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Search Count: 18

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8SWE image
Fgfr2 Kinase Domain Bound To Reversible Inhibitor Cmpd 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.24 Å Release Date: 2024-02-14
Classification: ONCOPROTEIN
Ligands: GOL, GSH, WXQ

8U1F image
Fgfr2 Kinase Domain Bound To Irreversible Inhibitor Cmpd 10

8STG image
Discovery And Clinical Validation Of Rly-4008, The First Highly Selective Fgfr2 Inhibitor With Activity Across Fgfr2 Alterations And Resistance Mutations

6UNP image
Crystal Structure Of The Kinase Domain Of Bmpr2-D485G
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.30 Å Release Date: 2021-07-07
Classification: TRANSFERASE
Ligands: ADP, MG, SO4, EDO

6UNQ image
Kinase Domain Of Alk2-K493A With Amppnp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.40 Å Release Date: 2021-07-07
Classification: TRANSFERASE
Ligands: ANP, MG

6UNR image
Kinase Domain Of Alk2-K492A/K493A With Amppnp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.20 Å Release Date: 2021-07-07
Classification: TRANSFERASE
Ligands: ANP, MG

6UNS image
Kinase Domain Of Alk2-K492A/K493A With Ldn-193189
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.30 Å Release Date: 2021-07-07
Classification: TRANSFERASE
Ligands: LDN

6JXT image
Crystal Structure Of Egfr 696-1022 Wt In Complex With Azd9291 Prepared By Cocrystallization
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.31 Å Release Date: 2020-04-29
Classification: TRANSFERASE
Ligands: YY3, CL

6JWL image
Crystal Structure Of Egfr 696-1022 L858R In Complex With Azd9291
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.55 Å Release Date: 2020-04-22
Classification: TRANSFERASE
Ligands: YY3

6JX0 image
Crystal Structure Of Egfr 696-1022 T790M In Complex With Azd9291 Prepared By Co-Crystallization
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.53 Å Release Date: 2020-04-22
Classification: TRANSFERASE
Ligands: YY3, CL

6JX4 image
Crystal Structure Of Egfr 696-1022 T790M In Complex With Azd9291 Prepared By Soaking
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.53 Å Release Date: 2020-04-22
Classification: TRANSFERASE
Ligands: YY3

6OP9 image
Her3 Pseudokinase Domain Bound To Bosutinib

5IEV image
Crystal Structure Of Bay 1000394 (Roniciclib) Bound To Cdk2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.03 Å Release Date: 2016-04-27
Classification: TRANSFERASE
Ligands: R0N

5IEX image
Crystal Structure Of (R,S)-S-{4-[(5-Bromo-4-{[(2R,3R)-2-Hydroxy-1-Methylpropyl]Oxy}- Pyrimidin-2-Yl)Amino]Phenyl}-S-Cyclopropylsulfoximide Bound To Cdk2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.03 Å Release Date: 2016-04-27
Classification: TRANSFERASE
Ligands: 6AF

5IEY image
Crystal Structure Of A Cdk Inhibitor Bound To Cdk2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.66 Å Release Date: 2016-04-27
Classification: TRANSFERASE
Ligands: 6AE

5IF1 image
Crystal Structure Apo Cdk2/Cyclin A


4FFB image
A Tog:Alpha/Beta-Tubulin Complex Structure Reveals Conformation-Based Mechanisms For A Microtubule Polymerase
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