Search Count: 23
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Bace1 In Complex With 4-(Cyclohexylamino)-1-(3-Fluorophenyl)-8-(3-Isopropoxybenzyl)-1,3,8-Triazaspiro[4.5]Dec-3-En-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2015-08-05 Classification: Hydrolase/hydrolase inhibitor Ligands: 4QA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-05
Ligands: 4QA
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Bace1 In Complex With 8-(3-((1-Aminopropan-2-Yl)Oxy)Benzyl)-4-(Cyclohexylamino)-1-(3-Fluorophenyl)-1,3,8-Triazaspiro[4.5]Dec-3-En-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2015-08-05 Classification: Hydrolase/Hydrolase inhibitor Ligands: 4QD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-05
Ligands: 4QD
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Bace1 In Complex With 8-Benzyl-4-(Cyclohexylamino)-1-(3-Fluorophenyl)-7-Methyl-1,3,8-Triazaspiro[4.5]Dec-3-En-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2015-08-05 Classification: Hydrolase/hydrolase inhibitor Ligands: 4QF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-05
Ligands: 4QF
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Synthesis And Evaluation Of Heterocyclic Catechol Mimics As Inhibitors Of Catechol-O-Methyltransferase (Comt): Structure With Cmpd18 (1-(Biphenyl-3-Yl)-3-Hydroxypyridin-4(1H)-One)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2015-04-15 Classification: transferase/transferase inhibitor Ligands: 43G, MG, SAM, MES |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-15
Ligands: 43G, MG, SAM, MES
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Synthesis And Evaluation Of Heterocyclic Catechol Mimics As Inhibitors Of Catechol-O-Methyltransferase (Comt): Structure With Cmpd32 ([1-(Biphenyl-3-Yl)-5-Hydroxy-4-Oxo-1,4-Dihydropyridin-3-Yl]Boronic Acid)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2015-04-15 Classification: transferase/transferase inhibitor Ligands: 43H, MG, SAM, MES |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-15
Ligands: 43H, MG, SAM, MES
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Synthesis And Evaluation Of Heterocyclic Catechol Mimics As Inhibitors Of Catechol-O-Methyltransferase (Comt): Structure With Cmpd27B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2015-04-15 Classification: transferase/transferase inhibitor Ligands: 43J, MG, SAM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-15
Ligands: 43J, MG, SAM
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Structure Of Dually Phosphorylated C-Met Receptor Kinase In Complex With An Mk-8033 Analog
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2013-12-11 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1JC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-12-11
Ligands: 1JC
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Structure Of Dually Phosphorylated C-Met Receptor Kinase In Complex With An Mk-2461 Analog
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2012-02-01 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: M61 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-02-01
Ligands: M61
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Structure Of The Apo Met Receptor Kinase In The Dually-Phosphorylated, Activated State
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2011-01-19 Classification: TRANSFERASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-01-19
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Structure Of Dually-Phosphorylated Met Receptor Kinase In Complex With An Mk-2461 Analog With Specificity For The Activated Receptor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2011-01-19 Classification: transferase/transferase inhibitor Ligands: Q6W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-01-19
Ligands: Q6W
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Hiv-1 Reverse Transcriptase With Inhibitor
Organism: Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION Resolution:2.79 Å Release Date: 2010-06-09 Classification: TRANSFERASE/HYDROLASE Ligands: MN, LP7, NVP |
Organism: Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION
Release Date: 2010-06-09
Ligands: MN, LP7, NVP
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Hiv-1 Reverse Transcriptase With Inhibitor
Organism: Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION Resolution:2.23 Å Release Date: 2010-06-09 Classification: TRANSFERASE/HYDROLASE Ligands: LP8, MN, NVP |
Organism: Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION
Release Date: 2010-06-09
Ligands: LP8, MN, NVP
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Hiv-1 Reverse Transcriptase With Inhibitor
Organism: Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2010-06-09 Classification: TRANSFERASE/HYDROLASE Ligands: LP9, MN |
Organism: Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION
Release Date: 2010-06-09
Ligands: LP9, MN
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P15 Hiv Rnaseh Domain With Inhibitor Mk3
Organism: Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2010-06-09 Classification: VIRAL PROTEIN Ligands: MN, LP9 |
Organism: Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION
Release Date: 2010-06-09
Ligands: MN, LP9
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Discovery Of Aminoheterocycles As A Novel Beta-Secretase Inhibitor Class
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2009-07-07 Classification: HYDROLASE Ligands: B35 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-07-07
Ligands: B35
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Crystal Structure Of Hiv-1 Protease Complexed With Pl-100
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2008-07-22 Classification: HYDROLASE Ligands: A00 |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2008-07-22
Ligands: A00
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Crystal Structure Of Vaccinia Virus L1 Protein
Organism: Vaccinia virus
Method: X-RAY DIFFRACTION Resolution:1.51 Å Release Date: 2005-03-01 Classification: VIRAL PROTEIN |
Organism: Vaccinia virus
Method: X-RAY DIFFRACTION
Release Date: 2005-03-01
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Crystal Structure Of A Human Vgamma9/Vdelta2 T Cell Receptor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.12 Å Release Date: 2001-06-20 Classification: IMMUNE SYSTEM Ligands: SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2001-06-20
Ligands: SO4
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Crystal Structure Of The Rna-Binding Domain Of The Transcriptional Terminator Protein Rho
Organism: Escherichia coli bl21(de3)
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 1998-06-17 Classification: TRANSCRIPTION TERMINATION |
Organism: Escherichia coli bl21(de3)
Method: X-RAY DIFFRACTION
Release Date: 1998-06-17
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The Nmr Structure Of The Rna Binding Domain Of E.Coli Rho Factor Suggests Possible Rna-Protein Interactions, 10 Structures
Organism: Escherichia coli bl21(de3)
Method: SOLUTION NMR Release Date: 1998-05-27 Classification: TRANSCRIPTION TERMINATION |
Organism: Escherichia coli bl21(de3)
Method: SOLUTION NMR
Release Date: 1998-05-27
