Search Count: 53
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Crystal Structure Of Pac1R In Complex With Peptide Antagonist
Organism: Homo sapiens, Lutzomyia longipalpis
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2021-03-24 Classification: SIGNALING PROTEIN/ANTAGONIST |
Organism: Homo sapiens, Lutzomyia longipalpis
Method: X-RAY DIFFRACTION
Release Date: 2021-03-24
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Crystal Structure Of Jztx-V
Organism: Chilobrachys guangxiensis
Method: X-RAY DIFFRACTION Resolution:1.05 Å Release Date: 2019-03-06 Classification: TOXIN Ligands: BR, SO4, GOL |
Organism: Chilobrachys guangxiensis
Method: X-RAY DIFFRACTION
Release Date: 2019-03-06
Ligands: BR, SO4, GOL
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Crystal Structure Of Human Pim-1 Kinase In Complex With A Quinazolinone-Pyrrolodihydropyrrolone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2019-01-16 Classification: TRANSFERASE Ligands: JYG, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-01-16
Ligands: JYG, GOL
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Jztx-V Toxin Peptide, Wild-Type
Organism: Chilobrachys guangxiensis
Method: SOLUTION NMR Release Date: 2018-05-16 Classification: TOXIN |
Organism: Chilobrachys guangxiensis
Method: SOLUTION NMR
Release Date: 2018-05-16
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Solution Nmr Structure Of Jztx-V, A Nav 1.7 Inhibitory Peptide
Organism: Chilobrachys guangxiensis
Method: SOLUTION NMR Release Date: 2018-05-02 Classification: TOXIN |
Organism: Chilobrachys guangxiensis
Method: SOLUTION NMR
Release Date: 2018-05-02
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Crystal Structure Of Human Pim-1 Kinase In Complex With An Imidazopyridazine Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2016-11-09 Classification: transferase/transferase inhibitor Ligands: 6YN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-09
Ligands: 6YN
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Crystal Structure Of Human Pim-1 Kinase In Complex With A Quinazolinone-Pyrrolopyrrolone Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2016-06-22 Classification: transferase/transferase inhibitor Ligands: 6CD, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-22
Ligands: 6CD, GOL
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Crystal Structure Of Human Pim-1 Kinase In Complex With A Macrocyclic Quinoxaline-Pyrrolodihydropiperidinone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2016-05-04 Classification: transferase/transferase inhibitor Ligands: 5QO, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-04
Ligands: 5QO, GOL
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X-Ray Structure Of Racemic Shk Q16K Toxin
Organism: Stoichactis helianthus
Method: X-RAY DIFFRACTION Resolution:1.20 Å Release Date: 2015-09-09 Classification: TOXIN Ligands: SO4 |
Organism: Stoichactis helianthus
Method: X-RAY DIFFRACTION
Release Date: 2015-09-09
Ligands: SO4
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Human Gkrp Bound To Amg2882 And Sorbitol-6-Phosphate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2015-05-13 Classification: sugar binding protein/inhibitor Ligands: 2WY, S6P, IOD, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-05-13
Ligands: 2WY, S6P, IOD, GOL, SO4
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Human Gkrp Bound To Amg-3295 And Sorbitol-6-Phosphate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.43 Å Release Date: 2015-05-13 Classification: sugar binding protein/inhibitor Ligands: 2WX, S6P, IOD, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-05-13
Ligands: 2WX, S6P, IOD, GOL, SO4
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Human Gkrp Bound To Amg-0696 And Sorbitol-6-Phosphate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2015-05-13 Classification: sugar binding protein/inhibitor Ligands: 2WZ, S6P, IOD, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-05-13
Ligands: 2WZ, S6P, IOD, GOL, SO4
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Human Gkrp Bound To Amg-0265 (N-[(R)-(2-Chlorophenyl){7-[4-(2-Hydroxypropan-2-Yl) Pyridin-2-Yl]-1-Benzothiophen-2-Yl}Methyl]Cyclopropanesulfonamide) And Sorbitol-6-Phosphate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2015-03-18 Classification: transferase/transferase inhibitor Ligands: 2Y6, S6P, IOD, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-03-18
Ligands: 2Y6, S6P, IOD, GOL, SO4
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Crystal Structure Of Human Pim-1 Kinase In Complex With A Thiazolamine-Indazole Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2015-02-11 Classification: transferase/transferase inhibitor Ligands: 3U5, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-02-11
Ligands: 3U5, GOL
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Crystal Structure Of Human Pim-1 Kinase In Complex With A Thiadiazolamine-Indole Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2015-02-11 Classification: transferase/transferase inhibitor Ligands: 3U6, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-02-11
Ligands: 3U6, GOL
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Co-Crystal Structure Of Pim1 With Compound 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.05 Å Release Date: 2015-02-04 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3UR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-02-04
Ligands: 3UR
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Crystal Structure Of Human Pim-1 Kinase In Complex With An Aminooxadiazole-Indole Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2015-02-04 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 38W, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-02-04
Ligands: 38W, GOL
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Crystal Structure Of Human Pim-1 Kinase In Complex With An Azaspiro Pyrazinyl-Indazole Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2015-02-04 Classification: transferase/transferase inhibitor Ligands: GOL, 3U1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-02-04
Ligands: GOL, 3U1
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Co-Crystal Structure Of Perk Bound To N-{5-[(6,7-Dimethoxyquinolin-4-Yl)Oxy]Pyridin-2-Yl}-1-Methyl-3-Oxo-2-Phenyl-5-(Pyridin-4-Yl)-2,3-Dihydro-1H-Pyrazole-4-Carboxamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2015-02-04 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3Z2, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-02-04
Ligands: 3Z2, SO4
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Co-Crystal Structure Of Perk With 2-Amino-N-[4-Methoxy-3-(Trifluoromethyl)Phenyl]-4-Methyl-3-[2-(Methylamino)Quinazolin-6-Yl]Benzamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2015-01-28 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3Z1, TLA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-01-28
Ligands: 3Z1, TLA
