Search Count: 385
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Synthesis And Biological Evaluation Of Novel Selective Androgen Receptor Modulators (Sarms). Part Ii: Optimization Of 4-(Pyrrolidin-1-Yl)Benzonitrile Derivatives
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2017-04-26 Classification: HORMONE RECEPTOR Ligands: GOL, 77T |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-04-26
Ligands: GOL, 77T
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Synthesis And Biological Evaluation Of Novel Selective Androgen Receptor Modulators (Sarms). Part Ii: Optimization Of 4-(Pyrrolidin-1-Yl)Benzonitrile Derivatives
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.71 Å Release Date: 2017-04-26 Classification: HORMONE RECEPTOR Ligands: GOL, 77U |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-04-26
Ligands: GOL, 77U
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Crystal Structure Of The Androgen Receptor Ligand Binding Domain (Lbd) With Dht And A Peptide Derived From Its Physiological Coactivator Ara70
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2005-01-25 Classification: HORMONE/GROWTH FACTOR Ligands: DHT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-01-25
Ligands: DHT
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Structural Basis For The Glucocorticoid Response In A Mutant Human Androgen Receptor (Arccr) Derived From An Androgen-Independent Prostate Cancer
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2003-01-16 Classification: ANDROGEN RECEPTOR Ligands: ZK5, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2003-01-16
Ligands: ZK5, PO4
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Crystal Structure Of The Human Androgen Receptor Ligand Binding Domain Bound With An Androgen Receptor Nh2-Terminal Peptide, Ar20-30, And R1881
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2004-11-16 Classification: TRANSCRIPTION Ligands: R18 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2004-11-16
Ligands: R18
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Human Androgen Receptor Ligand Binding In Complex With The Ligand Metribolone (R1881)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2001-06-14 Classification: ANDROGEN RECEPTOR Ligands: R18 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2001-06-14
Ligands: R18
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Crystal Structure Of The Human Androgen Receptor T877A Mutant Ligand-Binding Domain With Cyproterone Acetate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2007-03-27 Classification: HORMONE RECEPTOR Ligands: CA4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-03-27
Ligands: CA4
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Androgen Receptor With Small Molecule
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2007-09-25 Classification: HORMONE RECEPTOR Ligands: SO4, DHT, T3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-09-25
Ligands: SO4, DHT, T3
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Androgen Receptor With Small Molecule
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.58 Å Release Date: 2007-09-25 Classification: HORMONE RECEPTOR Ligands: DHT, T3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-09-25
Ligands: DHT, T3
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Androgen Receptor Lbd With Small Molecule
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.49 Å Release Date: 2007-09-25 Classification: HORMONE RECEPTOR Ligands: DHT, 4HY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-09-25
Ligands: DHT, 4HY
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Crystal Structure Of Human Androgen Receptor Ligand Binding Domain In Complex With Tetrahydrogestrinone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2006-05-16 Classification: Hormone/Growth Factor Receptor Ligands: SO4, 17H, DTT, EPE, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-05-16
Ligands: SO4, 17H, DTT, EPE, GOL
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Androgen Receptor Lbd With Small Molecule
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.76 Å Release Date: 2007-09-25 Classification: HORMONE RECEPTOR Ligands: SO4, DHT, 4HY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-09-25
Ligands: SO4, DHT, 4HY
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Androgen Receptor Lbd With Small Molecule
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2007-09-25 Classification: HORMONE RECEPTOR Ligands: SO4, DHT, RB1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-09-25
Ligands: SO4, DHT, RB1
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Androgen Receptor Lbd With Small Molecule
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2007-09-25 Classification: HORMONE RECEPTOR Ligands: SO4, DHT, ICO, K10 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-09-25
Ligands: SO4, DHT, ICO, K10
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Androgen Receptor Lbd With Small Molecule
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.12 Å Release Date: 2007-09-25 Classification: HORMONE RECEPTOR Ligands: DHT, 4HY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-09-25
Ligands: DHT, 4HY
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Androgen Receptor Lbd With Small Molecule
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2007-09-25 Classification: HORMONE RECEPTOR Ligands: SO4, DHT, NK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-09-25
Ligands: SO4, DHT, NK
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Androgen Receptor Lbd With Small Molecule
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.03 Å Release Date: 2007-09-25 Classification: HORMONE RECEPTOR Ligands: SO4, DHT, 2MI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-09-25
Ligands: SO4, DHT, 2MI
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Crystal Structure Of Human Androgen Receptor Ligand Binding Domain In Complex With Dihydrotestosterone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2006-05-16 Classification: Hormone/Growth Factor Receptor Ligands: SO4, DHT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-05-16
Ligands: SO4, DHT
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Crystal Structure Of Human Androgen Receptor Ligand Binding Domain In Complex With Testosterone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.64 Å Release Date: 2006-05-16 Classification: Hormone/Growth Factor Receptor Ligands: SO4, TES, DTT, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-05-16
Ligands: SO4, TES, DTT, GOL
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Crystal Structure Of The Androgen Receptor Ligand Binding Domain In Complex With 5-(2-Fluoro-4-Hydroxyphenyl)-1-Methyl-1H-Pyrrole-2-Carbonitrile
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2018-03-14 Classification: HORMONE RECEPTOR Ligands: 9FG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-14
Ligands: 9FG
