Search Count: 49
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Protac-Induced Ire1 Ternary Complex
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Resolution:2.60 Å Release Date: 2025-11-05 Classification: TRANSFERASE Ligands: A1BWF |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2025-11-05
Ligands: A1BWF
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Crystal Structure Of Selective Ire1A Inhibitor 29 At The Enzyme Active Site
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.43 Å Release Date: 2024-05-29 Classification: TRANSFERASE/INHIBITOR Ligands: EDO, XOE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-05-29
Ligands: EDO, XOE
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Structure Of Unphosphorylated Ire1 In Complex With G-1749
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.74 Å Release Date: 2020-12-09 Classification: TRANSFERASE Ligands: SJG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-09
Ligands: SJG
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Structure Of Unphosphorylated Ire1 In Complex With G-7658
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.61 Å Release Date: 2020-12-09 Classification: TRANSFERASE Ligands: SJM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-09
Ligands: SJM
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Structure Of Apo Unphosphorylated Ire1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.57 Å Release Date: 2020-12-09 Classification: TRANSFERASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-09
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Structure Of Phosphorylated Apo Ire1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2020-12-09 Classification: TRANSFERASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-09
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Structure Of Phosphorylated Ire1 In Complex With G-0701
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.74 Å Release Date: 2020-12-09 Classification: TRANSFERASE Ligands: SJV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-09
Ligands: SJV
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Structure Of Unphosphorylated Human Ire1 Bound To G-9807
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.08 Å Release Date: 2020-12-09 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SJS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-09
Ligands: SJS
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Pcsk9-Fab 7G7 Complex Bound To Cis-1-Amino-4-Phenylcyclohexaneacyl-Wnlk(Hr)Igllr - Nh2
Organism: Homo sapiens, Mus musculus, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.94 Å Release Date: 2020-02-05 Classification: HYDROLASE/HYDROLASE INHIBITOR/IMMUNE SYSTEM Ligands: CA |
Organism: Homo sapiens, Mus musculus, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2020-02-05
Ligands: CA
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Design Of Organo-Peptides As Bipartite Pcsk9 Antagonists
Organism: Homo sapiens, Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2020-02-05 Classification: HYDROLASE/HYDROLASE INHIBITOR/IMMUNE SYSTEM Ligands: CA |
Organism: Homo sapiens, Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2020-02-05
Ligands: CA
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Crystal Structure Of Ire1A In Complex With Compound 18
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2019-11-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: QFV, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-06
Ligands: QFV, GOL
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Taf1-Bd2 In Complex With Cpd27 (6-(But-3-En-1-Yl)-4-(1-Methyl-6-(Morpholine-4-Carbonyl)-1H-Benzo[D]Imidazol-4-Yl)-1,6-Dihydro-7H-Pyrrolo[2,3-C]Pyridin-7-One)
Organism: Oryctolagus cuniculus
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2018-11-14 Classification: Transcription/Inhibitor Ligands: G9V |
Organism: Oryctolagus cuniculus
Method: X-RAY DIFFRACTION
Release Date: 2018-11-14
Ligands: G9V
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Taf1-Bd2 In Complex With Cpd8 (6-(But-3-En-1-Yl)-4-(3-(Morpholine-4-Carbonyl)Phenyl)-1,6-Dihydro-7H-Pyrrolo[2,3-C]Pyridin-7-One)
Organism: Oryctolagus cuniculus
Method: X-RAY DIFFRACTION Resolution:1.30 Å Release Date: 2018-10-31 Classification: Transcription/Inhibitor Ligands: G9Y |
Organism: Oryctolagus cuniculus
Method: X-RAY DIFFRACTION
Release Date: 2018-10-31
Ligands: G9Y
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Crebbp Bromodomain In Complex With Cpd 4 (1-(1-(Cyclopropylmethyl)-3-(1H-Indol-4-Yl)-1,4,6,7-Tetrahydro-5H-Pyrazolo[4,3-C]Pyridin-5-Yl)Ethan-1-One)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.39 Å Release Date: 2018-08-08 Classification: PROTEIN BINDING/INHIBITOR Ligands: DMS, EDO, BKD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-08
Ligands: DMS, EDO, BKD
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E. Coli Msba In Complex With Lps And Inhibitor G907
Organism: Escherichia coli o6:h1 (strain cft073 / atcc 700928 / upec)
Method: X-RAY DIFFRACTION Resolution:2.91 Å Release Date: 2018-05-02 Classification: LIPID TRANSPORT Ligands: 3PE, AU7, FTT, PA1, PO4, DAO, MYR, DPO |
Organism: Escherichia coli o6:h1 (strain cft073 / atcc 700928 / upec)
Method: X-RAY DIFFRACTION
Release Date: 2018-05-02
Ligands: 3PE, AU7, FTT, PA1, PO4, DAO, MYR, DPO
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E. Coli Msba In Complex With Lps And Inhibitor G092
Organism: Escherichia coli o6:h1 (strain cft073 / atcc 700928 / upec)
Method: X-RAY DIFFRACTION Resolution:2.92 Å Release Date: 2018-05-02 Classification: LIPID TRANSPORT Ligands: E1M, FTT, DAO, 3PE, PO4, MYR |
Organism: Escherichia coli o6:h1 (strain cft073 / atcc 700928 / upec)
Method: X-RAY DIFFRACTION
Release Date: 2018-05-02
Ligands: E1M, FTT, DAO, 3PE, PO4, MYR
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Crebbp Bromodomain In Complex With Cpd3 ((S)-1-(3-(6-(1-Methyl-1H-Pyrazol-4-Yl)-3,4-Dihydroquinolin-1(2H)-Yl)-1-(Tetrahydrofuran-3-Yl)-1,4,6,7-Tetrahydro-5H-Pyrazolo[4,3-C]Pyridin-5-Yl)Ethan-1-One)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2018-03-07 Classification: TRANSCRIPTION REGULATOR/INHIBITOR Ligands: 9U7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-07
Ligands: 9U7
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Crebbp Bromodomain In Complex With Cpd8 (1-(3-(7-(Difluoromethyl)-6-(1-Methyl-1H-Pyrazol-4-Yl)-3,4-Dihydroquinolin-1(2H)-Yl)-1-(Tetrahydrofuran-3-Yl)-1,4,6,7-Tetrahydro-5H-Pyrazolo[4,3-C]Pyridin-5-Yl)Ethan-1-One)
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.43 Å Release Date: 2018-03-07 Classification: TRANSFERASE/INHIBITOR Ligands: 9UA, DMS, GOL |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2018-03-07
Ligands: 9UA, DMS, GOL
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Crebbp Bromodomain In Complex With Cpd10 (1-(3-(7-(Difluoromethyl)-6-(1-Methyl-1H-Pyrazol-4-Yl)-3,4-Dihydroquinolin-1(2H)-Yl)-1-(Tetrahydro-2H-Pyran-4-Yl)-1,4,6,7-Tetrahydro-5H-Pyrazolo[4,3-C]Pyridin-5-Yl)Ethan-1-One)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2018-03-07 Classification: TRANSCRIPTION REGULATOR/INHIBITOR Ligands: 9UD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-07
Ligands: 9UD
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Crebbp Bromodomain In Complex With Cpd17 (N,2,7-Trimethyl-2,3-Dihydro-4H-Benzo[B][1,4]Oxazine-4-Carboxamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2018-03-07 Classification: TRANSCRIPTION REGULATOR/INHIBITOR Ligands: SO4, 9UG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-07
Ligands: SO4, 9UG