Search Count: 21
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Potent Inhibition Of The Protein Arginine Deiminases (Pad1-4) By Targeting A Ca2+ Dependent Allosteric Binding Site
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.77 Å Release Date: 2025-05-28 Classification: HYDROLASE Ligands: CA, A1A8O |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-28
Ligands: CA, A1A8O
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Inhibiting Peptidylarginine Deiminases (Pad1-4) By Targeting A Ca2+ Dependent Allosteric Binding Site
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.44 Å Release Date: 2025-05-28 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: CA, A1BZK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-28
Ligands: CA, A1BZK
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Potent Inhibition Of The Protein Arginine Deiminases (Pad1-4) By Targeting A Ca2+ Dependent Allosteric Binding Site
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.41 Å Release Date: 2025-05-28 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: A1A9P, 3YZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-28
Ligands: A1A9P, 3YZ
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Crystal Structure Of The Human Pad2 Protein Bound To Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.64 Å Release Date: 2024-10-09 Classification: HYDROLASE Ligands: A1AJA, ACT, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-09
Ligands: A1AJA, ACT, CA
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Crystal Structure Of The Human Pad2 Protein Bound To Small Molecule
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2024-10-09 Classification: HYDROLASE Ligands: MPD, A1AJB, ACT, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-09
Ligands: MPD, A1AJB, ACT, CA
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Crystal Structure Of The Human Pad2 Protein Bound To Small Molecule
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2024-10-09 Classification: HYDROLASE Ligands: ACT, CA, A1AJC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-09
Ligands: ACT, CA, A1AJC
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Jak3 With Cyanamide Cp10
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2018-11-28 Classification: TRANSFERASE/INHIBITOR Ligands: G4V |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-11-28
Ligands: G4V
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Jak3 With Cyanamide Cp23
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2018-11-28 Classification: TRANSFERASE/INHIBITOR Ligands: G54 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-11-28
Ligands: G54
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Jak3 With Cyanamide Cp34
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.66 Å Release Date: 2018-11-28 Classification: TRANSFERASE/INHIBITOR Ligands: G4Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-11-28
Ligands: G4Y
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Jak3 With Cyanamide Cp12
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.66 Å Release Date: 2018-11-28 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: HB4, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-11-28
Ligands: HB4, SO4
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Jak3 With Covalent Inhibitor 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.34 Å Release Date: 2017-02-22 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: 7KU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: 7KU
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Jak3 With Covalent Inhibitor 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2017-02-22 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: 7KV, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: 7KV, SO4
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Jak3 With Covalent Inhibitor 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.93 Å Release Date: 2017-02-22 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: 7KX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: 7KX
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Jak3 With Covalent Inhibitor Pf-06651600
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2016-11-09 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: 7H4, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-09
Ligands: 7H4, SO4
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Binding Site Elucidation And Structure Guided Design Of Macrocyclic Il-17A Antagonists
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2016-08-31 Classification: IMMUNE SYSTEM/INHIBITOR Ligands: 63O |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2016-08-31
Ligands: 63O
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Binding Site Elucidation And Structure Guided Design Of Macrocyclic Il-17A Antagonists
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2016-08-31 Classification: IMMUNE SYSTEM/INHIBITOR Ligands: 63P |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2016-08-31
Ligands: 63P
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Binding Site Elucidation And Structure Guided Design Of Macrocyclic Il-17A Antagonists
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2016-08-31 Classification: IMMUNE SYSTEM/INHIBITOR Ligands: 63Q |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2016-08-31
Ligands: 63Q
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Yeast Poly(A) Polymerase In Complex With Fip1 Residues 80-105
Organism: Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2008-05-20 Classification: TRANSFERASE Ligands: MES, GOL |
Organism: Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION
Release Date: 2008-05-20
Ligands: MES, GOL
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Structure Of Yeast Poly(A) Polymerase With Atp And Oligo(A)
Organism: Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2007-08-28 Classification: Transferase/RNA Ligands: EDO, MG, ATP |
Organism: Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION
Release Date: 2007-08-28
Ligands: EDO, MG, ATP
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Structure Of Yeast Poly(A) Polymerase In A Closed Conformation.
Organism: Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2007-01-23 Classification: TRANSFERASE Ligands: FLC, MG |
Organism: Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION
Release Date: 2007-01-23
Ligands: FLC, MG
