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Search Count: 9

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3RWP image
Discovery Of A Novel, Potent And Selective Inhibitor Of 3-Phosphoinositide Dependent Kinase (Pdk1)

3RWQ image
Discovery Of A Novel, Potent And Selective Inhibitor Of 3-Phosphoinositide Dependent Kinase (Pdk1)

3SC1 image
Novel Isoquinolone Pdk1 Inhibitors Discovered Through Fragment-Based Lead Discovery

2XP2 image
Structure Of The Human Anaplastic Lymphoma Kinase In Complex With Crizotinib (Pf-02341066)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.90 Å Release Date: 2010-09-15
Classification: TRANSFERASE
Ligands: VGH

2WKM image
X-Ray Structure Of Pha-00665752 Bound To The Kinase Domain Of C-Met
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.20 Å Release Date: 2010-08-25
Classification: TRANSFERASE
Ligands: PFY

3JVR image
Characterization Of The Chk1 Allosteric Inhibitor Binding Site
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.76 Å Release Date: 2009-10-06
Classification: TRANSFERASE
Ligands: AGX

3JVS image
Characterization Of The Chk1 Allosteric Inhibitor Binding Site
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.90 Å Release Date: 2009-10-06
Classification: TRANSFERASE
Ligands: AGY

2WGJ image
X-Ray Structure Of Pf-02341066 Bound To The Kinase Domain Of C-Met
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.00 Å Release Date: 2009-06-02
Classification: TRANSFERASE
Ligands: VGH

1SPU image
Structure Of Oxidoreductase
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