Search Count: 17
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Binding Site Elucidation And Structure Guided Design Of Macrocyclic Il-17A Antagonists
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2016-08-31 Classification: IMMUNE SYSTEM/INHIBITOR Ligands: 63O |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2016-08-31
Ligands: 63O
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Binding Site Elucidation And Structure Guided Design Of Macrocyclic Il-17A Antagonists
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2016-08-31 Classification: IMMUNE SYSTEM/INHIBITOR Ligands: 63P |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2016-08-31
Ligands: 63P
 |
Binding Site Elucidation And Structure Guided Design Of Macrocyclic Il-17A Antagonists
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2016-08-31 Classification: IMMUNE SYSTEM/INHIBITOR Ligands: 63Q |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2016-08-31
Ligands: 63Q
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Chromo Domain Of Human Chromodomain Protein, Y-Like 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2016-05-25 Classification: PROTEIN BINDING |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-25
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Setd7 In Complex With Inhibitor (R)-Pfi-2 And S-Adenosyl-Methionine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2013-04-17 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SAM, 1L8, UNX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-04-17
Ligands: SAM, 1L8, UNX
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Setd7 In Complex With Inhibitor Pf-5426 And S-Adenosyl-Methionine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2013-03-27 Classification: transferase/transferase inhibitor Ligands: SAM, 1L4, UNX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-03-27
Ligands: SAM, 1L4, UNX
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Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With A Quinazolin Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.63 Å Release Date: 2012-10-31 Classification: PROTEIN BINDING/INHIBITOR Ligands: EDO, 15E |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-10-31
Ligands: EDO, 15E
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Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With A Quinazoline Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.69 Å Release Date: 2012-10-31 Classification: PROTEIN BINDING/INHIBITOR Ligands: EDO, 14Z, K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-10-31
Ligands: EDO, 14Z, K
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Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With A Quinazolin Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.62 Å Release Date: 2012-10-31 Classification: PROTEIN BINDING/INHIBITOR Ligands: 14X |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-10-31
Ligands: 14X
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Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With A Quinazolin Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.59 Å Release Date: 2012-10-31 Classification: SIGNALING PROTEIN/INHIBITOR Ligands: 13F, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-10-31
Ligands: 13F, EDO
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Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With The Inhibitor Pfi-1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.92 Å Release Date: 2012-04-18 Classification: PROTEIN BINDING/INHIBITOR Ligands: 0NS, NA, DMS, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-04-18
Ligands: 0NS, NA, DMS, EDO
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Set7/9 In Complex With Inhibitor (R)-(3-(3-Cyanophenyl)-1-Oxo-1-(Pyrrolidin-1-Yl)Propan-2-Yl)-1,2,3,4-Tetrahydroisoquinoline-6- Sulfonamide And S-Adenosylmethionine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2012-03-28 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SAM, 0N6, BME, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-03-28
Ligands: SAM, 0N6, BME, SO4
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Triazolopyridine Inhibitors Of P38 Kinase.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2011-11-30 Classification: TRANSFERASE Ligands: YIS, I46 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-11-30
Ligands: YIS, I46
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Triazolopyridine Inhibitors Of P38 Kinase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2011-11-30 Classification: TRANSFERASE Ligands: YIW, I46 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-11-30
Ligands: YIW, I46
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Triazolopyridine Inhibitors Of P38
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2011-11-30 Classification: TRANSFERASE Ligands: YIX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-11-30
Ligands: YIX
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Crystal Structure Of ((2S)-5-Amino-2-((1-N-Propyl-1H-Imidazol-4-Yl) Methyl)Pentanoic Acid) Uk396,082 A Tafia Inhibitor, Bound To Activated Porcine Pancreatic Carboxypeptidaseb
Organism: Sus scrofa
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2007-11-20 Classification: HYDROLASE Ligands: ZN, 720 |
Organism: Sus scrofa
Method: X-RAY DIFFRACTION
Release Date: 2007-11-20
Ligands: ZN, 720
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Crystal Structure Of The Potent Natural Product Inhibitor Balanol In Complex With The Catalytic Subunit Of Camp-Dependent Protein Kinase
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 1999-04-27 Classification: SERINE/THREONINE-PROTEIN KINASE Ligands: BA1 |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 1999-04-27
Ligands: BA1