Search Count: 26
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Halk In Complex With Compound 7 N-((1S)-1-(5-Fluoropyridin-2-Yl)Ethyl)-1-(5-Methyl-1H-Pyrazol-3-Yl)-3-(Oxetan-3-Ylsulfonyl)-1H-Pyrrolo[2,3-B]Pyridin-6-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2019-05-01 Classification: PROTEIN BINDING Ligands: HKJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-01
Ligands: HKJ
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Halk In Complex With Compound 9 (6-(((1S)-1-(5-Fluoropyridin-2-Yl)Ethyl)Amino)-1-(3-Methyl-1H-Pyrazol-5-Yl)-1H-Pyrrolo[2,3-B]Pyridin-3-Yl)(Morpholin-4-Yl)Methanone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.46 Å Release Date: 2019-05-01 Classification: TRANSFERASE/INHIBITOR Ligands: J3Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-01
Ligands: J3Y
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Halk In Complex With Compound 1 (S)-N-(1-(2,4-Difluorophenyl)Ethyl)-3-(3-Methyl-1H-Pyrazol-5-Yl)Imidazo[1,2-B]Pyridazin-6-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2019-05-01 Classification: TRANSFERASE/INHIBITOR Ligands: J4M |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-01
Ligands: J4M
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Adp Ribose Pyrophosphatase In Apo State At 0.91 Angstrom Resolution
Organism: Thermus thermophilus
Method: X-RAY DIFFRACTION Resolution:0.91 Å Release Date: 2016-04-27 Classification: HYDROLASE Ligands: SO4, GOL |
Organism: Thermus thermophilus
Method: X-RAY DIFFRACTION
Release Date: 2016-04-27
Ligands: SO4, GOL
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Adp Ribose Pyrophosphatase From Thermus Thermophilus Hb8 In Apo State At 0.92 Angstrom Resolution
Organism: Thermus thermophilus
Method: X-RAY DIFFRACTION Resolution:0.92 Å Release Date: 2016-04-27 Classification: HYDROLASE Ligands: GOL, SO4 |
Organism: Thermus thermophilus
Method: X-RAY DIFFRACTION
Release Date: 2016-04-27
Ligands: GOL, SO4
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Adp Ribose Pyrophosphatase From Thermus Thermophilus Hb8 In Es-State At 0.97 Angstrom Resolution
Organism: Thermus thermophilus hb8
Method: X-RAY DIFFRACTION Resolution:0.97 Å Release Date: 2016-04-27 Classification: HYDROLASE Ligands: AR6, GOL |
Organism: Thermus thermophilus hb8
Method: X-RAY DIFFRACTION
Release Date: 2016-04-27
Ligands: AR6, GOL
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Adp Ribose Pyrophosphatase From Thermus Thermophilus Hb8 In Es-State At 1.00 Angstrom Resolution
Organism: Thermus thermophilus hb8
Method: X-RAY DIFFRACTION Resolution:1.00 Å Release Date: 2016-04-27 Classification: HYDROLASE Ligands: AR6 |
Organism: Thermus thermophilus hb8
Method: X-RAY DIFFRACTION
Release Date: 2016-04-27
Ligands: AR6
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Adp Ribose Pyrophosphatase From Thermus Thermophilus Hb8 In Esm-State At Reaction Time Of 3 Min
Organism: Thermus thermophilus hb8
Method: X-RAY DIFFRACTION Resolution:1.15 Å Release Date: 2016-04-27 Classification: HYDROLASE Ligands: AR6, GOL, SO4, MN |
Organism: Thermus thermophilus hb8
Method: X-RAY DIFFRACTION
Release Date: 2016-04-27
Ligands: AR6, GOL, SO4, MN
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Adp Ribose Pyrophosphatase From Thermus Thermophilus Hb8 In Esm-State At Reaction Time Of 6 Min
Organism: Thermus thermophilus hb8
Method: X-RAY DIFFRACTION Resolution:1.12 Å Release Date: 2016-04-27 Classification: HYDROLASE Ligands: AR6, MN, GOL, SO4 |
Organism: Thermus thermophilus hb8
Method: X-RAY DIFFRACTION
Release Date: 2016-04-27
Ligands: AR6, MN, GOL, SO4
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Adp Ribose Pyrophosphatase From Thermus Thermophilus Hb8 In Esmm-State At Reaction Time Of 10 Min
Organism: Thermus thermophilus hb8
Method: X-RAY DIFFRACTION Resolution:1.09 Å Release Date: 2016-04-27 Classification: HYDROLASE Ligands: AR6, GOL, SO4, MN |
Organism: Thermus thermophilus hb8
Method: X-RAY DIFFRACTION
Release Date: 2016-04-27
Ligands: AR6, GOL, SO4, MN
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Adp Ribose Pyrophosphatase From Thermus Thermophilus Hb8 In Esmm-State At Reaction Time Of 15 Min
Organism: Thermus thermophilus hb8
Method: X-RAY DIFFRACTION Resolution:1.22 Å Release Date: 2016-04-27 Classification: HYDROLASE Ligands: AR6, MN, GOL, SO4 |
Organism: Thermus thermophilus hb8
Method: X-RAY DIFFRACTION
Release Date: 2016-04-27
Ligands: AR6, MN, GOL, SO4
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Adp Ribose Pyrophosphatase From Thermus Thermophilus Hb8 In Esmm-State At Reaction Time Of 20 Min
Organism: Thermus thermophilus hb8
Method: X-RAY DIFFRACTION Resolution:1.14 Å Release Date: 2016-04-27 Classification: HYDROLASE Ligands: AR6, MN, GOL, SO4 |
Organism: Thermus thermophilus hb8
Method: X-RAY DIFFRACTION
Release Date: 2016-04-27
Ligands: AR6, MN, GOL, SO4
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Dp Ribose Pyrophosphatase From Thermus Thermophilus Hb8 In E'-State At Reaction Time Of 30 Min
Organism: Thermus thermophilus hb8
Method: X-RAY DIFFRACTION Resolution:1.15 Å Release Date: 2016-04-27 Classification: HYDROLASE Ligands: GOL, SO4, MN |
Organism: Thermus thermophilus hb8
Method: X-RAY DIFFRACTION
Release Date: 2016-04-27
Ligands: GOL, SO4, MN
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Adp Ribose Pyrophosphatase From Thermus Thermophilus Hb8 In E'-State At Reaction Time Of 50 Min
Organism: Thermus thermophilus hb8
Method: X-RAY DIFFRACTION Resolution:1.10 Å Release Date: 2016-04-27 Classification: HYDROLASE Ligands: GOL, SO4, MN |
Organism: Thermus thermophilus hb8
Method: X-RAY DIFFRACTION
Release Date: 2016-04-27
Ligands: GOL, SO4, MN
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Egfr Kinase Domain Complexed With Compound 20A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2013-03-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: W32, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-03-06
Ligands: W32, SO4
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Egfr Kinase Domain Complexed With Compound 19B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2013-03-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: W19, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-03-06
Ligands: W19, SO4
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Egfr Kinase Domain T790M/L858R Mutant With Tak-285
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2013-01-16 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 03P |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-01-16
Ligands: 03P
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Egfr Kinase Domain T790M/L858R Mutant With Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2013-01-16 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: W2P |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-01-16
Ligands: W2P
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Egfr Kinase Domain T790M/L858R Mutant With Hki-272
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2013-01-16 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: HKI, MES |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-01-16
Ligands: HKI, MES
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Egfr Kinase Domain T790M/L858R Mutant With Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2013-01-16 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: W2R, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-01-16
Ligands: W2R, EDO
