Search Count: 24
 |
Structure Of Human Setd8 In Complex With Covalent Inhibitor Am2928
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2025-07-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: E1J, H81 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-07-30
Ligands: E1J, H81
 |
Structure Of Human G9A Set-Domain (Ehmt2) In Complex With Covalent Inhibitor (Compound 1)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2022-07-06 Classification: GENE REGULATION Ligands: ZN, SAM, G5U, G4R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-07-06
Ligands: ZN, SAM, G5U, G4R
 |
Structure Of Human Glp Set-Domain (Ehmt1) In Complex With Covalent Inhibitor (Compound 1)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.85 Å Release Date: 2022-07-06 Classification: TRANSFERASE/INHIBITOR Ligands: ZN, G4R, G5U |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-07-06
Ligands: ZN, G4R, G5U
 |
Crystal Structure Of Spindlin1 In Complex With The Inhibitor Ms31
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2019-07-17 Classification: CELL CYCLE Ligands: MPD, DMS, JC5, GLY, PO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-07-17
Ligands: MPD, DMS, JC5, GLY, PO4, GOL
 |
Crystal Structure Of The Second Bromodomain Of Human Brd4 In Complex With Ms417 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2019-06-26 Classification: PROTEIN BINDING/Inhibitor Ligands: 0S6, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-26
Ligands: 0S6, EDO
 |
Structure Of Human Setd8 In Complex With Covalent Inhibitor Ms4138
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2019-05-01 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: EDO, E1J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-01
Ligands: EDO, E1J
 |
Crystal Structure Of Human Bromodomain-Containing Protein 4 (Brd4) Bromodomain With Ms645
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.46 Å Release Date: 2018-07-25 Classification: TRANSCRIPTION/INHIBITOR Ligands: CF6, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-25
Ligands: CF6, EDO
 |
Crystal Structure Of Human Bromodomain-Containing Protein 4 (Brd4) Bromodomain With Ms660
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.96 Å Release Date: 2018-07-18 Classification: TRANSCRIPTION Ligands: H1V |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-18
Ligands: H1V
 |
Structure Of Human Nnmt In Complex With Bisubstrate Inhibitor Ms2756
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2018-06-13 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: F0P, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-06-13
Ligands: F0P, EDO
 |
Crystal Structure Of Catalytic Domain Of G9A With Ms0105
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.74 Å Release Date: 2018-03-21 Classification: TRANSFERASE Ligands: ZN, SAM, 90P, GOL, UNX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-21
Ligands: ZN, SAM, 90P, GOL, UNX
 |
Crystal Structure Of Catalytic Domain Of Glp With Ms0105
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.74 Å Release Date: 2018-03-21 Classification: TRANSFERASE Ligands: SAM, 90P, ZN, CL, UNX, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-21
Ligands: SAM, 90P, ZN, CL, UNX, DMS
 |
Crystal Structure Of Apo Human Setd8
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2018-03-07 Classification: TRANSFERASE Ligands: EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-07
Ligands: EDO
 |
Structure Of Human G9A Set-Domain (Ehmt2) In Complex With Inhibitor 17: N~2~-Cyclopentyl-6,7-Dimethoxy-N~2~-Methyl-N~4~-(1-Methylpiperidin-4-Yl)Quinazoline-2,4-Diamine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2017-07-19 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, SAM, 9HG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-07-19
Ligands: ZN, SAM, 9HG
 |
Structure Of Human G9A Set-Domain (Ehmt2) In Complex With Inhibitor 13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2017-07-12 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, SAM, 9HJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-07-12
Ligands: ZN, SAM, 9HJ
 |
Structure Of Human Glp Set-Domain (Ehmt1) In Complex With Inhibitor 13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2017-07-12 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SAM, ZN, 9HJ, DIO, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-07-12
Ligands: SAM, ZN, 9HJ, DIO, GOL
 |
Structure Of Human Glp Set-Domain (Ehmt1) In Complex With Inhibitor 17
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2017-07-12 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SAM, ZN, 9HG, DIO, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-07-12
Ligands: SAM, ZN, 9HG, DIO, GOL
 |
Structure Of Human G9A Set-Domain (Ehmt2) In Complex With Inhibitor Ms0124
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2017-02-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, SAM, 7L6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: ZN, SAM, 7L6
 |
Structure Of Human Glp Set-Domain (Ehmt1) In Complex With Inhibitor Ms0124
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2017-02-22 Classification: Transferase/Transferase Inhibitor Ligands: SAM, ZN, 7L6, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: SAM, ZN, 7L6, EDO
 |
Crystal Structure Of Catalytic Domain Of Glp With Ms012
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.66 Å Release Date: 2017-02-01 Classification: TRANSFERASE Ligands: SAM, 7KZ, ZN, CL, GOL, UNX, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-01
Ligands: SAM, 7KZ, ZN, CL, GOL, UNX, DMS
 |
Crystal Structure Of Catalytic Domain Of G9A With Ms012
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2016-12-21 Classification: TRANSFERASE Ligands: ZN, SAM, 7KZ, CL, UNX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-12-21
Ligands: ZN, SAM, 7KZ, CL, UNX