Search Count: 11
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6-Phenyl-1H-Imidazo[4,5-C]Pyridine-4-Carbonitrile As Cathepsin S Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2011-04-06 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: EF3, DMS, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-04-06
Ligands: EF3, DMS, SO4
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Cathepsin K Covalently Bound To A Cyano-Pyrimidine Inhibitor With Improved Selectivity Over Herg
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2011-03-30 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: O47 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-30
Ligands: O47
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Cathepsin S In Complex With A Covalent Inhibitor With An Aldehyde Warhead
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.49 Å Release Date: 2010-12-22 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: O64, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-12-22
Ligands: O64, DMS
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Cathepsin K In Complex With A Covalent Inhibitor With A Ketoamide Warhead
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.02 Å Release Date: 2010-12-22 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: O96, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-12-22
Ligands: O96, SO4
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Cathepsin K Covalently Bound To A 2-Cyano Pyrimidine Inhibitor With A Benzyl P3 Group.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2010-10-06 Classification: HYDROLASE Ligands: SO4, O75 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-10-06
Ligands: SO4, O75
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An Orally Active Inhibitor Bound At The Active Site Of Hpgds
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2010-09-01 Classification: ISOMERASE Ligands: GSH, KXO, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-09-01
Ligands: GSH, KXO, MG
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4-(3-Trifluoromethylphenyl)-Pyrimidine-2-Carbonitrile As Cathepsin S Inhibitors: N3, Not N1 Is Critically Important
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2010-07-14 Classification: HYDROLASE Ligands: PEG, DMS, 935, 93N, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-07-14
Ligands: PEG, DMS, 935, 93N, SO4, GOL
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X-Ray Structure Of Cathepsin K Covalently Bound To A Triazine Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2010-03-02 Classification: HYDROLASE Ligands: ORG, TFA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-03-02
Ligands: ORG, TFA
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Cathepsin K In Complex With A Non-Selective 2-Cyano-Pyrimidine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.49 Å Release Date: 2010-03-02 Classification: HYDROLASE Ligands: SO4, KWZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-03-02
Ligands: SO4, KWZ
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Cathepsin K In Complex With A Selective 2-Cyano-Pyrimidine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.51 Å Release Date: 2010-03-02 Classification: HYDROLASE Ligands: KX1, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-03-02
Ligands: KX1, SO4
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Alpha-Hemolysin From Staphylococcus Aureus
Organism: Staphylococcus aureus
Method: X-RAY DIFFRACTION Resolution:1.89 Å Release Date: 1998-01-14 Classification: CYTOLYTIC PROTEIN |
Organism: Staphylococcus aureus
Method: X-RAY DIFFRACTION
Release Date: 1998-01-14
