Search Count: 18
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Discovery Of An Anion-Dependent Farnesyltransferase Inhibitor From A Phenotypic Screen
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:2.28 Å Release Date: 2021-09-08 Classification: TRANSFERASE/INHIBITOR Ligands: ACE, 60I, ZN, MG, PPV |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2021-09-08
Ligands: ACE, 60I, ZN, MG, PPV
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Discovery Of An Anion-Dependent Farnesyltransferase Inhibitor From A Phenotypic Screen
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2021-09-08 Classification: TRANSFERASE/INHIBITOR Ligands: ACE, 60I, ZN, MG, DMA |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2021-09-08
Ligands: ACE, 60I, ZN, MG, DMA
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Structure Of Human Hdac2 In Complex With An Ethyl Ketone Inhibitor Containing A Spiro-Bicyclic Group (Compound 22)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.63 Å Release Date: 2021-08-11 Classification: HYDROLASE Ligands: ZN, SO4, CA, PEG, VJV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-08-11
Ligands: ZN, SO4, CA, PEG, VJV
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Structure Of Hdac2 In Complex With A Macrocyclic Inhibitor (Compound 4)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2021-07-14 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, SO4, CA, PEG, ZLV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-14
Ligands: ZN, SO4, CA, PEG, ZLV
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Structure Of Hdac2 In Complex With An Inhibitor (Compound 9)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.54 Å Release Date: 2021-07-14 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, SO4, CA, PEG, V1P |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-14
Ligands: ZN, SO4, CA, PEG, V1P
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Structure Of Hdac2 In Complex With An Inhibitor (Compound 14)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.69 Å Release Date: 2021-07-14 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, SO4, CA, PEG, ZLS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-14
Ligands: ZN, SO4, CA, PEG, ZLS
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Structure Of Hdac2 In Complex With An Inhibitor (Compound 19)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.78 Å Release Date: 2021-07-14 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, SO4, CA, PEG, ZLM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-14
Ligands: ZN, SO4, CA, PEG, ZLM
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Structure Of Hdac2 In Complex With A Macrocyclic Inhibitor (Compound 25)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.54 Å Release Date: 2021-07-14 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, SO4, CA, PEG, ZL4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-14
Ligands: ZN, SO4, CA, PEG, ZL4
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Structure Of Human Hdac2 In Complex With Apicidin
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2021-05-05 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, CA, PEG, YED |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-05
Ligands: ZN, CA, PEG, YED
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Structure Of Human Hdac2 In Complex With An Inhibitor That Lacks A Zinc Binding Group (Compound 12)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.59 Å Release Date: 2021-05-05 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, CA, ACT, PEG, YEM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-05
Ligands: ZN, CA, ACT, PEG, YEM
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Structure Of Human Hdac2 In Complex With An Inhibitor Lacking A Zinc Binding Group (Compound 19)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.49 Å Release Date: 2021-05-05 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, SO4, CA, ACT, PEG, YEV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-05
Ligands: ZN, SO4, CA, ACT, PEG, YEV
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Structure Of Human Hdac2 In Complex With A 2-Substituted Benzamide Inhibitor (Compound 20)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.26 Å Release Date: 2020-12-30 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, CA, SO4, PEG, WBA, DMS, WBD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-30
Ligands: ZN, CA, SO4, PEG, WBA, DMS, WBD
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Structure Of Human Hdac2 In Complex With A 2-Substituted Benzamide Inhibitor (Compound 16)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.68 Å Release Date: 2020-12-30 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, CA, PEG, WB4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-30
Ligands: ZN, CA, PEG, WB4
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Structure Of Human Hdac2 In Complex With Ketone Inhibitor (Compound E)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2020-08-12 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, SO4, CA, PEG, V1P |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-08-12
Ligands: ZN, SO4, CA, PEG, V1P
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Structure Of Human Hdac2 In Complex With Ketone Inhibitor (Compound O)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2020-08-12 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, SO4, CA, PEG, V1S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-08-12
Ligands: ZN, SO4, CA, PEG, V1S
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Structure Of Human Hdac2 In Complex With An Aryl Ketone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.56 Å Release Date: 2020-07-29 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, CA, SO4, PEG, V1D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-29
Ligands: ZN, CA, SO4, PEG, V1D
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Structure Of Human Hdac2 In Complex With An Ethyl Ketone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.46 Å Release Date: 2020-05-06 Classification: HYDROLASE/HYDROLASE Inhibitor Ligands: TV1, ZN, CA, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-05-06
Ligands: TV1, ZN, CA, PEG
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Structure Of Human Hdac2 In Complex With An Ethyl Ketone Inhibitor Containing A Spiro-Bicyclic Group
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.32 Å Release Date: 2020-05-06 Classification: HYDROLASE/HYDROLASE Inhibitor Ligands: ZN, SO4, CA, PEG, TV7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-05-06
Ligands: ZN, SO4, CA, PEG, TV7