Search Count: 19
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Ncs-1 Bound To Fda Ligand 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2026-04-08 Classification: METAL BINDING PROTEIN Ligands: CA, 0LI, NA, ACY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-04-08
Ligands: CA, 0LI, NA, ACY
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The Catalytic Domain Of Mekk2 In Complex With Ponatinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2025-11-26 Classification: SIGNALING PROTEIN Ligands: 0LI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-11-26
Ligands: 0LI
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C-Kit Kinase Domain In Complex With Ponatinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2025-09-03 Classification: TRANSFERASE Ligands: 0LI, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-03
Ligands: 0LI, CL
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Cryo-Em Structure Of Lrrk2 Bound To Type Ii Inhibitor Ponatinib
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2024-01-31 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 0LI, GDP |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2024-01-31
Ligands: 0LI, GDP
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Src Kinase Domain In Complex With Ponatinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.49 Å Release Date: 2022-06-22 Classification: ONCOPROTEIN Ligands: 0LI, TRS, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-06-22
Ligands: 0LI, TRS, GOL
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C-Src In Complex With Ponatinib
Organism: Gallus gallus
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2022-03-02 Classification: ONCOPROTEIN Ligands: 0LI |
Organism: Gallus gallus
Method: X-RAY DIFFRACTION
Release Date: 2022-03-02
Ligands: 0LI
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The Co-Crystal Structure Of Braf(V600E) With Ponatinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.11 Å Release Date: 2020-09-23 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0LI, SO4, NH4, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-09-23
Ligands: 0LI, SO4, NH4, EDO
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The Ror1 Pseudokinase Domain Bound To Ponatinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.94 Å Release Date: 2020-01-22 Classification: SIGNALING PROTEIN Ligands: 0LI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-22
Ligands: 0LI
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Irak4 In Complex With Ponatinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.41 Å Release Date: 2019-02-20 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0LI, SO4, CO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-20
Ligands: 0LI, SO4, CO
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Fgfr1 In Complex With Ponatinib (Co-Crystallisation).
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.33 Å Release Date: 2014-12-10 Classification: TRANSFERASE Ligands: SO4, EDO, 0LI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-10
Ligands: SO4, EDO, 0LI
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Fgfr1 In Complex With Ponatinib.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.12 Å Release Date: 2014-12-10 Classification: TRANSFERASE Ligands: EDO, 0LI, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-10
Ligands: EDO, 0LI, SO4
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Fgfr4 In Complex With Ponatinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2014-12-03 Classification: TRANSFERASE Ligands: SO4, 0LI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-03
Ligands: SO4, 0LI
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Crystal Structure Of The Tyrosine Kinase Domain Of Fgf Receptor 4 In Complex With Ponatinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2014-10-29 Classification: Transferase/transferase inhibitor Ligands: SO4, 0LI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-10-29
Ligands: SO4, 0LI
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Crystal Structure Of Kit In Complex With Ponatinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2014-10-08 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0LI, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-10-08
Ligands: 0LI, PO4
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Structural Analysis Of The Human Fibroblast Growth Factor Receptor 4 Kinase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2014-09-24 Classification: TRANSFERASE Ligands: 0LI, EDO, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-09-24
Ligands: 0LI, EDO, PO4
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Structure Of The Kinase Domain Of Human Ripk2 In Complex With Ponatinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.75 Å Release Date: 2013-10-16 Classification: TRANSFERASE Ligands: 0LI, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-10-16
Ligands: 0LI, EDO
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Structure Of The Ddr1 Kinase Domain In Complex With Ponatinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.92 Å Release Date: 2013-05-01 Classification: TRANSFERASE Ligands: 0LI, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-01
Ligands: 0LI, EDO
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Crystal Structure Of Abl Kinase Domain Bound With A Dfg-Out Inhibitor Ap24534
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2010-12-15 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0LI |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2010-12-15
Ligands: 0LI
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Ap24534, A Pan-Bcr-Abl Inhibitor For Chronic Myeloid Leukemia, Potently Inhibits The T315I Mutant And Overcomes Mutation-Based Resistance
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2009-11-03 Classification: TRANSFERASE Ligands: 0LI |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2009-11-03
Ligands: 0LI
