Search Count: 19
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Crystal Structure Of Parp1 Catalytic Domain Bound To Azd5305 (Saruparib)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.59 Å Release Date: 2024-12-04 Classification: TRANSFERASE Ligands: A1H63, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-04
Ligands: A1H63, SO4
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Crystal Structure Of Parp1 Catalytic Domain Bound To Azd9574
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.82 Å Release Date: 2024-12-04 Classification: TRANSFERASE Ligands: A1H64, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-04
Ligands: A1H64, SO4
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Krasg12C Ligand Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2023-07-12 Classification: SIGNALING PROTEIN Ligands: MG, GDP, PQI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-07-12
Ligands: MG, GDP, PQI
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Krasg12C Ligand Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.11 Å Release Date: 2023-07-12 Classification: SIGNALING PROTEIN Ligands: MG, GDP, PUO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-07-12
Ligands: MG, GDP, PUO
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Crystal Structure Of Pi3Kgamma With A Dihydropurinone Inhibitor (Compound 18)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.74 Å Release Date: 2022-07-13 Classification: SIGNALING PROTEIN Ligands: IGJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-07-13
Ligands: IGJ
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Parp1 Catalytic Domain In Complex With 8-Chloroquinazolinone-Based Inhibitor (Compound 9)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2021-09-15 Classification: TRANSFERASE Ligands: VKW, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-15
Ligands: VKW, SO4
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Parp1 Catalytic Domain In Complex With Isoquinolone-Based Inhibitor (Compound 16)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2021-09-15 Classification: TRANSFERASE Ligands: VKT, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-15
Ligands: VKT, SO4
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Parp1 Catalytic Domain In Complex With A Selective Pyridine Carboxamide-Based Inhibitor (Compound 22)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2021-09-15 Classification: TRANSFERASE Ligands: VKQ, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-15
Ligands: VKQ, SO4
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Crystal Structure Of The Kinase Domain Of Human C-Kit In Complex With A Type-Ii Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.38 Å Release Date: 2020-05-27 Classification: SIGNALING PROTEIN Ligands: O35 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-05-27
Ligands: O35
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Crystal Structure Of The Kinase Domain Of Human C-Kit In Complex With A Type-Ii Inhibitor Bearing An Acrylamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2020-05-27 Classification: SIGNALING PROTEIN Ligands: O2K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-05-27
Ligands: O2K
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Crystal Structure Of The Kinase Domain Of Human C-Kit With A Cyclic Imidate Inhibitor Covalently Bound To Cys788
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2020-05-27 Classification: SIGNALING PROTEIN Ligands: O2H |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-05-27
Ligands: O2H
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Crystal Structure Of The Kdr (Vegfr2) Kinase Domain In Complex With A Type-Ii Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.78 Å Release Date: 2020-05-27 Classification: SIGNALING PROTEIN Ligands: O35 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-05-27
Ligands: O35
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Crystal Structure Of The Kdr (Vegfr2) Kinase Domain In Complex With A Type-Ii Inhibitor Bearing An Acrylamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2020-05-27 Classification: SIGNALING PROTEIN Ligands: O3E |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-05-27
Ligands: O3E
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Crystal Structure Of The Csf1R Kinase Domain With A Dihydropurinone Inhibitor (Compound 4)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2020-01-01 Classification: TRANSFERASE Ligands: M9T, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-01
Ligands: M9T, SO4
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Crystal Structure Of Pi3Kgamma With A Dihydropurinone Inhibitor (Compound 4)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.01 Å Release Date: 2020-01-01 Classification: TRANSFERASE Ligands: M9T |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-01
Ligands: M9T
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Crystal Structure Of Pi3Kgamma In Complex With Dna-Pk Inhibitor Azd7648
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.62 Å Release Date: 2020-01-01 Classification: TRANSFERASE Ligands: MBW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-01
Ligands: MBW
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Mmp9-Inhibitor Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2002-05-16 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: CA, NFH, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2002-05-16
Ligands: CA, NFH, ZN
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Mmp9 Active Site Mutant-Inhibitor Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2002-05-16 Classification: HYDROLASE Ligands: CA, STN, BUM, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2002-05-16
Ligands: CA, STN, BUM, ZN
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Phosphatidylinositol 3-Kinase, P85-Alpha Subunit: C-Terminal Sh2 Domain Complexed With A Tyr751 Phosphopeptide From The Pdgf Receptor, Nmr, Minimized Mean Structure
Organism: Homo sapiens
Method: SOLUTION NMR Release Date: 1997-09-17 Classification: COMPLEX (PHOSPHOTRANSFERASE/RECEPTOR) |
Organism: Homo sapiens
Method: SOLUTION NMR
Release Date: 1997-09-17
