapiens, Periplaneta americana
Method: ELECTRON MICROSCOPY
Release Date: 2023-04-12
Ligands: NAG, PEE, Y01, X7L
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Structure Of Vsd4-Nav1.7-Navpas Channel Chimera Bound To The Acylsulfonamide Inhibitor Gdc-0310
Organism: Homo sapiens, Periplaneta americana
Method: ELECTRON MICROSCOPY Release Date: 2023-04-12 Classification: MEMBRANE PROTEIN/INHIBITOR Ligands: BMA, NAG, X7R, PEE, Y01 |
Organism: Homo sapiens, Periplaneta americana
Method: ELECTRON MICROSCOPY
Release Date: 2023-04-12
Ligands: BMA, NAG, X7R, PEE, Y01
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Structure Of Vsd4-Nav1.7-Navpas Channel Chimera Bound To The Arylsulfonamide Inhibitor Gne-3565
Organism: Homo sapiens, Periplaneta americana
Method: ELECTRON MICROSCOPY Release Date: 2023-04-12 Classification: MEMBRANE PROTEIN/INHIBITOR Ligands: NAG, X7W, PEE, Y01 |
Organism: Homo sapiens, Periplaneta americana
Method: ELECTRON MICROSCOPY
Release Date: 2023-04-12
Ligands: NAG, X7W, PEE, Y01
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Structure Of Vsd4-Nav1.7-Navpas Channel Chimera Bound To The Hybrid Inhibitor Gne-9296
Organism: Homo sapiens, Periplaneta americana, Diguetia canities
Method: ELECTRON MICROSCOPY Release Date: 2023-04-12 Classification: MEMBRANE PROTEIN/INHIBITOR Ligands: NAG, X80, PEE, Y01 |
Organism: Homo sapiens, Periplaneta americana, Diguetia canities
Method: ELECTRON MICROSCOPY
Release Date: 2023-04-12
Ligands: NAG, X80, PEE, Y01
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Bruton'S Tyrosine Kinase (Btk) With Pyridazinone Compound 9
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.39 Å Release Date: 2016-09-14 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, GOL, PG0, 6XL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-14
Ligands: SO4, GOL, PG0, 6XL
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Cdk8/Cycc In Complex With Compound 20
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.39 Å Release Date: 2016-04-20 Classification: Transferase/Transcription Ligands: 66X, FMT, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-20
Ligands: 66X, FMT, CL
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Crystal Structure Of Cdk8:Cyclin C Complex With Compound 22
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.24 Å Release Date: 2016-02-10 Classification: Transcription/Transferase/Inhibitor Ligands: EDO, FMT, 50R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-10
Ligands: EDO, FMT, 50R
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Bcl-Xl In Complex With Inhibitor (Compound 10)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2014-10-15 Classification: APOPTOSIS Ligands: 38H, EDO, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-10-15
Ligands: 38H, EDO, ACT
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Jak2 Kinase (Jh1 Domain) In Complex With The Inhibitor Trans-4-[(8As)-2-[(1R)-1-Hydroxyethyl]Imidazo[4,5-D]Pyrrolo[2,3-B]Pyridin-1(8Ah)-Yl]Cyclohexanecarbonitrile
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2013-05-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1J5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-22
Ligands: 1J5
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Jak1 Kinase (Jh1 Domain) In Complex With The Inhibitor Trans-4-{2-[(1R)-1-Hydroxyethyl]Imidazo[4,5-D]Pyrrolo[2,3-B]Pyridin-1(6H)-Yl}Cyclohexanecarbonitrile
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2013-05-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1J5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-22
Ligands: 1J5
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Jak1 Kinase (Jh1 Domain) In Complex With The Inhibitor (Trans-4-{2-[(1R)-1-Hydroxyethyl]Imidazo[4,5-D]Pyrrolo[2,3-B]Pyridin-1(6H)-Yl}Cyclohexyl)Acetonitrile
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2013-05-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1J6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-22
Ligands: 1J6
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Jak1 Kinase (Jh1 Domain) In Complex With Compound 34
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.93 Å Release Date: 2013-05-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 15T |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-22
Ligands: 15T
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Jak1 Kinase (Jh1 Domain) In Complex With Compound 72
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2012-11-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0UJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-11-07
Ligands: 0UJ
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The Jak1 Kinase Domain In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.17 Å Release Date: 2012-07-04 Classification: Transferase/Transferase Inhibitor Ligands: JAK, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-07-04
Ligands: JAK, EDO
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Jak1 Kinase (Jh1 Domain) In Complex With Compound 20
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.22 Å Release Date: 2012-07-04 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0Q2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-07-04
Ligands: 0Q2
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Discovery And Optimization Of C-2 Methyl Imidazo-Pyrrolopyridines As Potent And Orally Bioavailable Jak1 Inhibitors With Selectivity Over Jak2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.82 Å Release Date: 2012-07-04 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1RS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-07-04
Ligands: 1RS
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Discovery And Optimization Of C-2 Methyl Imidazo-Pyrrolopyridines As Potent And Orally Bioavailable Jak1 Inhibitors With Selectivity Over Jak2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2012-07-04 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: JAK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-07-04
Ligands: JAK
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Structure Of An Ml-Iap/Xiap Chimera Bound To A Peptidomimetic
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2010-03-09 Classification: APOPTOSIS Ligands: ZN, 516 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-03-09
Ligands: ZN, 516
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Structure Of An Ml-Iap/Xiap Chimera Bound To A Peptidomimetic
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2010-03-09 Classification: APOPTOSIS Ligands: ZN, 851, LI, BTB, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-03-09
Ligands: ZN, 851, LI, BTB, EDO