Search Count: 9
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Structure Of Human Hdac2 In Complex With A 2-Substituted Benzamide Inhibitor (Compound 20)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.26 Å Release Date: 2020-12-30 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, CA, SO4, PEG, WBA, DMS, WBD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-30
Ligands: ZN, CA, SO4, PEG, WBA, DMS, WBD
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Structure Of Human Hdac2 In Complex With A 2-Substituted Benzamide Inhibitor (Compound 16)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.68 Å Release Date: 2020-12-30 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, CA, PEG, WB4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-30
Ligands: ZN, CA, PEG, WB4
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Co-Structure Of Btk Kinase Domain With L-005085737 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2020-07-22 Classification: TRANSFERASE Ligands: ULV, 5WE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-22
Ligands: ULV, 5WE
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Co-Structure Of Btk Kinase Domain With L-005191930 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2020-07-22 Classification: TRANSFERASE Ligands: ULY, 5WE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-22
Ligands: ULY, 5WE
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Co-Structure Of Btk Kinase Domain With L-005298385 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.34 Å Release Date: 2020-07-22 Classification: TRANSFERASE Ligands: UM4, EDO, BTB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-22
Ligands: UM4, EDO, BTB
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Discovery Of Mk-8353: An Orally Bioavailable Dual Mechanism Erk Inhibitor For Oncology
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2018-08-08 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, G67 |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2018-08-08
Ligands: SO4, G67
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Discovery Of 3(S)-Thiomethyl Pyrrolidine Erk Inhibitors For Oncology
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2018-05-23 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: SO4, F8V |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2018-05-23
Ligands: SO4, F8V
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Btk-Inhibitor Co-Structure
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.89 Å Release Date: 2016-03-23 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: 5WH, 5WE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-03-23
Ligands: 5WH, 5WE
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Btk Kinase Domain With Inhibitor 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2016-02-03 Classification: TRANSFERASE Ligands: 5WF, 5WE, CL, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-03
Ligands: 5WF, 5WE, CL, EDO
