Search Count: 17
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Translation Initiation Factor Eif-2B Complex With The Isohexide Diamine Gsk735
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2026-03-04 Classification: TRANSLATION Ligands: PRO, SO4, EDO, A1C32 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-03-04
Ligands: PRO, SO4, EDO, A1C32
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X-Ray Structure Of Furin Bound To Bos-318, A Small Molecule Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.24 Å Release Date: 2022-01-12 Classification: HYDROLASE/INHIBITOR Ligands: CA, XTA, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-12
Ligands: CA, XTA, EDO
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Crystal Structure Of Gsk6157 Bound To Perk (R587-R1092, Delete A660-T867) At 2.34A Resolution
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.34 Å Release Date: 2014-09-03 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 27D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-09-03
Ligands: 27D
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Crystal Structure Of Gsk6414 Bound To Perk (R587-R1092, Delete A660-T867) At 2.28 A Resolution
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.28 Å Release Date: 2012-08-08 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GOL, 0WH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-08-08
Ligands: GOL, 0WH
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Crystal Structure Of Gsk6924 Bound To Perk (R587-R1092, Delete A660-T867) At 2.70 A Resolution
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2012-08-08 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 924 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-08-08
Ligands: 924
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X-Ray Structure Of Polypeptide Deformylase Bound To A Acylprolinamide Inhibitor
Organism: Streptococcus pneumoniae
Method: X-RAY DIFFRACTION Resolution:1.78 Å Release Date: 2012-05-30 Classification: hydrolase/hydrolase inhibitor Ligands: NI, 0S5 |
Organism: Streptococcus pneumoniae
Method: X-RAY DIFFRACTION
Release Date: 2012-05-30
Ligands: NI, 0S5
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Phosphoinositide-Dependent Kinase-1 (Pdk1) With Lead Compound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2011-06-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GOL, SO4, JMZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-06-22
Ligands: GOL, SO4, JMZ
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Phosphoinositide-Dependent Kinase-1 (Pdk1) With Fragment8
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.75 Å Release Date: 2011-05-25 Classification: TRANSFERASE Ligands: GOL, JNZ, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-05-25
Ligands: GOL, JNZ, SO4
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Phosphoinositide-Dependent Kinase-1 (Pdk1) With Fragment11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2011-05-25 Classification: TRANSFERASE Ligands: GOL, SO4, JOZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-05-25
Ligands: GOL, SO4, JOZ
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Phosphoinositide-Dependent Kinase-1 (Pdk1) With Fragment17
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2011-05-25 Classification: TRANSFERASE Ligands: GOL, SO4, JPZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-05-25
Ligands: GOL, SO4, JPZ
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Phosphoinositide-Dependent Kinase-1 (Pdk1) Kinase Domain With 6-(3-Amino-1H-Indazol-6-Yl)-N4-Ethyl-2,4-Pyrimidinediamine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2011-03-09 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GOL, SO4, 3Q0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-09
Ligands: GOL, SO4, 3Q0
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Phosphoinositide-Dependent Kinase-1 (Pdk1) Kinase Domain With 6-[2-Amino-6-(4-Morpholinyl)-4-Pyrimidinyl]-1H-Indazol-3-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.49 Å Release Date: 2011-03-09 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GOL, SO4, 3Q1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-09
Ligands: GOL, SO4, 3Q1
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Phosphoinositide-Dependent Kinase-1 (Pdk1) Kinase Domain With 6-{2-Amino-6-[(3R)-3-Methyl-4-Morpholinyl]-4-Pyrimidinyl}-1H-Indazol-3-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2011-03-09 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GOL, SO4, 3Q2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-09
Ligands: GOL, SO4, 3Q2
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Phosphoinositide-Dependent Kinase-1 (Pdk1) Kinase Domain With 4-[2-Amino-6-(3-Amino-1H-Indazol-6-Yl)-4-Pyrimidinyl]-N-Phenyl-2-Morpholinecarboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2011-03-09 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GOL, SO4, 3Q3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-09
Ligands: GOL, SO4, 3Q3
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Phosphoinositide-Dependent Kinase-1 (Pdk1) Kinase Domain With (2R,5S)-1-[2-Amino-6-(3-Amino-1H-Indazol-6-Yl)-4-Pyrimidinyl]-6-Methyl-N-Phenyl-3-Piperidinecarboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2011-03-09 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GOL, SO4, 3Q4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-09
Ligands: GOL, SO4, 3Q4
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Phosphoinositide-Dependent Kinase-1 (Pdk1) Kinase Domain With 1,1-Dimethylethyl {(3R,6S)-1-[2-Amino-6-(3-Amino-1H-Indazol-6-Yl)-4-Pyrimidinyl]-6-Methyl-3-Piperidinyl}Carbamate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2011-03-09 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3Q5, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-09
Ligands: 3Q5, SO4, GOL
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Phosphoinositide-Dependent Kinase-1 (Pdk1) Kinase Domain With 1,1-Dimethylethyl{(3R,5R)-1-[2-Amino-6-(3-Amino-1H-Indazol-6-Yl)-4-Pyrimidinyl]-5-Methyl-3-Piperidinyl}Carbamate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2011-03-09 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3Q6, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-09
Ligands: 3Q6, SO4