Search Count: 16
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Crystal Structure Of An Allosteric Inhibitor Bound To Human Ripk1 Kinase Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.98 Å Release Date: 2025-12-24 Classification: IMMUNE SYSTEM Ligands: A1IX7, IOD, 1HX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-12-24
Ligands: A1IX7, IOD, 1HX
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Crystal Structure Of An Allosteric Inhibitor Bound To Human Ripk1 Kinase Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.29 Å Release Date: 2025-12-24 Classification: IMMUNE SYSTEM Ligands: A1IX9, IOD, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-12-24
Ligands: A1IX9, IOD, PEG
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Crystal Structure Of Trim24 Phd-Bromodomain Complexed With 1-Methyl-5-(2-Methyl-1 3-Thiazol-4-Yl)-2 3-Dihydro-1H-Indol-2-One (1)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2015-06-24 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: ZN, 4CN, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-24
Ligands: ZN, 4CN, SO4
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Crystal Structure Of Trim24 Phd-Bromodomain Complexed With 2,4-Dimethoxy-N-(1-Methyl-2-Oxo-1,2,3,4-Tetrahydroquinolin-6-Yl)Benzene-1-Sulfonamide (3B)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.73 Å Release Date: 2015-06-24 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: ZN, 4A7, GOL, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-24
Ligands: ZN, 4A7, GOL, CL
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Crystal Structure Of Trim24 Phd-Bromodomain Complexed With N-(1,3-Dimethyl-2-Oxo-2,3-Dihydro-1H-1,3-Benzodiazol-5-Yl)-4-Methoxybenzene-1-Sulfonamide (5B)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.18 Å Release Date: 2015-06-24 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: ZN, 4A8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-24
Ligands: ZN, 4A8
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Crystal Structure Of Trim24 Phd-Bromodomain Complexed With N-[6-(4-Methoxyphenoxy)-1,3-Dimethyl-2-Oxo-2,3-Dihydro-1H-1,3-Benzodiazol-5-Yl]Benzenesulfonamide (5G)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2015-06-24 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: 4AE, ZN, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-24
Ligands: 4AE, ZN, GOL, SO4
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Crystal Structure Of Trim24 Phd-Bromodomain Complexed With N-{6-[3-(Benzyloxy)Phenoxy]-1,3-Dimethyl-2-Oxo-2,3-Dihydro-1H-1,3-Benzodiazol-5-Yl}-3,4-Dimethoxybenzene-1-Sulfonamide (7B)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.46 Å Release Date: 2015-06-24 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: ZN, GOL, 4BJ, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-24
Ligands: ZN, GOL, 4BJ, SO4
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Crystal Structure Of Trim24 Phd-Bromodomain Complexed With N-{1,3-Dimethyl-6-[3-(2-Methylpropoxy)Phenoxy]-2-Oxo-2,3-Dihydro-1H-1,3-Benzodiazol-5-Yl}-1,2-Dimethyl-1H-Imidazole-4-Sulfonamide (7G)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2015-06-24 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: ZN, 4BK, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-24
Ligands: ZN, 4BK, DMS
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Crystal Structure Of Trim24 Phd-Bromodomain Complexed With N-{1,3-Dimethyl-2-Oxo-6-[3-(Oxolan-3-Ylmethoxy)Phenoxy]-2,3-Dihydro-1H-1,3-Benzodiazol-5-Yl}-1-Methyl-1H-Imidazole-4-Sulfonamide (7L)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.82 Å Release Date: 2015-06-24 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: ZN, DMS, 4BV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-24
Ligands: ZN, DMS, 4BV
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Crystal Structure Of Trim24 Phd-Bromodomain Complexed With N-(6-{3-[4-(Dimethylamino)Butoxy]-5-Propoxyphenoxy}-1,3-Dimethyl-2-Oxo-2,3-Dihydro-1H-1,3-Benzodiazol-5-Yl)-3,4-Dimethoxybenzene-1-Sulfonamide (8I)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.82 Å Release Date: 2015-06-24 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: ZN, GOL, 4C1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-24
Ligands: ZN, GOL, 4C1
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Crystal Structure Of Atad2A Bromodomain Complexed With H4(1-20)K5Ac Peptide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2014-12-24 Classification: GENE REGULATION |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-24
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Crystal Structure Of Atad2A Bromodomain Complexed With H3(1-21)K14Ac Peptide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2014-12-24 Classification: GENE REGULATION Ligands: SO4, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-24
Ligands: SO4, CL
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Crystal Structure Of Atad2A Bromodomain Double Mutant N1063A-Y1064A In Apo Form
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2014-12-24 Classification: GENE REGULATION Ligands: SO4, CL, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-24
Ligands: SO4, CL, GOL
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Crystal Structure Of Atad2A Bromodomain Complexed With Methyl 3-Amino-5-(3,5-Dimethyl-1,2-Oxazol-4-Yl)Benzoate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2014-12-24 Classification: GENE REGULATION Ligands: SO4, CL, GOL, 36Z |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-24
Ligands: SO4, CL, GOL, 36Z
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Crystal Structure Of Atad2A Bromodomain Complexed With 3-(3,5-Dimethyl-1,2-Oxazol-4-Yl)-5-[(Phenylsulfonyl)Amino]Benzoicacid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.73 Å Release Date: 2014-12-24 Classification: GENE REGULATION Ligands: SO4, GOL, 37N, CL, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-24
Ligands: SO4, GOL, 37N, CL, DMS
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Crystal Structure Of Apo Atad2A Bromodomain With N1064 Alternate Conformation
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.27 Å Release Date: 2014-12-24 Classification: GENE REGULATION Ligands: SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-24
Ligands: SO4