Search Count: 39
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Kat6A In Complex With Small Molecule Inhibitor Bay-184
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.69 Å Release Date: 2024-11-06 Classification: TRANSFERASE Ligands: ZN, A1IDR, EPE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-11-06
Ligands: ZN, A1IDR, EPE
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X-Ray Structure Of Smyd3 In Complex With Benzodiazepine-Type Inhibitor Compound 15
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.57 Å Release Date: 2021-07-07 Classification: TRANSFERASE Ligands: UZT, SAM, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-07
Ligands: UZT, SAM, ZN
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X-Ray Structure Of Smyd3 In Complex With Benzodiazepine-Type Inhibitor 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.03 Å Release Date: 2021-07-07 Classification: TRANSFERASE Ligands: UZQ, ZN, SAM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-07
Ligands: UZQ, ZN, SAM
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X-Ray Structure Of Smyd3 In Complex With The Benzodiazepine-Based Probe Bay-6035
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.52 Å Release Date: 2021-07-07 Classification: TRANSFERASE Ligands: UZK, SAM, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-07
Ligands: UZK, SAM, ZN
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X-Ray Structure Of Human K-Ras G12C In Complex With Covalent Isoquinolinone Inhibitor (Compound 3)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.64 Å Release Date: 2020-04-08 Classification: HYDROLASE Ligands: GDP, MG, MZQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-08
Ligands: GDP, MG, MZQ
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X-Ray Structure Of Human K-Ras G12C In Complex With Covalent Isoquinolinone Inhibitor (Compound 17)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.16 Å Release Date: 2020-04-08 Classification: HYDROLASE Ligands: GDP, MG, MZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-08
Ligands: GDP, MG, MZN
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Human Gpx4 In Complex With Covalent Inhibitor Ml162 (S Enantiomer)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.54 Å Release Date: 2020-04-01 Classification: OXIDOREDUCTASE Ligands: G9N, SO4, EDO, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-01
Ligands: G9N, SO4, EDO, DMS
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Wildtype Form (Apo) Of Human Gpx4 With Se-Cys46
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.01 Å Release Date: 2020-04-01 Classification: OXIDOREDUCTASE Ligands: CL, EOH, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-01
Ligands: CL, EOH, GOL
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Ras Guanine Nucleotide Exchange Factor Sos1 (Rem-Cdc25) In New Crystal Form
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2019-02-06 Classification: SIGNALING PROTEIN Ligands: EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-06
Ligands: EDO
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Ras Guanine Nucleotide Exchange Factor Sos1 (Rem-Cdc25) In Complex With Small Molecule Inhibitor Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2019-02-06 Classification: SIGNALING PROTEIN Ligands: EDO, AXE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-06
Ligands: EDO, AXE
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Ras Guanine Nucleotide Exchange Factor Sos1 (Rem-Cdc25) In Complex With Small Molecule Inhibitor Compound 17
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.01 Å Release Date: 2019-02-06 Classification: SIGNALING PROTEIN Ligands: AWT, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-06
Ligands: AWT, EDO
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Ras Guanine Nucleotide Exchange Factor Sos1 (Rem-Cdc25) In Complex With Small Molecule Inhibitor Compound 18
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2019-02-06 Classification: SIGNALING PROTEIN Ligands: AWZ, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-06
Ligands: AWZ, EDO
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Ras Guanine Nucleotide Exchange Factor Sos1 (Rem-Cdc25) In Complex With Small Molecule Inhibitor Compound 21
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2019-02-06 Classification: SIGNALING PROTEIN Ligands: AWW, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-06
Ligands: AWW, EDO
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Ras Guanine Nucleotide Exchange Factor Sos1 (Rem-Cdc25) In Complex With Small Molecule Inhibitor Bay-293 (Compound 23)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2019-02-06 Classification: SIGNALING PROTEIN Ligands: AXH, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-06
Ligands: AXH, EDO
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Ras Guanine Nucleotide Exchange Factor Sos2 (Rem-Cdc25), With Surface Mutations
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.72 Å Release Date: 2019-02-06 Classification: SIGNALING PROTEIN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-06
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Ras Guanine Exchange Factor Sos1 (Rem-Cdc25) In Complex With Kras(G12C)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2019-02-06 Classification: SIGNALING PROTEIN Ligands: GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-06
Ligands: GOL
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Ras Guanine Nucleotide Exchange Factor Sos1 (Rem-Cdc25) In Complex With Kras(G12C) And Fragment Screening Hit F1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2019-02-06 Classification: SIGNALING PROTEIN Ligands: GOL, BQ5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-06
Ligands: GOL, BQ5
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Ras Guanine Exchange Factor Sos1 (Rem-Cdc25) In Complex With Kras(G12C) And Fragment Screening Hit F2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2019-02-06 Classification: SIGNALING PROTEIN Ligands: GOL, BQ2, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-06
Ligands: GOL, BQ2, DMS
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Ras Guanine Exchange Factor Sos1 (Rem-Cdc25) In Complex With Kras(G12C) And Fragment Screening Hit F3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2019-02-06 Classification: SIGNALING PROTEIN Ligands: GOL, BPW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-06
Ligands: GOL, BPW
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Ras Guanine Exchange Factor Sos1 (Rem-Cdc25) In Complex With Kras(G12C) And Fragment Screening Hit F4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2019-02-06 Classification: SIGNALING PROTEIN Ligands: GOL, BOQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-06
Ligands: GOL, BOQ
