Search Count: 9
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Discovery Of A Novel, Potent And Selective Inhibitor Of 3-Phosphoinositide Dependent Kinase (Pdk1)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.92 Å Release Date: 2011-11-16 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GOL, SO4, ABQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-11-16
Ligands: GOL, SO4, ABQ
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Discovery Of A Novel, Potent And Selective Inhibitor Of 3-Phosphoinositide Dependent Kinase (Pdk1)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2011-11-16 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3RW, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-11-16
Ligands: 3RW, GOL, SO4
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Novel Isoquinolone Pdk1 Inhibitors Discovered Through Fragment-Based Lead Discovery
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2011-10-26 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3S1, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-10-26
Ligands: 3S1, SO4, GOL
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Structure Of The Human Anaplastic Lymphoma Kinase In Complex With Crizotinib (Pf-02341066)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2010-09-15 Classification: TRANSFERASE Ligands: VGH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-09-15
Ligands: VGH
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X-Ray Structure Of Pha-00665752 Bound To The Kinase Domain Of C-Met
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2010-08-25 Classification: TRANSFERASE Ligands: PFY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-08-25
Ligands: PFY
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Characterization Of The Chk1 Allosteric Inhibitor Binding Site
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.76 Å Release Date: 2009-10-06 Classification: TRANSFERASE Ligands: AGX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-10-06
Ligands: AGX
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Characterization Of The Chk1 Allosteric Inhibitor Binding Site
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2009-10-06 Classification: TRANSFERASE Ligands: AGY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-10-06
Ligands: AGY
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X-Ray Structure Of Pf-02341066 Bound To The Kinase Domain Of C-Met
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2009-06-02 Classification: TRANSFERASE Ligands: VGH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-06-02
Ligands: VGH
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Structure Of Oxidoreductase
Organism: Escherichia coli
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 1997-03-12 Classification: OXIDOREDUCTASE Ligands: CU, CA |
Organism: Escherichia coli
Method: X-RAY DIFFRACTION
Release Date: 1997-03-12
Ligands: CU, CA
