Search Count: 22
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Crystal Structure Of Monkey Tlr7 Ectodomain With Compound 5
Organism: Macaca mulatta
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2024-02-07 Classification: IMMUNE SYSTEM Ligands: NAG, QEC, SO4 |
Organism: Macaca mulatta
Method: X-RAY DIFFRACTION
Release Date: 2024-02-07
Ligands: NAG, QEC, SO4
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Crystal Structure Of Monkey Tlr7 Ectodomain With Compound 20
Organism: Macaca mulatta
Method: X-RAY DIFFRACTION Resolution:3.14 Å Release Date: 2024-02-07 Classification: IMMUNE SYSTEM Ligands: NAG, SO4, QCX |
Organism: Macaca mulatta
Method: X-RAY DIFFRACTION
Release Date: 2024-02-07
Ligands: NAG, SO4, QCX
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Crystal Structure Of Ntmt1 In Complex With Compound Yd206
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.17 Å Release Date: 2022-12-14 Classification: TRANSFERASE/INHIBITOR Ligands: SAH, KYF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-12-14
Ligands: SAH, KYF
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Crystal Structure Of The Human Brd2 Bd1 Bromodomain In Complex With 9-(Cyclopropylmethyl)-7-[(2R,6S)-2,6-Dimethylmorpholine-4-Carbonyl]-3-(3,5-Dimethyl-1,2-Oxazol-4-Yl)-9H-Carbazole-1-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.49 Å Release Date: 2021-09-29 Classification: CELL CYCLE Ligands: YW1, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-29
Ligands: YW1, EDO
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Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With 9-Benzyl-2-(3,5-Dimethyl-1,2-Oxazol-4-Yl)-7-(2-Hydroxypropan-2-Yl)-9H-Carbazole-4-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2021-09-29 Classification: CELL CYCLE Ligands: YW4, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-29
Ligands: YW4, EDO
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Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With 2-(3,5-Dimethyl-1,2-Oxazol-4-Yl)-7-(2-Hydroxypropan-2-Yl)-9-[(S)-(Oxan-4-Yl)(Phenyl)Methyl]-9H-Carbazole-4-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2021-09-29 Classification: CELL CYCLE Ligands: YW7, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-29
Ligands: YW7, EDO
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Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With Bms-986158, 2-{3-(1,4-Dimethyl-1H-1,2,3-Triazol-5-Yl)-5-[(S)-(Oxan-4-Yl)(Phenyl)Methyl]-5H-Pyrido[3,2-B]Indol-7-Yl}Propan-2-Ol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2021-09-29 Classification: CELL CYCLE Ligands: YWA, IOD, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-29
Ligands: YWA, IOD, EDO
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Crystal Structure Of Rar-Related Orphan Receptor C (Nhis-Rorgt(244-487)-L6-Src1(678-692)) In Complex With {3,5-Dichloro-4-[4-Methoxy-3-(Propan-2-Yl)Phenoxy]Phenyl}Methanol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.62 Å Release Date: 2021-01-20 Classification: TRANSFERASE/Agonist Ligands: Z7G |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-20
Ligands: Z7G
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Crystal Structure Of Rar-Related Orphan Receptor C (Nhis-Rorgt(244-487)-L6-Src1(678-692)) In Complex With {3,5-Dichloro-4-[4-Methoxy-3-(Propan-2-Yl)Phenoxy]Phenyl}Methanol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.42 Å Release Date: 2021-01-20 Classification: TRANSFERASE/Agonist Ligands: Z7H |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-20
Ligands: Z7H
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Crystal Structure Of Rar-Related Orphan Receptor C (Nhis-Rorgt(244-487)-L6-Src1(678-692)) In Complex With {3,5-Dichloro-4-[4-Methoxy-3-(Propan-2-Yl)Phenoxy]Phenyl}Methanol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.14 Å Release Date: 2021-01-20 Classification: TRANSFERASE/Agonist Ligands: Z7I |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-20
Ligands: Z7I
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Substituted Benzyloxytricyclic Compounds As Retinoic Acid-Related Orphan Receptor Gamma T Agonists
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.26 Å Release Date: 2020-06-17 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: Z7F |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-06-17
Ligands: Z7F
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Substituted Benzyloxytricyclic Compounds As Retinoic Acid-Related Orphan Receptor Gamma T Agonists
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2020-04-29 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: TKJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-29
Ligands: TKJ
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Substituted Benzyloxytricyclic Compounds As Retinoic Acid-Related Orphan Receptor Gamma T Agonists
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.61 Å Release Date: 2020-04-29 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: Z7D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-29
Ligands: Z7D
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Tyrosine-Protein Kinase Lck Bound To Compound 11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.81 Å Release Date: 2019-10-09 Classification: SIGNALING PROTEIN/INHIBITOR Ligands: ODJ, CXS, SO4, NI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-10-09
Ligands: ODJ, CXS, SO4, NI
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Crystal Structure Of Human Baff In Complex With Fab Fragment Of Anti-Baff Antibody Belimumab
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2018-04-04 Classification: IMMUNE SYSTEM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-04-04
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Structure Of Apo-Tbaldh3
Organism: Trypanosoma brucei
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2017-04-19 Classification: OXIDOREDUCTASE Ligands: GOL |
Organism: Trypanosoma brucei
Method: X-RAY DIFFRACTION
Release Date: 2017-04-19
Ligands: GOL
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The First Bet Bromodomain Of Brd4 Bound To Compound 13 In A Bivalent Manner
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.48 Å Release Date: 2016-09-21 Classification: Transcription Factor Ligands: XNH, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-21
Ligands: XNH, GOL
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Plasmodium Vivax N-Myristoyltransferase With Quinoline Inhibitor
Organism: Plasmodium vivax
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2012-06-27 Classification: TRANSFERASE Ligands: 9MT, NHW, CL, MG, SO4 |
Organism: Plasmodium vivax
Method: X-RAY DIFFRACTION
Release Date: 2012-06-27
Ligands: 9MT, NHW, CL, MG, SO4
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Structure Of Rabbit Muscle Glycogen Phosphorylase In Complex With Ligand
Organism: Oryctolagus cuniculus
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2007-02-13 Classification: TRANSFERASE Ligands: SO4, PLR, 2TH |
Organism: Oryctolagus cuniculus
Method: X-RAY DIFFRACTION
Release Date: 2007-02-13
Ligands: SO4, PLR, 2TH
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Structure Of Rabbit Muscle Glycogen Phosphorylase In Complex With Thienopyrrole
Organism: Oryctolagus cuniculus
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2007-02-13 Classification: TRANSFERASE Ligands: PLR, 3TH |
Organism: Oryctolagus cuniculus
Method: X-RAY DIFFRACTION
Release Date: 2007-02-13
Ligands: PLR, 3TH
