Search Count: 14
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Scaffold Hopping Via Ring Opening Enables Identification Of Acyclic Compounds As New Complement Factor D Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.17 Å Release Date: 2022-11-02 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: QIE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-02
Ligands: QIE
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Scaffold Hopping Via Ring Opening Enables Identification Of Acyclic Compounds As New Complement Factor D Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.21 Å Release Date: 2022-11-02 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: R7X, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-02
Ligands: R7X, GOL
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Scaffold Hopping Via Ring Opening Enables Identification Of Acyclic Compounds As New Complement Factor D Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2022-11-02 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: S7X |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-02
Ligands: S7X
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Crystal Structure Of Bcx7353(Orladeyo) In Complex With Human Plasma Kallikrein Serine Protease Domain At 2.1 Angstrom Resolution
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2021-09-15 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 0RI, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-15
Ligands: 0RI, PO4
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Crystal Structure Analysis Of Human Factor Viia , Souluble Tissue Factor Complexed With Bcx-3607
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2008-02-19 Classification: BLOOD CLOTTING Ligands: ASO, FUC, CA, 24X |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-02-19
Ligands: ASO, FUC, CA, 24X
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Structure Of 3,4-Dichloroisocoumarin-Inhibited Factor D
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 1999-07-22 Classification: SERINE PROTEASE Ligands: DIC, O |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 1999-07-22
Ligands: DIC, O
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Human Complement Factor D In Complex With Isatoic Anhydride Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 1999-06-22 Classification: SERINE PROTEASE Ligands: SOA, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 1999-06-22
Ligands: SOA, GOL
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Human Complement Factor D In A P21 Crystal Form
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 1999-06-22 Classification: SERINE PROTEASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 1999-06-22
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Factor D Inhibited By Diisopropyl Fluorophosphate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 1998-02-25 Classification: SERINE PROTEASE Ligands: DFP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 1998-02-25
Ligands: DFP
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Three-Dimensional Structure Of Influenza A N9 Neuraminidase And Its Complex With The Inhibitor 2-Deoxy 2,3-Dehydro-N-Acetyl Neuraminic Acid
Organism: Influenza a virus
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 1994-04-30 Classification: HYDROLASE(O-GLYCOSYL) Ligands: CA |
Organism: Influenza a virus
Method: X-RAY DIFFRACTION
Release Date: 1994-04-30
Ligands: CA
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Three-Dimensional Structure Of Influenza A N9 Neuraminidase And Its Complex With The Inhibitor 2-Deoxy 2,3-Dehydro-N-Acetyl Neuraminic Acid
Organism: Influenza a virus
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 1994-04-30 Classification: HYDROLASE(O-GLYCOSYL) Ligands: CA, DAN |
Organism: Influenza a virus
Method: X-RAY DIFFRACTION
Release Date: 1994-04-30
Ligands: CA, DAN
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Application Of Crystallographic And Modeling Methods In The Design Of Purine Nucleoside Phosphorylase Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.75 Å Release Date: 1993-01-15 Classification: PENTOSYLTRANSFERASE Ligands: SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 1993-01-15
Ligands: SO4
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Application Of Crystallographic And Modeling Methods In The Design Of Purine Nucleoside Phosphorylase Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.75 Å Release Date: 1993-01-15 Classification: PENTOSYLTRANSFERASE Ligands: SO4, GUN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 1993-01-15
Ligands: SO4, GUN
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Structure Of Calmodulin Refined At 2.2 Angstroms Resolution
Organism: Rattus rattus
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 1988-07-16 Classification: CALCIUM BINDING PROTEIN Ligands: CA |
Organism: Rattus rattus
Method: X-RAY DIFFRACTION
Release Date: 1988-07-16
Ligands: CA
