Search Count: 18
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Fgfr2 Kinase Domain Bound To Reversible Inhibitor Cmpd 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.24 Å Release Date: 2024-02-14 Classification: ONCOPROTEIN Ligands: GOL, GSH, WXQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-02-14
Ligands: GOL, GSH, WXQ
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Fgfr2 Kinase Domain Bound To Irreversible Inhibitor Cmpd 10
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.33 Å Release Date: 2024-02-14 Classification: Transferase/Inhibitor Ligands: GOL, UIM, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-02-14
Ligands: GOL, UIM, SO4
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Discovery And Clinical Validation Of Rly-4008, The First Highly Selective Fgfr2 Inhibitor With Activity Across Fgfr2 Alterations And Resistance Mutations
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.79 Å Release Date: 2023-06-07 Classification: TRANSFERASE/INHIBITOR Ligands: WCJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-06-07
Ligands: WCJ
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Crystal Structure Of The Kinase Domain Of Bmpr2-D485G
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2021-07-07 Classification: TRANSFERASE Ligands: ADP, MG, SO4, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-07
Ligands: ADP, MG, SO4, EDO
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Kinase Domain Of Alk2-K493A With Amppnp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2021-07-07 Classification: TRANSFERASE Ligands: ANP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-07
Ligands: ANP, MG
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Kinase Domain Of Alk2-K492A/K493A With Amppnp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2021-07-07 Classification: TRANSFERASE Ligands: ANP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-07
Ligands: ANP, MG
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Kinase Domain Of Alk2-K492A/K493A With Ldn-193189
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2021-07-07 Classification: TRANSFERASE Ligands: LDN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-07
Ligands: LDN
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Crystal Structure Of Egfr 696-1022 Wt In Complex With Azd9291 Prepared By Cocrystallization
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.31 Å Release Date: 2020-04-29 Classification: TRANSFERASE Ligands: YY3, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-29
Ligands: YY3, CL
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Crystal Structure Of Egfr 696-1022 L858R In Complex With Azd9291
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2020-04-22 Classification: TRANSFERASE Ligands: YY3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-22
Ligands: YY3
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Crystal Structure Of Egfr 696-1022 T790M In Complex With Azd9291 Prepared By Co-Crystallization
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.53 Å Release Date: 2020-04-22 Classification: TRANSFERASE Ligands: YY3, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-22
Ligands: YY3, CL
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Crystal Structure Of Egfr 696-1022 T790M In Complex With Azd9291 Prepared By Soaking
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.53 Å Release Date: 2020-04-22 Classification: TRANSFERASE Ligands: YY3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-22
Ligands: YY3
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Her3 Pseudokinase Domain Bound To Bosutinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2019-08-21 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: DB8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-08-21
Ligands: DB8
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Crystal Structure Of Bay 1000394 (Roniciclib) Bound To Cdk2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.03 Å Release Date: 2016-04-27 Classification: TRANSFERASE Ligands: R0N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-27
Ligands: R0N
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Crystal Structure Of (R,S)-S-{4-[(5-Bromo-4-{[(2R,3R)-2-Hydroxy-1-Methylpropyl]Oxy}- Pyrimidin-2-Yl)Amino]Phenyl}-S-Cyclopropylsulfoximide Bound To Cdk2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.03 Å Release Date: 2016-04-27 Classification: TRANSFERASE Ligands: 6AF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-27
Ligands: 6AF
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Crystal Structure Of A Cdk Inhibitor Bound To Cdk2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.66 Å Release Date: 2016-04-27 Classification: TRANSFERASE Ligands: 6AE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-27
Ligands: 6AE
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Crystal Structure Apo Cdk2/Cyclin A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.61 Å Release Date: 2016-04-27 Classification: TRANSFERASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-27
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Tog2:Alpha/Beta-Tubulin Complex
Organism: Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION Resolution:2.81 Å Release Date: 2014-08-20 Classification: STRUCTURAL PROTEIN/Protein binding Ligands: MG, GTP |
Organism: Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION
Release Date: 2014-08-20
Ligands: MG, GTP
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A Tog:Alpha/Beta-Tubulin Complex Structure Reveals Conformation-Based Mechanisms For A Microtubule Polymerase
Organism: Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION Resolution:2.88 Å Release Date: 2012-08-15 Classification: HYDROLASE Ligands: MG, GTP |
Organism: Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION
Release Date: 2012-08-15
Ligands: MG, GTP
