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5T8E image
Synthesis And Biological Evaluation Of Novel Selective Androgen Receptor Modulators (Sarms). Part Ii: Optimization Of 4-(Pyrrolidin-1-Yl)Benzonitrile Derivatives
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.71 Å Release Date: 2017-04-26
Classification: HORMONE RECEPTOR
Ligands: GOL, 77U

5T8J image
Synthesis And Biological Evaluation Of Novel Selective Androgen Receptor Modulators (Sarms). Part Ii: Optimization Of 4-(Pyrrolidin-1-Yl)Benzonitrile Derivatives
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.70 Å Release Date: 2017-04-26
Classification: HORMONE RECEPTOR
Ligands: GOL, 77T

1T5Z image
Crystal Structure Of The Androgen Receptor Ligand Binding Domain (Lbd) With Dht And A Peptide Derived From Its Physiological Coactivator Ara70
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.30 Å Release Date: 2005-01-25
Classification: HORMONE/GROWTH FACTOR
Ligands: DHT

1GS4 image
Structural Basis For The Glucocorticoid Response In A Mutant Human Androgen Receptor (Arccr) Derived From An Androgen-Independent Prostate Cancer
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.95 Å Release Date: 2003-01-16
Classification: ANDROGEN RECEPTOR
Ligands: ZK5, PO4

1XOW image
Crystal Structure Of The Human Androgen Receptor Ligand Binding Domain Bound With An Androgen Receptor Nh2-Terminal Peptide, Ar20-30, And R1881
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.80 Å Release Date: 2004-11-16
Classification: TRANSCRIPTION
Ligands: R18

1E3G image
Human Androgen Receptor Ligand Binding In Complex With The Ligand Metribolone (R1881)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.40 Å Release Date: 2001-06-14
Classification: ANDROGEN RECEPTOR
Ligands: R18

2OZ7 image
Crystal Structure Of The Human Androgen Receptor T877A Mutant Ligand-Binding Domain With Cyproterone Acetate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.80 Å Release Date: 2007-03-27
Classification: HORMONE RECEPTOR
Ligands: CA4

2PIW image
Androgen Receptor With Small Molecule
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.58 Å Release Date: 2007-09-25
Classification: HORMONE RECEPTOR
Ligands: DHT, T3

2PIV image
Androgen Receptor With Small Molecule
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.95 Å Release Date: 2007-09-25
Classification: HORMONE RECEPTOR
Ligands: SO4, DHT, T3

2PKL image
Androgen Receptor Lbd With Small Molecule
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.49 Å Release Date: 2007-09-25
Classification: HORMONE RECEPTOR
Ligands: DHT, 4HY

2AMB image
Crystal Structure Of Human Androgen Receptor Ligand Binding Domain In Complex With Tetrahydrogestrinone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.75 Å Release Date: 2006-05-16
Classification: Hormone/Growth Factor Receptor
Ligands: SO4, 17H, DTT, EPE, GOL

2PIU image
Androgen Receptor Lbd With Small Molecule
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.12 Å Release Date: 2007-09-25
Classification: HORMONE RECEPTOR
Ligands: DHT, 4HY

2PIP image
Androgen Receptor Lbd With Small Molecule
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.80 Å Release Date: 2007-09-25
Classification: HORMONE RECEPTOR
Ligands: SO4, DHT, ICO, K10

2PIQ image
Androgen Receptor Lbd With Small Molecule
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.40 Å Release Date: 2007-09-25
Classification: HORMONE RECEPTOR
Ligands: SO4, DHT, RB1

2PIT image
Androgen Receptor Lbd With Small Molecule
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.76 Å Release Date: 2007-09-25
Classification: HORMONE RECEPTOR
Ligands: SO4, DHT, 4HY

2PIR image
Androgen Receptor Lbd With Small Molecule
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.10 Å Release Date: 2007-09-25
Classification: HORMONE RECEPTOR
Ligands: SO4, DHT, NK

2PIO image
Androgen Receptor Lbd With Small Molecule
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.03 Å Release Date: 2007-09-25
Classification: HORMONE RECEPTOR
Ligands: SO4, DHT, 2MI

2AMA image
Crystal Structure Of Human Androgen Receptor Ligand Binding Domain In Complex With Dihydrotestosterone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.90 Å Release Date: 2006-05-16
Classification: Hormone/Growth Factor Receptor
Ligands: SO4, DHT

2AM9 image
Crystal Structure Of Human Androgen Receptor Ligand Binding Domain In Complex With Testosterone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.64 Å Release Date: 2006-05-16
Classification: Hormone/Growth Factor Receptor
Ligands: SO4, TES, DTT, GOL

5VO4 image
Crystal Structure Of The Androgen Receptor Ligand Binding Domain In Complex With 5-(2-Fluoro-4-Hydroxyphenyl)-1-Methyl-1H-Pyrrole-2-Carbonitrile
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.35 Å Release Date: 2018-03-14
Classification: HORMONE RECEPTOR
Ligands: 9FG
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