Search Count: 33
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Pad2 With An Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.18 Å Release Date: 2025-07-30 Classification: HYDROLASE Ligands: A1CE0, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-07-30
Ligands: A1CE0, CA
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Potent Inhibition Of The Protein Arginine Deiminases (Pad1-4) By Targeting A Ca2+ Dependent Allosteric Binding Site
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.77 Å Release Date: 2025-05-28 Classification: HYDROLASE Ligands: CA, A1A8O |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-28
Ligands: CA, A1A8O
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Inhibiting Peptidylarginine Deiminases (Pad1-4) By Targeting A Ca2+ Dependent Allosteric Binding Site
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.44 Å Release Date: 2025-05-28 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: CA, A1BZK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-28
Ligands: CA, A1BZK
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Potent Inhibition Of The Protein Arginine Deiminases (Pad1-4) By Targeting A Ca2+ Dependent Allosteric Binding Site
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.41 Å Release Date: 2025-05-28 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: A1A9P, 3YZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-28
Ligands: A1A9P, 3YZ
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Crystal Structure Of The Human Pad2 Protein Bound To Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.64 Å Release Date: 2024-10-09 Classification: HYDROLASE Ligands: A1AJA, ACT, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-09
Ligands: A1AJA, ACT, CA
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Crystal Structure Of The Human Pad2 Protein Bound To Small Molecule
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2024-10-09 Classification: HYDROLASE Ligands: MPD, A1AJB, ACT, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-09
Ligands: MPD, A1AJB, ACT, CA
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Crystal Structure Of The Human Pad2 Protein Bound To Small Molecule
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2024-10-09 Classification: HYDROLASE Ligands: ACT, CA, A1AJC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-09
Ligands: ACT, CA, A1AJC
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Crystal Structure Of Jak2 With Compound 11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2020-11-25 Classification: TRANSFERASE Ligands: UWP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-11-25
Ligands: UWP
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Crystal Structure Of Tyk2 With Compound 11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2020-11-25 Classification: TRANSFERASE Ligands: UWP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-11-25
Ligands: UWP
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Crystal Structure Of Tyk2 With Compound 22
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.21 Å Release Date: 2020-11-25 Classification: TRANSFERASE Ligands: UWM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-11-25
Ligands: UWM
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Crystal Structure Of Tyk2 Kinase With Compound 13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.09 Å Release Date: 2020-04-08 Classification: TRANSFERASE/INHIBITOR Ligands: R5D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-08
Ligands: R5D
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Crystal Structure Of Tyk2 Kinase With Compound 14
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2020-04-08 Classification: TRANSFERASE/INHIBITOR Ligands: R4Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-08
Ligands: R4Y
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Crystal Structure Of Tyk2 Kinase With Compound 19
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.18 Å Release Date: 2020-04-08 Classification: TRANSFERASE/INHIBITOR Ligands: R4V |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-08
Ligands: R4V
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Crystal Structure Of Tyk2 Kinase With Compound 10
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2020-04-08 Classification: TRANSFERASE/INHIBITOR Ligands: R4S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-08
Ligands: R4S
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Crystal Structure Of Jak1 Kinase With Compound 10
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.11 Å Release Date: 2020-04-08 Classification: TRANSFERASE/INHIBITOR Ligands: R4S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-08
Ligands: R4S
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Jak3 With Cyanamide Cp10
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2018-11-28 Classification: TRANSFERASE/INHIBITOR Ligands: G4V |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-11-28
Ligands: G4V
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Jak3 With Cyanamide Cp23
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2018-11-28 Classification: TRANSFERASE/INHIBITOR Ligands: G54 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-11-28
Ligands: G54
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Jak3 With Cyanamide Cp34
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.66 Å Release Date: 2018-11-28 Classification: TRANSFERASE/INHIBITOR Ligands: G4Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-11-28
Ligands: G4Y
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Jak3 With Cyanamide Cp12
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.66 Å Release Date: 2018-11-28 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: HB4, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-11-28
Ligands: HB4, SO4
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Tyk2 With Compound 8
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2018-08-29 Classification: TRANSFERASE Ligands: G5D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-29
Ligands: G5D
