Search Count: 11
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Pyrrole-3-Carboxamides As Potent And Selective Jak2 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.77 Å Release Date: 2014-07-23 Classification: TRANSFERASE Ligands: GOL, VVQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-23
Ligands: GOL, VVQ
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Pyrrole-3-Carboxamides As Potent And Selective Jak2 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.82 Å Release Date: 2014-07-23 Classification: TRANSFERASE Ligands: 953, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-23
Ligands: 953, GOL
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Pyrrole-3-Carboxamides As Potent And Selective Jak2 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.66 Å Release Date: 2014-07-23 Classification: TRANSFERASE Ligands: BJG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-23
Ligands: BJG
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Structure Of Hsp90 With Nms-E973 Inhibitor Bound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2013-05-29 Classification: CHAPERONE Ligands: 9UN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-29
Ligands: 9UN
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Crystal Structure Of Polo-Like Kinase 1 In Complex With A 5-(2-Amino- Pyrimidin-4-Yl)-1H-Pyrrole Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2012-01-11 Classification: TRANSFERASE Ligands: ZN, TLA, 939 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-01-11
Ligands: ZN, TLA, 939
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Crystal Structure Of Polo-Like Kinase 1 In Complex With A 2-(2-Amino- Pyrimidin-4-Yl)-1,5,6,7-Tetrahydro-Pyrrolopyridin-4-One Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2012-01-11 Classification: TRANSFERASE Ligands: ZN, TLA, 664 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-01-11
Ligands: ZN, TLA, 664
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Crystal Structure Of Polo-Like Kinase 1 In Complex With A Pyrazoloquinazoline Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2010-05-19 Classification: TRANSFERASE Ligands: 071, ZN, TLA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-05-19
Ligands: 071, ZN, TLA
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Optimisation Of 6,6-Dimethyl Pyrrolo 3,4-C Pyrazoles: Identification Of Pha-793887, A Potent Cdk Inhibitor Suitable For Intravenous Dosing
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.51 Å Release Date: 2010-02-23 Classification: CELL CYCLE Ligands: SO4, 889 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-02-23
Ligands: SO4, 889
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Structure Of Cdk2-Cyclin A With A Pyrazolo(4,3-H) Quinazoline-3- Carboxamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2010-02-23 Classification: TRANSFERASE Ligands: WXV, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-02-23
Ligands: WXV, SO4
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Structure Of Cdk2-Cyclin A With Pha-848125
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2009-07-28 Classification: TRANSFERASE Ligands: P48, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-07-28
Ligands: P48, SO4
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Structure Of Cdk2-Cyclin A Complexed With 8-Anilino-1-Methyl-4,5-Dihydro- 1H-Pyrazolo[4,3-H] Quinazoline-3-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2009-07-28 Classification: TRANSFERASE Ligands: P49, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-07-28
Ligands: P49, SO4
