Search Count: 79
![]() |
Crystal Structure Of Myst Acetyltransferase Domain In Complex With Inhibitor 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2026-02-11 Classification: TRANSFERASE/INHIBITOR Ligands: R7L, ZN, NA, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-02-11
Ligands: R7L, ZN, NA, GOL
![]() |
Crystal Structure Of Myst Acetyltransferase Domain In Complex With Inhibitor 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.39 Å Release Date: 2026-02-11 Classification: TRANSFERASE/INHIBITOR Ligands: ZN, SO4, NA, CL, GOL, A1CD4, A1CD3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-02-11
Ligands: ZN, SO4, NA, CL, GOL, A1CD4, A1CD3
![]() |
Crystal Structure Of Myst Acetyltransferase Domain In Complex With Inhibitor 8
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2026-02-11 Classification: TRANSFERASE/INHIBITOR Ligands: A1CDK, ZN, CL, NA, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-02-11
Ligands: A1CDK, ZN, CL, NA, GOL
![]() |
Crystal Structure Of Myst Acetyltransferase Domain In Complex With Inhibitor 10A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2026-02-11 Classification: TRANSFERASE/INHIBITOR Ligands: ZN, CL, GOL, A1CDJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-02-11
Ligands: ZN, CL, GOL, A1CDJ
![]() |
Crystal Structure Of Myst Acetyltransferase Domain In Complex With Inhibitor 10C
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2026-02-11 Classification: TRANSFERASE/INHIBITOR Ligands: ZN, CL, GOL, A1CDI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-02-11
Ligands: ZN, CL, GOL, A1CDI
![]() |
Crystal Structure Of Myst Acetyltransferase Domain In Complex With Inhibitor 10D
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2026-02-11 Classification: TRANSFERASE/INHIBITOR Ligands: ZN, CL, GOL, A1CDH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-02-11
Ligands: ZN, CL, GOL, A1CDH
![]() |
Crystal Structure Of Myst Acetyltransferase Domain In Complex With Inhibitor 10E
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.68 Å Release Date: 2026-02-11 Classification: TRANSFERASE/INHIBITOR Ligands: ZN, CL, GOL, A1CDG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-02-11
Ligands: ZN, CL, GOL, A1CDG
![]() |
Crystal Structure Of Myst Acetyltransferase Domain In Complex With Inhibitor 10B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2026-02-11 Classification: TRANSFERASE/INHIBITOR Ligands: ZN, CL, GOL, A1CDF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-02-11
Ligands: ZN, CL, GOL, A1CDF
![]() |
Crystal Structure Of Myst Acetyltransferase Domain In Complex With Inhibitor 18C
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.82 Å Release Date: 2026-02-11 Classification: TRANSFERASE/INHIBITOR Ligands: ZN, CL, GOL, A1CDE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-02-11
Ligands: ZN, CL, GOL, A1CDE
![]() |
Ptp1B In Complex With 182
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2023-08-02 Classification: HYDROLASE/INHIBITOR Ligands: CL, NA, V2O, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-08-02
Ligands: CL, NA, V2O, EDO
![]() |
Structure Of Full Length Human Ampk (A2B1G1) In Complex With A Small Molecule Activator Msg011
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.95 Å Release Date: 2022-06-29 Classification: SIGNALING PROTEIN Ligands: 4O7, ZQV, AMP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-06-29
Ligands: 4O7, ZQV, AMP
![]() |
Crystal Structure Of The Mertk Kinase Domain In Complex With Inhibitor Mips15692
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.06 Å Release Date: 2021-10-06 Classification: SIGNALING PROTEIN/INHIBITOR Ligands: YR7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-10-06
Ligands: YR7
![]() |
Crystal Structure Of Bcl-Xl Bound To Compound 8: (R)-3-(Benzylthio)-2-(3-(2-((4'-Chloro-[1,1'-Biphenyl]-2-Yl)Methyl)-1,2,3,4-Tetrahydroisoquinoline-6-Carbonyl)-3-(4-Methylbenzyl)Ureido)Propanoic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2021-05-05 Classification: Apoptosis/INHIBITOR Ligands: XOY, SO4, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-05
Ligands: XOY, SO4, EDO
![]() |
Crystal Structure Of Bcl-Xl Bound To Compound 2: (2R)-3-(Benzylsulfanyl)-2-({[(4-Methylphenyl)Methyl] [(4 Phenylphenyl)Carbonyl] Carbamoyl}Amino) Propanoic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2021-05-05 Classification: Apoptosis/INHIBITOR Ligands: XOU, SO4, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-05
Ligands: XOU, SO4, EDO
![]() |
Crystal Structure Of Bcl-Xl Bound To Compound 7: (R)-3-(Benzylthio)-2-(3-(4-Chloro-[1,1':2',1'':3'',1'''-Quaterphenyl]-4'''-Carbonyl)-3-(4-Methylbenzyl)Ureido)Propanoic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.87 Å Release Date: 2021-05-05 Classification: Apoptosis/INHIBITOR Ligands: QHV, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-05
Ligands: QHV, EDO
![]() |
Crystal Structure Of Bcl-Xl Bound To Compound 12: (R)-2-(3-([1,1'-Biphenyl]-4-Carbonyl)-3-(4-Methylbenzyl)Ureido)-3-((Cyclohexylmethyl)Sulfonyl)Propanoic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.24 Å Release Date: 2021-05-05 Classification: Apoptosis/INHIBITOR Ligands: SO4, EDO, QHS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-05
Ligands: SO4, EDO, QHS
![]() |
Crystal Structure Of Bcl-Xl Bound To Compound 13: (R)-2-(3-([1,1'-Biphenyl]-4-Carbonyl)-3-(4-Methylbenzyl)Ureido)-3-(((3R,5R,7R)-Adamantan-1-Ylmethyl)Sulfonyl)Propanoic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2021-05-05 Classification: Apoptosis/INHIBITOR Ligands: QHP, SO4, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-05
Ligands: QHP, SO4, EDO
![]() |
Crystal Structure Of Bcl-Xl Bound To Compound 15: (R)-2-(3-(2-((4'-Chloro-[1,1'-Biphenyl]-2-Yl)Methyl)-1,2,3,4-Tetrahydroisoquinoline-6-Carbonyl)-3-(4-Methylbenzyl)Ureido)-3-((Cyclohexylmethyl)Sulfonyl)Propanoic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.19 Å Release Date: 2021-05-05 Classification: Apoptosis/INHIBITOR Ligands: EDO, SO4, QHJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-05
Ligands: EDO, SO4, QHJ
![]() |
Crystal Structure Of Myst Acetyltransferase Domain In Complex With Inhibitor 92
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2020-04-01 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, GOL, NBJ, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-01
Ligands: ZN, GOL, NBJ, DMS
![]() |
Crystal Structure Of Myst Acetyltransferase Domain In Complex With Inhibitor 85
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2020-04-01 Classification: TRANSFERASE/TRANSERASE INHIBITOR Ligands: ZN, NB7, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-01
Ligands: ZN, NB7, GOL
