Search Count: 21
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Structure-Based Discovery Of Novel Non-Covalent Small Molecule Inhibitors Of Usp30
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.58 Å Release Date: 2025-05-21 Classification: HYDROLASE Ligands: A1L7W, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-21
Ligands: A1L7W, ZN
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Identification Of Small-Molecule Binding Sites Of A Ubiquitin-Conjugating Enzyme-Ube2T Through Fragment-Based Screening
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.54 Å Release Date: 2024-02-28 Classification: LIGASE Ligands: V23, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-02-28
Ligands: V23, EDO
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Identification Of Small-Molecule Binding Sites Of A Ubiquitin-Conjugating Enzyme-Ube2T Through Fragment-Based Screening
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2024-02-28 Classification: LIGASE Ligands: V2R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-02-28
Ligands: V2R
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Identification And Characterization Of Inhibitors Covalently Modifying Catalytic Cysteine Of Ube2T And Blocking Ubiquitin Transfer
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.76 Å Release Date: 2023-11-29 Classification: LIGASE/INHIBITOR Ligands: V6C, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-29
Ligands: V6C, EDO
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Identification And Characterization Of Inhibitors Covalently Modifying Catalytic Cysteine Of Ube2T And Blocking Ubiquitin Transfer
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.06 Å Release Date: 2023-11-29 Classification: LIGASE/INHIBITOR Ligands: V5L, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-29
Ligands: V5L, EDO
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Structure-Activity Relationship Studies Of Allosteric Inhibitors Of Eya2 Tyrosine Phosphatase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.49 Å Release Date: 2021-12-29 Classification: TRANSCRIPTION Ligands: 1RI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-12-29
Ligands: 1RI
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Structure-Activity Relationship Studies Of Allosteric Inhibitors Of Eya2 Tyrosine Phosphatase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.30 Å Release Date: 2021-12-29 Classification: TRANSCRIPTION Ligands: 1SI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-12-29
Ligands: 1SI
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Fragment-Based Lead Discovery Of Indazole-Based Compounds As Axl Kinase Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.15 Å Release Date: 2021-10-13 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: E56 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-10-13
Ligands: E56
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Strategic Design Of Catalytic Lysine-Targeting Reversible Covalent Bcr-Abl Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.72 Å Release Date: 2021-06-09 Classification: TRANSFERASE Ligands: FVC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-06-09
Ligands: FVC
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Strategic Design Of Catalytic Lysine-Targeting Reversible Covalent Bcr-Abl Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2021-06-09 Classification: TRANSFERASE Ligands: HJ9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-06-09
Ligands: HJ9
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Structural Basis For An Allosteric Eya2 Phosphatase Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.18 Å Release Date: 2019-06-05 Classification: TRANSCRIPTION Ligands: 9FX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-05
Ligands: 9FX
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Crystal Structure Of An Unlignaded Peptide-Substrate-Binding Domain Of Human Type Ii Collagen Prolyl 4-Hydroxylase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.87 Å Release Date: 2018-09-12 Classification: HYDROLASE Ligands: SO4, DMS, GLY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-09-12
Ligands: SO4, DMS, GLY
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Crystal Structure Of A Pro-9 Complexed Peptide-Substrate-Binding Domain Of Human Type Ii Collagen Prolyl 4-Hydroxylase
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2018-09-12 Classification: HYDROLASE Ligands: SO4, DMS |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2018-09-12
Ligands: SO4, DMS
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Crystal Structure Of Peptide-Substrate-Binding Domain Of Human Type Ii Collagen Prolyl 4-Hydroxylase Complex With Pro-Pro-Gly-Pro-Ala-Gly-Pro-Pro-Gly.
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.48 Å Release Date: 2018-09-12 Classification: HYDROLASE Ligands: SO4, DMS |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2018-09-12
Ligands: SO4, DMS
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Crystal Structure The Peptide-Substrate-Binding Domain Of Human Type Ii Collagen Prolyl 4-Hydroxylase Complexed With Pro-Pro-Gly-Pro-Arg-Gly-Pro-Pro-Gly.
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2018-09-12 Classification: HYDROLASE Ligands: SO4, DMS |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2018-09-12
Ligands: SO4, DMS
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Crystal Structure The Peptide-Substrate-Binding Domain Of Human Type Ii Collagen Prolyl 4-Hydroxylase Complexed With Pro-Pro-Gly-Pro-Glu-Gly-Pro-Pro-Gly.
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.68 Å Release Date: 2018-09-12 Classification: HYDROLASE Ligands: SO4, DMS |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2018-09-12
Ligands: SO4, DMS
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Crystal Structure Of The Semet-Labeled N-Terminal Domain And Peptide Substrate Binding Domain Of Alpha Subunit Of Prolyl-4 Hydroxylase Type I From Human.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.99 Å Release Date: 2013-10-09 Classification: OXIDOREDUCTASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-10-09
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Crystal Structure Of The Apo Form Of N-Terminal Domain And Peptide Substrate Binding Domain Of Prolyl-4 Hydroxylase Type I From Human
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2013-10-09 Classification: OXIDOREDUCTASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-10-09
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Crystal Structure Of The Peptide(Pro-Pro-Gly)3 Bound Complex Of N- Terminal Domain And Peptide Substrate Binding Domain Of Prolyl-4 Hydroxylase (Residues 1-238) Type I From Human
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2013-10-09 Classification: OXIDOREDUCTASE |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2013-10-09
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Crystal Structure Of The Peptide(Pro-Pro-Gly)3 Bound Complex Of N- Terminal Domain And Peptide Substrate Binding Domain Of Prolyl-4 Hydroxylase (Residues 1-244) Type I From Human
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.95 Å Release Date: 2013-10-09 Classification: OXIDOREDUCTASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-10-09