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Search Count: 12

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6U4J image
Crystal Structure Of Idh1 R132H Mutant In Complex With Ft-2102

6O2Y image
Crystal Structure Of Idh1 R132H Mutant In Complex With Compound 24

6O2Z image
Crystal Structure Of Idh1 R132H Mutant In Complex With Compound 32

2YDI image
Discovery Of Checkpoint Kinase Inhibitor Azd7762 By Structure Based Design And Optimization Of Thiophene Carboxamide Ureas
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.60 Å Release Date: 2012-04-04
Classification: TRANSFERASE
Ligands: SO4, YDI

2YDK image
Discovery Of Checkpoint Kinase Inhibitor Azd7762 By Structure Based Design And Optimization Of Thiophene Carboxamide Ureas
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.90 Å Release Date: 2012-04-04
Classification: TRANSFERASE
Ligands: SO4, GOL, YDK

2YER image
Synthesis And Evaluation Of Triazolones As Checkpoint Kinase 1 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.83 Å Release Date: 2012-03-14
Classification: TRANSFERASE
Ligands: TQ1, SO4, EDO

2YEX image
Synthesis And Evaluation Of Triazolones As Checkpoint Kinase 1 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.30 Å Release Date: 2012-03-14
Classification: TRANSFERASE
Ligands: GOL, YEX, SO4

2YDJ image
Discovery Of Checkpoint Kinase Inhibitor Azd7762 By Structure Based Design And Optimization Of Thiophene Carboxamide Ureas
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.85 Å Release Date: 2012-01-25
Classification: TRANSFERASE
Ligands: YDJ, PO4

3PZE image
Jnk1 In Complex With Inhibitor

2X8D image
Discovery Of A Novel Class Of Triazolones As Checkpoint Kinase Inhibitors - Hit To Lead Exploration
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.90 Å Release Date: 2010-08-11
Classification: TRANSFERASE
Ligands: X8D, SO4

2X8E image
Discovery Of A Novel Class Of Triazolones As Checkpoint Kinase Inhibitors - Hit To Lead Exploration
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.50 Å Release Date: 2010-08-11
Classification: TRANSFERASE
Ligands: X8E, SO4

2X8I image
Discovery Of A Novel Class Of Triazolones As Checkpoint Kinase Inhibitors - Hit To Lead Exploration
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.92 Å Release Date: 2010-08-11
Classification: TRANSFERASE
Ligands: X8I, SO4, GOL
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