Search Count: 20
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Optimization Of 3,5-Disubstitued Piperidine: Discovery Of Non-Peptide Mimetics As An Orally Active Renin Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2017-10-18 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: NAG, 7EK, PGE, PEG, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-10-18
Ligands: NAG, 7EK, PGE, PEG, DMS
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Optimization Of 3,5-Disubstitued Piperidine: Discovery Of Non-Peptide Mimetics As An Orally Active Renin Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2017-10-18 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: NAG, 7EJ, DMS, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-10-18
Ligands: NAG, 7EJ, DMS, PEG
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Discovery Of Tak-272: A Novel, Potent And Orally Active Renin In-Hibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2017-07-05 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: NAG, 6VU, PGE, PEG, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-07-05
Ligands: NAG, 6VU, PGE, PEG, DMS
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Discovery Of Tak-272: A Novel, Potent And Orally Active Renin In-Hibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.41 Å Release Date: 2016-11-16 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: NAG, 6VS, DMS, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-16
Ligands: NAG, 6VS, DMS, PEG
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Discovery Of Tak-272: A Novel, Potent And Orally Active Renin In-Hibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2016-11-02 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: NAG, 6VR, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-02
Ligands: NAG, 6VR, PEG
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Structure-Based Design Of A New Series Of N-Piperidin-3-Ylpyrimidine-5-Carboxamides As Renin Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2016-11-02 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 74U, PEG, NAG, PGE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-02
Ligands: 74U, PEG, NAG, PGE
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Structure-Based Design Of A New Series Of N-Piperidin-3-Ylpyrimidine-5-Carboxamides As Renin Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2016-11-02 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NAG, 74V, PGE, DMS, 1PE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-02
Ligands: NAG, 74V, PGE, DMS, 1PE
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Structure-Based Design Of A New Series Of N-Piperidin-3-Ylpyrimidine-5-Carboxamides As Renin Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2016-11-02 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NAG, 74Z, DMS, PEG, 1PE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-02
Ligands: NAG, 74Z, DMS, PEG, 1PE
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Structure-Based Design Of A New Series Of N-Piperidin-3-Ylpyrimidine-5-Carboxamides As Renin Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.85 Å Release Date: 2016-11-02 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NAG, 74Y, PEG, PGE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-02
Ligands: NAG, 74Y, PEG, PGE
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Novel Approach Of Fragment-Based Lead Discovery Applied To Renin Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.64 Å Release Date: 2016-10-26 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: NAG, PG6, DMS, 77O, PGE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-10-26
Ligands: NAG, PG6, DMS, 77O, PGE
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The Structure Of Rice Weevil Pectin Methyl Esterase
Organism: Sitophilus oryzae
Method: X-RAY DIFFRACTION Resolution:1.79 Å Release Date: 2014-11-12 Classification: HYDROLASE |
Organism: Sitophilus oryzae
Method: X-RAY DIFFRACTION
Release Date: 2014-11-12
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Crystal Structure Of Faah In Complex With Inhibitor
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:2.91 Å Release Date: 2013-02-06 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 17J |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2013-02-06
Ligands: 17J
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Human Carbonic Anhydrase Ii With A Sulfonamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:0.90 Å Release Date: 2010-05-12 Classification: LYASE/LYASE INHIBITOR Ligands: HGB, ZN, SUA, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-05-12
Ligands: HGB, ZN, SUA, GOL
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Full Matrix Error Analysis Of Carbonic Anhydrase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:0.95 Å Release Date: 2003-09-09 Classification: LYASE Ligands: ZN, HG, MBO, SUA, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2003-09-09
Ligands: ZN, HG, MBO, SUA, GOL
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Human Dna Topoisomerase I In Covalent Complex With A 22 Base Pair Dna Duplex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.20 Å Release Date: 2002-12-04 Classification: ISOMERASE/DNA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2002-12-04
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Human Dna Topoisomerase I (70 Kda) In Complex With The Poison Topotecan And Covalent Complex With A 22 Base Pair Dna Duplex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2002-12-04 Classification: ISOMERASE/DNA Ligands: TTG, TTC, HG, PG4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2002-12-04
Ligands: TTG, TTC, HG, PG4
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Crystal Structure Of Bovine Rhodopsin
Organism: Bos taurus
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2001-07-04 Classification: SIGNALING PROTEIN Ligands: BNG, HG, ZN, PLM, RET, HTO |
Organism: Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2001-07-04
Ligands: BNG, HG, ZN, PLM, RET, HTO
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Crystal Structure Of Bovine Rhodopsin
Organism: Bos taurus
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2000-08-04 Classification: SIGNALING PROTEIN Ligands: HG, ZN, RET |
Organism: Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2000-08-04
Ligands: HG, ZN, RET
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Bifunctional Hageman Factor/Amylase Inhibitor From Maize
Organism: Zea mays
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 1998-08-12 Classification: SERINE PROTEASE INHIBITOR |
Organism: Zea mays
Method: X-RAY DIFFRACTION
Release Date: 1998-08-12
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Recombinant Bifunctional Hageman Factor/Amylase Inhibitor From Maize
Organism: Zea mays
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 1998-08-12 Classification: SERINE PROTEASE INHIBITOR |
Organism: Zea mays
Method: X-RAY DIFFRACTION
Release Date: 1998-08-12