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Crystal Structure Of Human Nuak1-Mark3 Kinase Domain Chimera Bound With Azepane (R)-#50 Small Molecule Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2024-11-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: X5I, EDO, CL, BEZ |
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Crystal Structure Of Human Nuak1-Mark3 Kinase Domain Chimera Bound With Small Molecule Inhibitor #10
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2024-10-23 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: EDO, NI, X4W |
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Crystal Structure Of Human Nuak1-Mark3 Kinase Domain Chimera Bound With Small Molecule Inhibitor #65
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2024-10-23 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: X3Q, EDO |
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Crystal Structure Of Human Nuak1-Mark3 (7 Mutations) Kinase Domain Chimera Bound With Small Molecule Inhibitor #31
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2024-10-23 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: X5N, EDO |
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Crystal Structure Of Human Nuak1-Mark3 (6 Mutations) Kinase Domain Chimera Bound With Small Molecule Inhibitor #31
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2024-10-23 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: X4H, EDO |
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Structure Of Plasmepsin X (Pm10, Pmx) From Plasmodium Falciparum 3D7 In Complex With Ucb7362
Organism: Plasmodium falciparum 3d7
Method: X-RAY DIFFRACTION Resolution:2.85 Å Release Date: 2022-10-19 Classification: HYDROLASE Ligands: TWU |






