Search Count: 62
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Crystal Structure Of Bace1 In Complex With (Z)-Fluoro-Olefin Containing Compound 15
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.86 Å Release Date: 2020-06-03 Classification: HYDROLASE/HYDROLASE Inhibitor Ligands: U64, IOD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-06-03
Ligands: U64, IOD
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Crystal Structure Of Human Kras G12C Covalently Bound To A Phthalazine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2019-12-25 Classification: SIGNALING PROTEIN/Inhibitor Ligands: MG, GDP, OJ1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-25
Ligands: MG, GDP, OJ1
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Crystal Structure Of Human Kras G12C Covalently Bound To A Quinazolinone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2019-12-25 Classification: SIGNALING PROTEIN/Inhibitor Ligands: GDP, CA, OHY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-25
Ligands: GDP, CA, OHY
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Co-Crystal Structure Of Bace With Inhibitor Am-6494
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2019-10-23 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: IOD, GOL, P6J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-10-23
Ligands: IOD, GOL, P6J
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Crystal Structure Of Human Kras G12C Covalently Bound To An Acryloylazetidine Acetamide Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2019-08-28 Classification: SIGNALING PROTEIN/Inhibitor Ligands: CA, GDP, O67 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-08-28
Ligands: CA, GDP, O67
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Crystal Structure Of Human Kras G12C Covalently Bound To An Acryloylazetidine Acetamide Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.11 Å Release Date: 2019-08-28 Classification: SIGNALING PROTEIN/Inhibitor Ligands: CA, GDP, O5V |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-08-28
Ligands: CA, GDP, O5V
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Crystal Structure Of Human Kras G12C Covalently Bound To An Acryloylazetidine Acetamide Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.31 Å Release Date: 2019-08-28 Classification: SIGNALING PROTEIN/Inhibitor Ligands: MG, GDP, O5Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-08-28
Ligands: MG, GDP, O5Y
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Crystal Structure Of Human Kras G12C Covalently Bound To An Acryloylazetidine Acetamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2019-08-28 Classification: SIGNALING PROTEIN/Inhibitor Ligands: CA, GDP, O5S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-08-28
Ligands: CA, GDP, O5S
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Crystal Structure Of Rat Cathepsin D With (5S)-3-(5,6-Dihydro-2H-Pyran-3-Yl)-1-Fluoro- 7-(2-Fluoropyridin-3-Yl)Spiro[Chromeno[2,3- C]Pyridine-5,4'-[1,3]Oxazol]-2'-Amine
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:2.81 Å Release Date: 2018-06-13 Classification: HYDROLASE Ligands: NAG, 3UT |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2018-06-13
Ligands: NAG, 3UT
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Structure Of Bace-1 (Beta-Secretase) In Complex With : N-(3-((1R,5S,6R)-3-Amino-5-Methyl-2-Oxa-4-Azabicyclo[4.1.0]Hept-3-En-5-Yl)-4-Fluorophenyl)-5-Methoxypyrazine-2-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2018-02-21 Classification: Hydrolase/Hydrolase Inhibitor Ligands: IOD, GOL, SO4, EJ7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-02-21
Ligands: IOD, GOL, SO4, EJ7
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Crystal Structure Of Bace1 In Complex With 2-Aminooxazoline-3-Azaxanthene Compound 12
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2017-05-17 Classification: HYDROLASE Ligands: IOD, 8QV, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-17
Ligands: IOD, 8QV, GOL
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Crystal Structure Of Bace1 In Complex With Aminoquinoline Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.62 Å Release Date: 2016-03-30 Classification: Hydrolase/Hydrolase Inhibitor Ligands: IOD, 68M, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-03-30
Ligands: IOD, 68M, GOL
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Crystal Structure Of Bace1 In Complex With 2-Aminooxazoline-3-Azaxanthene Inhibitor 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2016-03-30 Classification: Hydrolase/Hydrolase Inhibitor Ligands: IOD, GOL, SO4, 68L |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-03-30
Ligands: IOD, GOL, SO4, 68L
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Crystal Structure Of Bace1 In Complex With Aminoquinoline Inhibitor 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2016-03-30 Classification: HYDROLASE/HYDROLASE Inhibitor Ligands: 68J, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-03-30
Ligands: 68J, GOL
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Crystal Structure Of Bace1 In Complex With Aminoquinoline Inhibitor 9
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2016-03-30 Classification: HYDROLASE/HYDROLASE Inhibitor Ligands: 68K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-03-30
Ligands: 68K
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Crystal Structure Of Bace1 In Complex With 3-(2-Amino-6-(O-Tolyl)Quinolin-3-Yl)-N-(3,3-Dimethylbutyl)Propanamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2016-03-30 Classification: HYDROLASE Ligands: IOD, GOL, 6BS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-03-30
Ligands: IOD, GOL, 6BS
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Human Gkrp Bound To Amg2882 And Sorbitol-6-Phosphate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2015-05-13 Classification: sugar binding protein/inhibitor Ligands: 2WY, S6P, IOD, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-05-13
Ligands: 2WY, S6P, IOD, GOL, SO4
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Human Gkrp Bound To Amg-3295 And Sorbitol-6-Phosphate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.43 Å Release Date: 2015-05-13 Classification: sugar binding protein/inhibitor Ligands: 2WX, S6P, IOD, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-05-13
Ligands: 2WX, S6P, IOD, GOL, SO4
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Human Gkrp Bound To Amg-0696 And Sorbitol-6-Phosphate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2015-05-13 Classification: sugar binding protein/inhibitor Ligands: 2WZ, S6P, IOD, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-05-13
Ligands: 2WZ, S6P, IOD, GOL, SO4
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Human Gkrp Bound To Amg-0265 (N-[(R)-(2-Chlorophenyl){7-[4-(2-Hydroxypropan-2-Yl) Pyridin-2-Yl]-1-Benzothiophen-2-Yl}Methyl]Cyclopropanesulfonamide) And Sorbitol-6-Phosphate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2015-03-18 Classification: transferase/transferase inhibitor Ligands: 2Y6, S6P, IOD, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-03-18
Ligands: 2Y6, S6P, IOD, GOL, SO4