Search Count: 36
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Structure Of 1 In Complex With Gdp-Kras
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.18 Å Release Date: 2025-08-06 Classification: HYDROLASE Ligands: GDP, MG, EDO, A1I1P |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-08-06
Ligands: GDP, MG, EDO, A1I1P
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Structure Of 5 In Complex With Gdp-Kras
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.00 Å Release Date: 2025-08-06 Classification: HYDROLASE Ligands: GDP, MG, EDO, A1I1R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-08-06
Ligands: GDP, MG, EDO, A1I1R
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Structure Of 10 In Complex With Gdp-Kras
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:0.95 Å Release Date: 2025-08-06 Classification: HYDROLASE Ligands: GDP, MG, EDO, WYU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-08-06
Ligands: GDP, MG, EDO, WYU
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Structure Of 12 In Complex With Gdp-Kras
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.06 Å Release Date: 2025-08-06 Classification: HYDROLASE Ligands: GDP, MG, EDO, A1I1Z |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-08-06
Ligands: GDP, MG, EDO, A1I1Z
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Structure Of 18 (Bi-2493) In Complex With Gdp-Kras
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.01 Å Release Date: 2025-08-06 Classification: HYDROLASE Ligands: GDP, MG, EDO, VU6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-08-06
Ligands: GDP, MG, EDO, VU6
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Identification Of Multiple Ligand Hotspots On Sos2, Compound 9
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2025-02-05 Classification: SIGNALING PROTEIN Ligands: A1ASY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-02-05
Ligands: A1ASY
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Identification Of Multiple Ligand Hotspots On Sos2, Compound 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.82 Å Release Date: 2025-02-05 Classification: SIGNALING PROTEIN Ligands: A1ASX, DMS, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-02-05
Ligands: A1ASX, DMS, SO4
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Identification Of Multiple Ligand Hotspots On Sos2, Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.79 Å Release Date: 2025-02-05 Classification: SIGNALING PROTEIN Ligands: A1ASW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-02-05
Ligands: A1ASW
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Sos2 In Complex With Compound 11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.06 Å Release Date: 2025-02-05 Classification: HYDROLASE Ligands: A1IL1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-02-05
Ligands: A1IL1
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Discovery Of A Kras G12V Inhibitor In Vivo Tool Compound Starting From An Hsqc-Nmr Based Fragment Hit
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2022-11-09 Classification: SIGNALING PROTEIN Ligands: 2XO, GDP, MG, LX6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-09
Ligands: 2XO, GDP, MG, LX6
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Crystal Structure Of Kras-G12C In Complex With Compound 23 (Bi-0474)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.12 Å Release Date: 2022-11-09 Classification: ONCOPROTEIN Ligands: GDP, MG, LXD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-09
Ligands: GDP, MG, LXD
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Crystal Structure Of Kras-G12C In Complex With Compound 12
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.41 Å Release Date: 2022-11-09 Classification: ONCOPROTEIN Ligands: GDP, MG, LXK, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-09
Ligands: GDP, MG, LXK, SO4
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Crystal Structure Of Bit-Blocked Kras-G12V-S39C In Complex With Compound 20A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.63 Å Release Date: 2022-11-09 Classification: ONCOPROTEIN Ligands: GDP, 2XO, MG, LXU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-09
Ligands: GDP, 2XO, MG, LXU
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Ras:Sos:Ras In Complex With A Small Molecule Activator
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.48 Å Release Date: 2019-03-27 Classification: SIGNALING PROTEIN Ligands: MG, GNP, FVV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-03-27
Ligands: MG, GNP, FVV
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Ras:Sos:Ras In Complex With A Small Molecule Activator
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.73 Å Release Date: 2019-02-06 Classification: SIGNALING PROTEIN Ligands: GNP, MG, FMT, FFS, GOL, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-06
Ligands: GNP, MG, FMT, FFS, GOL, NA
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Ras:Sos:Ras In Complex With A Small Molecule Activator
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2019-02-06 Classification: SIGNALING PROTEIN Ligands: GNP, MG, FFV, FMT, GOL, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-06
Ligands: GNP, MG, FFV, FMT, GOL, NA
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Ras:Sos:Ras In Complex With A Small Molecule Activator
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.73 Å Release Date: 2019-02-06 Classification: SIGNALING PROTEIN Ligands: GNP, MG, FFY, FMT, GOL, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-06
Ligands: GNP, MG, FFY, FMT, GOL, NA
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Ras:Sos:Ras In Complex With A Small Molecule Activator
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2018-10-24 Classification: SIGNALING PROTEIN Ligands: GNP, MG, EC4, FMT, GOL, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-24
Ligands: GNP, MG, EC4, FMT, GOL, NA
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Ras:Sos:Ras In Complex With A Small Molecule Activator
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2018-10-24 Classification: SIGNALING PROTEIN Ligands: GNP, MG, EAS, FMT, GOL, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-24
Ligands: GNP, MG, EAS, FMT, GOL, NA
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Ras:Sos:Ras In Complex With A Small Molecule Activator
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2018-10-24 Classification: SIGNALING PROTEIN Ligands: GNP, MG, EAV, FMT, GOL, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-24
Ligands: GNP, MG, EAV, FMT, GOL, NA
