Search Count: 13
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Crystal Structure Of Erk2 In Complex With Compound 22
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.76 Å Release Date: 2016-07-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6QB, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-07-06
Ligands: 6QB, EDO
 |
Crystal Structure Of Cdk2 In Complex With Compound 22
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2016-07-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6QB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-07-06
Ligands: 6QB
 |
Lactate Dehydrogenase A In Complex With A Trisubstituted Piperidine-2,4-Dione Inhibitor Gne-140
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2016-05-18 Classification: Oxidoreductase/Oxidoreductase Inhibitor Ligands: NAD, SO4, GN0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-18
Ligands: NAD, SO4, GN0
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Back Pocket Flexibility Provides Group-Ii Pak Selectivity For Type 1 Kinase Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2014-02-12 Classification: transferase/transferase inhibitor Ligands: 7KC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-02-12
Ligands: 7KC
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Back Pocket Flexibility Provides Group-Ii Pak Selectivity For Type 1 Kinase Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2014-02-12 Classification: transferase/transferase inhibitor Ligands: 2OL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-02-12
Ligands: 2OL
 |
Back Pocket Flexibility Provides Group-Ii Pak Selectivity For Type 1 Kinase Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2014-02-12 Classification: transferase/transferase inhibitor Ligands: 2OL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-02-12
Ligands: 2OL
 |
Back Pocket Flexibility Provides Group-Ii Pak Selectivity For Type 1 Kinase Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.48 Å Release Date: 2014-02-12 Classification: transferase/transferase inhibitor Ligands: 2OQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-02-12
Ligands: 2OQ
 |
Back Pocket Flexibility Provides Group-Ii Pak Selectivity For Type 1 Kinase Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2014-02-12 Classification: transferase/transferase inhibitor Ligands: 2OO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-02-12
Ligands: 2OO
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Discovery Of Thiazolobenzoxepin Pi3-Kinase Inhibitors That Spare The Pi3-Kinase Beta Isoform
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2013-08-28 Classification: Transferase/Transferase Inhibitor Ligands: 1JV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-08-28
Ligands: 1JV
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Crystal Structure Of Mek1 Kinase Bound To Gdc0973
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2013-08-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ANP, MG, EUI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-08-07
Ligands: ANP, MG, EUI
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Discovery Of Novel Allosteric Mek Inhibitors Possessing Classical And Non-Classical Bidentate Ser212 Interactions.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.71 Å Release Date: 2012-05-09 Classification: Transferase/Inhibitor Ligands: 3V0, ATP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-05-09
Ligands: 3V0, ATP, MG
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Discovery Of Novel Allosteric Mek Inhibitors Possessing Classical And Non-Classical Bidentate Ser212 Interactions.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2012-05-09 Classification: Transferase/Inhibitor Ligands: V04, ATP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-05-09
Ligands: V04, ATP, MG
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Crystal Structure Of C-Raf (Raf-1)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:4.00 Å Release Date: 2010-09-15 Classification: TRANSFERASE Ligands: SM5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-09-15
Ligands: SM5