Search Count: 21
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Human Acetylcholinesterase In Complex With Reactivator, Hlo7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.42 Å Release Date: 2019-06-12 Classification: HYDROLASE Ligands: NAG, HLO, FUC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-12
Ligands: NAG, HLO, FUC
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Crystal Structure Of Irak4 In Complex With Compound 9
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.64 Å Release Date: 2017-05-24 Classification: TRANSFERASE Ligands: 8BV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-24
Ligands: 8BV
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Crystal Structure Of Irak4 In Complex With Compound 11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.64 Å Release Date: 2017-05-24 Classification: TRANSFERASE Ligands: 8BY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-24
Ligands: 8BY
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Crystal Structure Of Irak4 In Complex With Compound 12
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2017-05-24 Classification: TRANSFERASE Ligands: 8C1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-24
Ligands: 8C1
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Crystal Structure Of Irak4 In Complex With Compound 14
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.84 Å Release Date: 2017-05-24 Classification: TRANSFERASE Ligands: 8CD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-24
Ligands: 8CD
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Crystal Structure Of Irak4 In Complex With Compound 30
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.02 Å Release Date: 2017-05-24 Classification: TRANSFERASE Ligands: 8CG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-24
Ligands: 8CG
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Crystal Structure Of Itk In Complex With Compound 1 [4-(Carbamoylamino)-1-(Naphthalen-1-Yl)-1H-Pyrazole-3-Carboxamide]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2014-04-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: M0Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: M0Y
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Crystal Structure Of Itk In Complex With Compound 5 {4-(Carbamoylamino)-1-(7-Methoxynaphthalen-1-Yl)-1H-Pyrazole-3-Carboxamide}
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2014-04-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: M0Z |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: M0Z
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Crystal Structure Of Itk In Complex With Compound 7 [4-(Carbamoylamino)-1-(7-Ethoxynaphthalen-1-Yl)-1H-Pyrazole-3-Carboxamide]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2014-04-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1YZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: 1YZ
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Crystal Structure Of Itk In Complex With Compound 8 [4-(Carbamoylamino)-1-(7-Propoxynaphthalen-1-Yl)-1H-Pyrazole-3-Carboxamide]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2014-04-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1E0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: 1E0
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Crystal Structure Of Itk In Complex With Compound 9 [4-(Carbamoylamino)-1-[7-(Propan-2-Yloxy)Naphthalen-1-Yl]-1H-Pyrazole-3-Carboxamide]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2014-04-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: QWS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: QWS
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Crystal Structure Of Itk In Complex With Compound 9 [4-(Carbamoylamino)-1-[7-(Propan-2-Yloxy)Naphthalen-1-Yl]-1H-Pyrazole-3-Carboxamide] And Adp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.52 Å Release Date: 2014-04-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: QWS, ADP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: QWS, ADP
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Crystal Structure Of Itk In Complex With Compound 52
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.48 Å Release Date: 2012-11-14 Classification: transferase/transferase inhibitor Ligands: 18R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-11-14
Ligands: 18R
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Crystal Structure Of Itk In Complext With Compound 40
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.43 Å Release Date: 2012-11-14 Classification: transferase/transferase inhibitor Ligands: 13L |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-11-14
Ligands: 13L
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Crystal Structure Of Itk In Complex With Compound 53
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.48 Å Release Date: 2012-11-14 Classification: transferase/transferase inhibitor Ligands: 13J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-11-14
Ligands: 13J
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Inhibitor Bound To A Dfg-Out Structure Of The Kinase Domain Of Csf-1R
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.40 Å Release Date: 2010-09-15 Classification: TRANSFERASE Ligands: LC0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-09-15
Ligands: LC0
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Inhibitor Bound To A Dfg-In Structure Of The Kinase Domain Of Csf-1R
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2010-03-02 Classification: TRANSFERASE Ligands: SO4, BDY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-03-02
Ligands: SO4, BDY
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Crystal Structure Of An Optimzied Benzothiophene Inhibitor Bound To Mapkap Kinase-2 (Mk-2)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.80 Å Release Date: 2009-04-07 Classification: TRANSFERASE Ligands: B97 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-04-07
Ligands: B97
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Crystal Structure Of A Benzthiophene Lead Bound To Mapkap Kinase-2 (Mk-2)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.50 Å Release Date: 2009-04-07 Classification: TRANSFERASE Ligands: B98 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-04-07
Ligands: B98
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Crystal Structure Of A Benzthiophene Inhibitor Bound To Human Cyclin-Dependent Kinase-2 (Cdk-2)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2009-04-07 Classification: TRANSFERASE Ligands: B98 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-04-07
Ligands: B98
