Search Count: 79
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Isopenicillin N Synthase With Ac-O-Methyl-D-Threonine
Organism: Emericella nidulans (strain fgsc a4 / atcc 38163 / cbs 112.46 / nrrl 194 / m139)
Method: X-RAY DIFFRACTION Resolution:1.82 Å Release Date: 2013-06-26 Classification: OXIDOREDUCTASE Ligands: M2W, FE, SO4, GOL |
Organism: Emericella nidulans (strain fgsc a4 / atcc 38163 / cbs 112.46 / nrrl 194 / m139)
Method: X-RAY DIFFRACTION
Release Date: 2013-06-26
Ligands: M2W, FE, SO4, GOL
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Isopenicillin N Synthase With The Dipeptide Substrate Analogue Ahc
Organism: Aspergillus nidulans fgsc a4
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2013-04-17 Classification: OXIDOREDUCTASE Ligands: FE, KKA, SO4 |
Organism: Aspergillus nidulans fgsc a4
Method: X-RAY DIFFRACTION
Release Date: 2013-04-17
Ligands: FE, KKA, SO4
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Isopenicillin N Synthase With Substrate Analogue Ahcmc
Organism: Emericella nidulans (strain fgsc a4 / atcc 38163 / cbs 112.46 / nrrl 194 / m139)
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2013-03-20 Classification: OXIDOREDUCTASE Ligands: FE, WT4, SO4, GOL |
Organism: Emericella nidulans (strain fgsc a4 / atcc 38163 / cbs 112.46 / nrrl 194 / m139)
Method: X-RAY DIFFRACTION
Release Date: 2013-03-20
Ligands: FE, WT4, SO4, GOL
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Isopenicillin N Synthase With Substrate Analogue Ahcv
Organism: Emericella nidulans (strain fgsc a4 / atcc 38163 / cbs 112.46 / nrrl 194 / m139)
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2013-02-06 Classification: OXIDOREDUCTASE Ligands: FE, HCV |
Organism: Emericella nidulans (strain fgsc a4 / atcc 38163 / cbs 112.46 / nrrl 194 / m139)
Method: X-RAY DIFFRACTION
Release Date: 2013-02-06
Ligands: FE, HCV
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Isopenicillin N Synthase With Ac-D-Methionine
Organism: Emericella nidulans (strain fgsc a4 / atcc 38163 / cbs 112.46 / nrrl 194 / m139)
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2012-02-08 Classification: OXIDOREDUCTASE Ligands: M8F, FE, SO4, GOL |
Organism: Emericella nidulans (strain fgsc a4 / atcc 38163 / cbs 112.46 / nrrl 194 / m139)
Method: X-RAY DIFFRACTION
Release Date: 2012-02-08
Ligands: M8F, FE, SO4, GOL
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Clinically Useful Alkyl Amine Renin Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.19 Å Release Date: 2011-11-30 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NAG, CL, RX5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-11-30
Ligands: NAG, CL, RX5
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Clinically Useful Alkyl Amine Renin Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.16 Å Release Date: 2011-11-30 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: CL, RX6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-11-30
Ligands: CL, RX6
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Isopenicillin N Synthase With Ac-D-S-Methyl-3R-Methylcysteine
Organism: Emericella nidulans (strain fgsc a4 / atcc 38163 / cbs 112.46 / nrrl 194 / m139)
Method: X-RAY DIFFRACTION Resolution:1.79 Å Release Date: 2011-08-31 Classification: OXIDOREDUCTASE Ligands: M9F, FE, SO4 |
Organism: Emericella nidulans (strain fgsc a4 / atcc 38163 / cbs 112.46 / nrrl 194 / m139)
Method: X-RAY DIFFRACTION
Release Date: 2011-08-31
Ligands: M9F, FE, SO4
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Alkyl Amine Renin Inhibitors: Filling S1 From S3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2011-08-03 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: RX0, GOL, NAG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-08-03
Ligands: RX0, GOL, NAG
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Isopenicillin N Synthase With Substrate Analogue L,L,D-Acd2Ab (Unexposed)
Organism: Emericella nidulans (strain fgsc a4 / atcc 38163 / cbs 112.46 / nrrl 194 / m139)
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2010-07-21 Classification: OXIDOREDUCTASE Ligands: FE2, ASV |
Organism: Emericella nidulans (strain fgsc a4 / atcc 38163 / cbs 112.46 / nrrl 194 / m139)
Method: X-RAY DIFFRACTION
Release Date: 2010-07-21
Ligands: FE2, ASV
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Optimization Of Orally Bioavailable Alkyl Amine Renin Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2010-01-12 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 22X, NAG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-01-12
Ligands: 22X, NAG
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Crystal Structure Of Human Renin Complexed With A Novel Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2009-06-23 Classification: Hydrolase/Hydrolase inhibitor Ligands: 72X, GOL, CL, NAG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-06-23
Ligands: 72X, GOL, CL, NAG
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Isopenicillin N Synthase With Substrate Analogue L,L,L-Acab (Unexposed)
Organism: Emericella nidulans (strain fgsc a4 / atcc 38163 / cbs 112.46 / nrrl 194 / m139)
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2008-11-04 Classification: OXIDOREDUCTASE Ligands: FE2, VB1, SO4 |
Organism: Emericella nidulans (strain fgsc a4 / atcc 38163 / cbs 112.46 / nrrl 194 / m139)
Method: X-RAY DIFFRACTION
Release Date: 2008-11-04
Ligands: FE2, VB1, SO4
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Isopenicillin N Synthase With Substrate Analogue Asmcov
Organism: Emericella nidulans (strain fgsc a4 / atcc 38163 / cbs 112.46 / nrrl 194 / m139)
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2008-11-04 Classification: OXIDOREDUCTASE Ligands: FE2, M11, SO4 |
Organism: Emericella nidulans (strain fgsc a4 / atcc 38163 / cbs 112.46 / nrrl 194 / m139)
Method: X-RAY DIFFRACTION
Release Date: 2008-11-04
Ligands: FE2, M11, SO4
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Isopenicillin N Synthase With Substrate Analogue Asmcov (Oxygen Exposed 1Min 20Bar)
Organism: Emericella nidulans (strain fgsc a4 / atcc 38163 / cbs 112.46 / nrrl 194 / m139)
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2008-11-04 Classification: OXIDOREDUCTASE Ligands: FE2, W2X, M11 |
Organism: Emericella nidulans (strain fgsc a4 / atcc 38163 / cbs 112.46 / nrrl 194 / m139)
Method: X-RAY DIFFRACTION
Release Date: 2008-11-04
Ligands: FE2, W2X, M11
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Isopenicillin N Synthase With Substrate Analogue L,L,L-Acomp (Unexposed)
Organism: Emericella nidulans (strain fgsc a4 / atcc 38163 / cbs 112.46 / nrrl 194 / m139)
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2008-09-23 Classification: OXIDOREDUCTASE Ligands: FE2, V10 |
Organism: Emericella nidulans (strain fgsc a4 / atcc 38163 / cbs 112.46 / nrrl 194 / m139)
Method: X-RAY DIFFRACTION
Release Date: 2008-09-23
Ligands: FE2, V10
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Isopenicillin N Synthase With Substrate Analogue Acomp (Unexposed)
Organism: Emericella nidulans (strain fgsc a4 / atcc 38163 / cbs 112.46 / nrrl 194 / m139)
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2008-07-29 Classification: OXIDOREDUCTASE Ligands: FE2, V20 |
Organism: Emericella nidulans (strain fgsc a4 / atcc 38163 / cbs 112.46 / nrrl 194 / m139)
Method: X-RAY DIFFRACTION
Release Date: 2008-07-29
Ligands: FE2, V20
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Isopenicillin N Synthase With Substrate Analogue Acomp (35Minutes Oxygen Exposure)
Organism: Emericella nidulans (strain fgsc a4 / atcc 38163 / cbs 112.46 / nrrl 194 / m139)
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2008-07-29 Classification: OXIDOREDUCTASE Ligands: VAZ, FE2, SO4, GOL |
Organism: Emericella nidulans (strain fgsc a4 / atcc 38163 / cbs 112.46 / nrrl 194 / m139)
Method: X-RAY DIFFRACTION
Release Date: 2008-07-29
Ligands: VAZ, FE2, SO4, GOL
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Isopenicillin N Synthase With A 2-Thiabicycloheptan-6-One Product Analogue
Organism: Emericella nidulans (strain fgsc a4 / atcc 38163 / cbs 112.46 / nrrl 194 / m139)
Method: X-RAY DIFFRACTION Resolution:1.30 Å Release Date: 2007-10-16 Classification: OXIDOREDUCTASE Ligands: A14, FE, SO4, GOL |
Organism: Emericella nidulans (strain fgsc a4 / atcc 38163 / cbs 112.46 / nrrl 194 / m139)
Method: X-RAY DIFFRACTION
Release Date: 2007-10-16
Ligands: A14, FE, SO4, GOL
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Isopenicillin N Synthase From Aspergillus Nidulans (Anaerobic Ac- Methyl-Cyclopropylglycine Fe Complex)
Organism: Emericella nidulans (strain fgsc a4 / atcc 38163 / cbs 112.46 / nrrl 194 / m139)
Method: X-RAY DIFFRACTION Resolution:1.30 Å Release Date: 2007-04-10 Classification: OXIDOREDUCTASE Ligands: ACW, SO4, FE2 |
Organism: Emericella nidulans (strain fgsc a4 / atcc 38163 / cbs 112.46 / nrrl 194 / m139)
Method: X-RAY DIFFRACTION
Release Date: 2007-04-10
Ligands: ACW, SO4, FE2
