Search Count: 23
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Crystal Structure Of Bptf Bromodomain In Complex With 4-Chloro-5-{4-[(Dimethylamino)Methyl]Anilino}-2-Methylpyridazin-3(2H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.39 Å Release Date: 2022-08-24 Classification: GENE REGULATION/INHIBITOR Ligands: 7WE, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-24
Ligands: 7WE, EDO
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Crystal Structure Of Bptf Bromodomain In Complex With 4-Chloro-2-Methyl-5-[(1,2,3,4-Tetrahydroisoquinolin-7-Yl)Amino]Pyridazin-3(2H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.58 Å Release Date: 2022-08-24 Classification: GENE REGULATION/INHIBITOR Ligands: 7WN, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-24
Ligands: 7WN, EDO
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Crystal Structure Of Bptf Bromodomain In Complex With 5-[4-(Aminomethyl)Anilino]-4-Chloro-2-Methylpyridazin-3(2H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.73 Å Release Date: 2022-08-24 Classification: GENE REGULATION/INHIBITOR Ligands: 7WZ, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-24
Ligands: 7WZ, CA
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Crystal Structure Of Bptf Bromodomain In Complex With 4-Chloro-2-Methyl-5-[(1,2,3,4-Tetrahydroisoquinolin-6-Yl)Amino]Pyridazin-3(2H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2022-08-24 Classification: GENE REGULATION/INHIBITOR Ligands: 7XE, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-24
Ligands: 7XE, CA
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Crystal Structure Of Bptf Bromodomain In Complex With Inhibitor Pdy-3-077
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.66 Å Release Date: 2022-08-10 Classification: GENE REGULATION/INHIBITOR Ligands: P2L, DMS, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-10
Ligands: P2L, DMS, EDO
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Crystal Structure Of Bptf Bromodomain In Complex With Inhibitor Hz-03-112
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.39 Å Release Date: 2022-08-10 Classification: GENE REGULATION/INHIBITOR Ligands: Y9P, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-10
Ligands: Y9P, EDO
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Crystal Structure Of Bptf Bromodomain In Complex With Inhibitor Pdy-3-093
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.44 Å Release Date: 2022-08-10 Classification: GENE REGULATION/INHIBITOR Ligands: YC4, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-10
Ligands: YC4, EDO
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Crystal Structure Of Bptf Bromodomain In Complex With Inhibitor Hz-01-105
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2022-08-10 Classification: GENE REGULATION/INHIBITOR Ligands: DMS, YBV, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-10
Ligands: DMS, YBV, EDO
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Crystal Structure Of Bptf Bromodomain In Complex With Cb02-092
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2022-02-16 Classification: GENE REGULATION Ligands: YOV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-02-16
Ligands: YOV
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Cocrystal Of Brd4(D1) With N,N-Dimethyl-2-[(3R)-3-(5-{2-[2-Methyl-5-(Propan-2-Yl)Phenoxy]Pyrimidin-4-Yl}-4-[4-(Trifluoromethyl)Phenyl]-1H-Imidazol-1-Yl)Pyrrolidin-1-Yl]Ethan-1-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2022-01-19 Classification: GENE REGULATION/INHIBITOR Ligands: EDO, 2IR, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-19
Ligands: EDO, 2IR, CL
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Crystal Structure Of Brd4(D1) With 4-[4-(4-Bromophenyl)-1-(Piperidin-4-Yl)-1H-Imidazol-5-Yl]-N-(3,5-Dimethylphenyl)Pyrimidin-2-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.41 Å Release Date: 2022-01-19 Classification: GENE REGULATION/INHIBITOR Ligands: EDO, 7ZB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-19
Ligands: EDO, 7ZB
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Crystal Of Brd4(D1) With 2-[(3S)-3-{5-[2-(3,5-Dimethylphenoxy)Pyrimidin-4-Yl]-4-(4-Iodophenyl)-1H-Imidazol-1-Yl}Pyrrolidin-1-Yl]Ethan-1-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.43 Å Release Date: 2022-01-19 Classification: GENE REGULATION/INHIBITOR Ligands: EDO, 7ZT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-19
Ligands: EDO, 7ZT
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Crystal Of Brd4(D1) With 2-[(3R)-3-{5-[2-(3,5-Dimethylphenoxy)Pyrimidin-4-Yl]-4-(4-Iodophenyl)-1H-Imidazol-1-Yl}Pyrrolidin-1-Yl]Ethan-1-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.68 Å Release Date: 2022-01-19 Classification: GENE REGULATION/INHIBITOR Ligands: 7ZK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-19
Ligands: 7ZK
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Crystal Structure Of Bptf Bromodomain Labelled With 5-Fluoro-Tryptophan
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.06 Å Release Date: 2021-07-28 Classification: GENE REGULATION |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-28
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X-Ray Crystal Structure Of Human Brd4(D1) In Complex With 2-(4-{5-[6-(2,5-Dibromophenoxy)Pyridin-2-Yl]-4-Methyl-1H-1,2,3-Triazol-1-Yl}Piperidin-1-Yl)-N,N-Dimethylethan-1-Amine (Compound 26)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.32 Å Release Date: 2021-07-28 Classification: GENE REGULATION/INHIBITOR Ligands: EDO, ZHV, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-28
Ligands: EDO, ZHV, CL
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X-Ray Crystal Structure Of Human Brd4(D1) In Complex With 2-(4-{5-[6-(3,5-Dimethylphenoxy)Pyridin-2-Yl]-4-Methyl-1H-1,2,3-Triazol-1- Yl}Piperidin-1-Yl)-N,N-Dimethylethan-1-Amine (Dw34)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.20 Å Release Date: 2021-07-28 Classification: GENE REGULATION/INHIBITOR Ligands: EDO, ZHS, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-28
Ligands: EDO, ZHS, NA
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X-Ray Crystal Structure Of Human Brd4(D1) In Complex With 2-(2,5-Dibromophenoxy)-6-[4-Methyl-1-(Piperidin-4-Yl)-1H-1,2,3-Triazol-5-Yl]Pyridine (Compound 23)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.26 Å Release Date: 2021-07-28 Classification: GENE REGULATION/INHIBITOR Ligands: ZHM, EDO, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-28
Ligands: ZHM, EDO, CL
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Crystal Structure Of The Bromodomain (Bd) Of Human Bromodomain And Phd Finger-Containing Transcription Factor (Bptf) Bound To Gsk4027
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2020-12-09 Classification: GENE REGULATION Ligands: 9ST, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-09
Ligands: 9ST, EDO
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Crystal Structure Of The Bromodomain (Bd) Of Human Bromodomain And Phd Finger-Containing Transcription Factor (Bptf) Bound To Compound 4 (Skt1174)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.23 Å Release Date: 2020-12-09 Classification: GENE REGULATION Ligands: VYM, EDO, GOL, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-09
Ligands: VYM, EDO, GOL, CL
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Crystal Structure Of The Bromodomain (Bd) Of Human Bromodomain And Phd Finger-Containing Transcription Factor (Bptf) Bound To Compound 6 (Hz01052)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.71 Å Release Date: 2020-12-09 Classification: GENE REGULATION Ligands: WCV, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-09
Ligands: WCV, EDO