Search Count: 19
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C-Terminal Bromodomain Of Human Brd2 With 5-(1-Benzyl-4-Chloro-1H-Imidazol-2-Yl)-1,3-Dimethylpyridin-2(1H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2024-06-26 Classification: TRANSCRIPTION Ligands: EDO, PE4, A1IBV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-06-26
Ligands: EDO, PE4, A1IBV
 |
N-Terminal Bromodomain Of Human Brd4 With (5-(4-Chloro-1-((Tetrahydro-2H-Pyran-4-Yl)Methyl)-1H-Imidazol-2-Yl)-1,3-Dimethylpyridin-2(1H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2024-06-26 Classification: TRANSCRIPTION Ligands: EDO, A1IB5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-06-26
Ligands: EDO, A1IB5
 |
N-Terminal Bromodomain Of Human Brd4 With Gsk789
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.62 Å Release Date: 2020-07-29 Classification: TRANSCRIPTION Ligands: QAN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-29
Ligands: QAN
 |
N-Terminal Bromodomain Of Human Brd4 (3R,4R)-N-Cyclohexyl-4-((3-Methyl-2-Oxo-1,2-Dihydro-1,7-Naphthyridin-8-Yl)Amino)Piperidine-3-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.26 Å Release Date: 2020-07-29 Classification: TRANSCRIPTION Ligands: QAZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-29
Ligands: QAZ
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Crystal Structure Of Human Atad2 Bromodomain In Complex With N-(4-Bromo-3-(3-Methylpyrrolidin-1-Yl)Sulfonyl)Phenyl)-2-(-4-Cyclopropyl-4-Methyl-2,5-Dioxoimidazolidin-1-Yl)Acetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2020-05-06 Classification: TRANSCRIPTION Ligands: SO4, EDO, OJH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-05-06
Ligands: SO4, EDO, OJH
 |
N-Terminal Bromodomain Of Human Brd2 With 5-(4-(4-Fluorophenyl)-1H-Imidazol-5-Yl)-1-Methylpyridin-2(1H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.26 Å Release Date: 2020-02-19 Classification: TRANSCRIPTION Ligands: SO4, NUQ, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-02-19
Ligands: SO4, NUQ, EDO
 |
N-Terminal Bromodomain Of Human Brd4 With 1-((1-Acetylpiperidin-4-Yl)Methyl)-2-(4-Hydroxy-3,5-Dimethylphenyl)-N-Methyl-1H-Benzo[D]Imidazole-5-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.48 Å Release Date: 2020-01-15 Classification: TRANSCRIPTION Ligands: NUW, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-15
Ligands: NUW, EDO
 |
N-Terminal Bromodomain Of Human Brd4 With 1,3-Dimethyl-5-(1-((Tetrahydro-2H-Pyran-4-Yl)Methyl)-1H-Benzo[D]Imidazol-2-Yl)Pyridin-2(1H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2020-01-15 Classification: TRANSCRIPTION Ligands: EDO, NUB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-15
Ligands: EDO, NUB
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N-Terminal Bromodomain Of Human Brd4 With 5-(1-(1,3-Dimethoxypropan-2-Yl)-5-Morpholino-1H-Benzo[D]Imidazol-2-Yl)-1,3-Dimethylpyridin-2(1H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.30 Å Release Date: 2020-01-15 Classification: TRANSCRIPTION Ligands: EDO, NV2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-15
Ligands: EDO, NV2
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N-Terminal Bromodomain Of Human Brd4 With 5-(1-(1,3-Dimethoxypropan-2-Yl)-5-Morpholino-1H-Benzo[D]Imidazol-2-Yl)-1,3-Dimethylpyridin-2(1H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2020-01-15 Classification: TRANSCRIPTION Ligands: SO4, NUH, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-15
Ligands: SO4, NUH, EDO
 |
Crystal Structure Of Human Atad2 Bromodomain In Complex With 3-Methyl-8-((8-Methyl-8-Azabicyclooctan-3-Yl)Amino)-1,7-Naphthyridin-2(1H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2018-09-26 Classification: TRANSCRIPTION Ligands: SO4, EDO, FZB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-09-26
Ligands: SO4, EDO, FZB
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Crystal Structure Of Human Atad2 Bromodomain In Complex With 8-(((1R,2R,3R,5S)-2-(2-(1,1-Dioxidotetrahydro-2H-Thiopyran-4-Yl)Ethyl)-8-Azabicyclo[3.2.1]Octan-3-Yl)Amino)-3-Methyl-5-(5-Methylpyridin-3-Yl)Quinolin-2(1H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.61 Å Release Date: 2018-09-26 Classification: TRANSCRIPTION Ligands: EDO, FZH, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-09-26
Ligands: EDO, FZH, SO4
 |
N-Terminal Bromodomain Of Human Brd4 With : 8-(((1R,2R,3R,5S)-2-(2-(4,4-Difluorocyclohexyl)Ethyl)-8-Azabicyclo[3.2.1]Octan-3-Yl)Amino)-3-Methyl-5-(5-Methylpyridin-3-Yl)-1,7-Naphthyridin-2(1H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2018-09-26 Classification: TRANSCRIPTION Ligands: EDO, FZE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-09-26
Ligands: EDO, FZE
 |
Bromodomain Of Human Brpf1 With N-1,3-Dimethyl-6-2R-2- Methylpiperazin-1-Yl-2-Oxo-2,3-Dihydro-1H-1,3-Benzodiazol-5-Yl-2- Methoxybenzamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.96 Å Release Date: 2016-07-06 Classification: TRANSCRIPTION Ligands: LF1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-07-06
Ligands: LF1
 |
Bromodomain Of Human Brpf1 With N-1,3-Dimethyl-6-2R-2- Methylpiperazin-1-Yl-2-Oxo-2,3-Dihydro-1H-1,3-Benzodiazol-5-Yl-N- Ethyl-2-Methoxybenzamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2016-07-06 Classification: TRANSCRIPTION Ligands: 8VI, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-07-06
Ligands: 8VI, EDO
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Crystal Structure Of Human Atad2 Bromodomain In Complex With 8-(3R,4R) -3-(Cyclohexylmethoxy)Piperidin-4-Yl-Amino-3-Methyl-1,2-Dihydro-1,7- Naphthyridin-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.03 Å Release Date: 2015-08-12 Classification: HYDROLASE Ligands: EDO, 78J, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-12
Ligands: EDO, 78J, SO4
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Crystal Structure Of Human Atad2 Bromodomain In Complex With 4-(3R,4R) -4-(3-Methyl-2-Oxo-1,2-Dihydro-1,7-Naphthyridin-8-Yl)Aminopiperidin-3- Yloxymethyl)-1-Thiane-1,1-Dione
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.86 Å Release Date: 2015-08-12 Classification: INHIBITOR Ligands: EDO, YEJ, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-12
Ligands: EDO, YEJ, SO4
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Crystal Structure Of Human Atad2 Bromodomain In Complex With 4-((3R, 4R)-4-3-Methyl-5-(5-Methylpyridin-3-Yl)-2-Oxo-1,2-Dihydroquinolin-8- Yl-Aminopiperidin-3-Yloxymethyl)-1-Thiane-1,1-Dione
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.09 Å Release Date: 2015-08-12 Classification: HYDROLASE Ligands: EDO, YD3, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-12
Ligands: EDO, YD3, SO4
 |
N-Terminal Bromodomain Of Human Brd4 With 8-(3R,4R)-3-(Cyclohexylmethoxy)Piperidin-4-Ylamino-3-Methyl-1,2-Dihydro-1,7- Naphthyridin-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2015-08-12 Classification: HYDROLASE Ligands: EDO, 78J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-12
Ligands: EDO, 78J