Search Count: 33
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Crystal Structure Of Rhodesain In Complex With A Macrolactam Inhibitor
Organism: Trypanosoma brucei rhodesiense
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2018-04-11 Classification: HYDROLASE Ligands: C2K, EDO |
Organism: Trypanosoma brucei rhodesiense
Method: X-RAY DIFFRACTION
Release Date: 2018-04-11
Ligands: C2K, EDO
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Crystal Structure Of Rhodesain In Complex With A Macrolactam Inhibitor
Organism: Trypanosoma brucei rhodesiense
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2018-04-11 Classification: HYDROLASE Ligands: EDO, C3E |
Organism: Trypanosoma brucei rhodesiense
Method: X-RAY DIFFRACTION
Release Date: 2018-04-11
Ligands: EDO, C3E
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Crystal Structure Of Rhodesain In Complex With A Macrolactam Inhibitor
Organism: Trypanosoma brucei rhodesiense
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2018-04-11 Classification: HYDROLASE Ligands: EDO, C2W |
Organism: Trypanosoma brucei rhodesiense
Method: X-RAY DIFFRACTION
Release Date: 2018-04-11
Ligands: EDO, C2W
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Cathepsin L In Complex With (3S,14E)-19-Chloro-N-(1-Cyanocyclopropyl)-5-Oxo-12,17-Dioxa-4-Azatricyclo[16.2.2.06,11]Docosa-1(21),6(11),7,9,14,18(22),19-Heptaene-3-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.37 Å Release Date: 2018-04-11 Classification: HYDROLASE Ligands: C3E, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-04-11
Ligands: C3E, GOL
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Cathepsin L In Complex With (3S,14E)-19-Chloro-N-(1-Cyanocyclopropyl)-5-Oxo-17-Oxa-4-Azatricyclo[16.2.2.06,11]Docosa-1(21),6,8,10,14,18(22),19-Heptaene-3-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.34 Å Release Date: 2018-04-11 Classification: HYDROLASE Ligands: C7Q |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-04-11
Ligands: C7Q
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Cathepsin L In Complex With (3S,14E)-8-(Azetidin-3-Yl)-19-Chloro-N-(1-Cyanocyclopropyl)-5-Oxo-12,17-Dioxa-4-Azatricyclo[16.2.2.06,11]Docosa-1(21),6,8,10,14,18(22),19-Heptaene-3-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.02 Å Release Date: 2018-04-11 Classification: HYDROLASE Ligands: C7T, ZN, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-04-11
Ligands: C7T, ZN, CL
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Mouse Cathepsin S With Covalent Ligand (3S,4S)-N-[(2E)-2-Iminoethyl]-4-(Morpholin-4-Ylcarbonyl)-1-(Phenylsulfonyl)Pyrrolidine-3-Carboxamide
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.47 Å Release Date: 2014-09-10 Classification: hydrolase/hydrolase inhibitor Ligands: 2EW |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2014-09-10
Ligands: 2EW
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Mouse Cathepsin S With Covalent Ligand (3S,4S)-1-[(2-Chlorophenyl)Sulfonyl]-N-[(2E)-2-Iminoethyl]-4-(Morpholin-4-Ylcarbonyl)Pyrrolidine-3-Carboxamide
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2014-08-20 Classification: hydrolase/hydrolase inhibitor Ligands: 2EV |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2014-08-20
Ligands: 2EV
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Mouse Cathepsin S With Covalent Ligand
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.25 Å Release Date: 2013-11-27 Classification: HYDROLASE Ligands: MG2 |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2013-11-27
Ligands: MG2
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Mouse Cathepsin S With Covalent Ligand
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.96 Å Release Date: 2013-11-27 Classification: HYDROLASE Ligands: QQV, SO4 |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2013-11-27
Ligands: QQV, SO4
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Cathepsin L With A Nitrile Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.15 Å Release Date: 2011-11-23 Classification: HYDROLASE Ligands: YJ2, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-11-23
Ligands: YJ2, GOL
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Cathepsin L With A Nitrile Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.30 Å Release Date: 2011-11-23 Classification: HYDROLASE Ligands: YJ8, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-11-23
Ligands: YJ8, GOL
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Cathepsin L With A Nitrile Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.35 Å Release Date: 2011-11-23 Classification: HYDROLASE Ligands: YJ9, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-11-23
Ligands: YJ9, GOL
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Cathepsin L With A Nitrile Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2011-11-23 Classification: HYDROLASE Ligands: YJ9, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-11-23
Ligands: YJ9, GOL
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Cathepsin L With A Nitrile Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.14 Å Release Date: 2011-11-23 Classification: HYDROLASE Ligands: 424 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-11-23
Ligands: 424
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Cathepsin L With A Nitrile Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2011-01-12 Classification: HYDROLASE Ligands: 424 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-01-12
Ligands: 424
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Cathepsin L With A Nitrile Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:0.90 Å Release Date: 2011-01-12 Classification: HYDROLASE Ligands: XU3, BTB, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-01-12
Ligands: XU3, BTB, CL
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Cathepsin L With A Nitrile Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.12 Å Release Date: 2011-01-12 Classification: HYDROLASE Ligands: DJT, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-01-12
Ligands: DJT, GOL
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Cathepsin L With A Nitrile Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2011-01-12 Classification: HYDROLASE Ligands: XU5, GOL, FLC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-01-12
Ligands: XU5, GOL, FLC
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Factor Xa In Complex With A Pyrrolidine-3,4-Dicarboxylic Acid Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.66 Å Release Date: 2010-08-04 Classification: BLOOD CLOTTING Ligands: XBV, CA, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-08-04
Ligands: XBV, CA, NA
