Search Count: 17
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Braf In Complex With N-(4-Methyl-3-(1-Methyl-2-Oxo-2,3-Dihydro-1H-Benzo[D]Imidazol-5-Yl)Phenyl)-3-(Trifluoromethyl)Benzamide.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.04 Å Release Date: 2019-10-23 Classification: transferase/transferase inhibitor Ligands: K7S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-10-23
Ligands: K7S
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Braf In Complex With N-(3-(2-(2-Hydroxyethoxy)-6-Morpholinopyridin-4-Yl)-4-Methylphenyl)-2-(Trifluoromethyl)Isonicotinamide (Lxh254)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.37 Å Release Date: 2019-09-04 Classification: transferase/transferase inhibitor Ligands: K81 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-09-04
Ligands: K81
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Monophosphorylated Pser33 B-Catenin Peptide, B-Trcp/Skp1, Nrx-2776 Ternary Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2019-04-03 Classification: LIGASE Ligands: J91, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-04-03
Ligands: J91, PO4
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Monophosphorylated Pser33 B-Catenin Peptide, B-Trcp/Skp1, Nrx-103094 Ternary Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2019-04-03 Classification: LIGASE Ligands: J97, PO4, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-04-03
Ligands: J97, PO4, CL
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Monophosphorylated Pser33 B-Catenin Peptide, B-Trcp/Skp1, Nrx-2663 Ternary Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2019-04-03 Classification: LIGASE Ligands: J8V, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-04-03
Ligands: J8V, PO4
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Monophosphorylated Pser33 B-Catenin Peptide, B-Trcp/Skp1, Nrx-1933 Ternary Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2019-04-03 Classification: LIGASE Ligands: J8Y, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-04-03
Ligands: J8Y, PO4
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Monophosphorylated Pser33 B-Catenin Peptide Bound To B-Trcp/Skp1 Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2019-04-03 Classification: LIGASE Ligands: PO4, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-04-03
Ligands: PO4, DMS
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Braf In Complex With N-(3-(Tert-Butyl)Phenyl)-4-Methyl-3-(6-Morpholinopyrimidin-4-Yl)Benzamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.26 Å Release Date: 2017-06-28 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: 92D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-28
Ligands: 92D
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Braf In Complex With Raf709
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2017-06-28 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: 92J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-28
Ligands: 92J
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The Co-Structure Of (R)-4-(6-(1-(Cyclopropylsulfonyl)Cyclopropyl)-2-(1H-Indol-4-Yl)Pyrimidin-4-Yl)-3-Methylmorpholine And A Rationally Designed Pi3K-Alpha Mutant That Mimics Atr
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2017-06-14 Classification: TRANSFERASE/SIGNALING PROTEIN/INHIBITOR Ligands: 8DV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-14
Ligands: 8DV
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The Co-Structure Of N,N-Dimethyl-4-[(6R)-6-Methyl-5-(1H-Pyrrolo[2,3- B]Pyridin-4-Yl)-4,5,6,7-Tetrahydropyrazolo[1,5- A]Pyrazin-3-Yl]Benzenesulfonamide And A Rationally Designed Pi3K-Alpha Mutant That Mimics Atr
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2017-05-10 Classification: TRANSFERASE/SIGNALING PROTEIN/INHIBITOR Ligands: 3K6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-10
Ligands: 3K6
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The Co-Structure Of 3-Amino-6-(4-((1-(Dimethylamino)Propan-2-Yl)Sulfonyl)Phenyl)-N-Phenylpyrazine-2-Carboxamide And A Rationally Designed Pi3K-Alpha Mutant That Mimics Atr
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2017-05-10 Classification: TRANSFERASE/SIGNALING PROTEIN/INHIBITOR Ligands: 8DY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-10
Ligands: 8DY
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Crystal Structure Of A Novel Tetrahydropyrazolo[1,5-A]Pyrazine In An Engineered Pi3K Alpha
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.39 Å Release Date: 2014-12-31 Classification: transferase/transferase inhibitor Ligands: 3K6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-31
Ligands: 3K6
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Crystal Structure Of Hsp90-Alpha N-Domain Bound To The Inhibitor Nvp-Hsp990
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2014-11-26 Classification: CHAPERONE/INHIBITOR Ligands: 3JC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-11-26
Ligands: 3JC
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Crystal Structure Of Hsp90-Alpha N-Domain Bound To The Inhibitor Nvp-Hsp990
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2014-11-19 Classification: CHAPERONE Ligands: 990 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-11-19
Ligands: 990
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Co-Crystal Structure Of The Human Kinesin Eg5 With A Novel Tetrahydro-Beta-Carboline
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2009-12-15 Classification: MOTOR PROTEIN Ligands: MG, ADP, L31, NO3, CL, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-12-15
Ligands: MG, ADP, L31, NO3, CL, PEG
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4-(Aminoalkylamino)-3-Benzimidazole-Quinolinones As Potent Chk1 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2007-03-20 Classification: TRANSFERASE Ligands: SO4, 12C |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-03-20
Ligands: SO4, 12C