Search Count: 46
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Structure Of Kras G12C Bound To Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.84 Å Release Date: 2026-03-11 Classification: ONCOPROTEIN Ligands: A1CQ2, GDP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-03-11
Ligands: A1CQ2, GDP, MG
 |
Structure Of Kras G12C Bound To Divarasib (Gdc6036)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.17 Å Release Date: 2026-03-11 Classification: ONCOPROTEIN Ligands: GDP, MG, DMS, EDO, A1AWR, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-03-11
Ligands: GDP, MG, DMS, EDO, A1AWR, PEG
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Crystal Structure Of Htdo2 Bound To Inhibitor Gne1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.18 Å Release Date: 2020-05-06 Classification: OXIDOREDUCTASE/Inhibitor Ligands: HEM, QVY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-05-06
Ligands: HEM, QVY
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Structure Of The Human Jak1 Kinase Domain With Compound 15
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.64 Å Release Date: 2019-04-24 Classification: IMMUNE SYSTEM Ligands: KEJ, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-04-24
Ligands: KEJ, GOL
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Structure Of The Human Jak1 Kinase Domain With Compound 21
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2019-04-24 Classification: IMMUNE SYSTEM Ligands: KEP, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-04-24
Ligands: KEP, GOL
 |
Structure Of The Human Jak1 Kinase Domain With Compound 20
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.27 Å Release Date: 2019-04-24 Classification: IMMUNE SYSTEM Ligands: KES, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-04-24
Ligands: KES, GOL
 |
Structure Of The Human Jak1 Kinase Domain With Compound 39
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.33 Å Release Date: 2019-04-24 Classification: IMMUNE SYSTEM Ligands: GOL, KEV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-04-24
Ligands: GOL, KEV
 |
Structure Of The Human Jak1 Kinase Domain With Compound 38
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.81 Å Release Date: 2019-04-24 Classification: IMMUNE SYSTEM Ligands: KEY, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-04-24
Ligands: KEY, GOL
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Structure Of The Human Jak1 Kinase Domain With Compound 56
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.69 Å Release Date: 2019-04-24 Classification: IMMUNE SYSTEM Ligands: KF1, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-04-24
Ligands: KF1, GOL
 |
Structure Of The Human Jak1 Kinase Domain With Compound 54
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.78 Å Release Date: 2019-04-24 Classification: IMMUNE SYSTEM Ligands: KF4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-04-24
Ligands: KF4, GOL
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Structure Of The Human Glun1/Glun2A Lbd In Complex With Compound 2 (Gne9178)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2016-11-30 Classification: TRANSPORT PROTEIN Ligands: ACT, GLU, 7H0, CA, GLY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-30
Ligands: ACT, GLU, 7H0, CA, GLY
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Structure Of The Human Glun1/Glun2A Lbd In Complex With Compound 9 (Gne3500)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.48 Å Release Date: 2016-11-30 Classification: TRANSPORT PROTEIN Ligands: GLU, 7H2, GLY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-30
Ligands: GLU, 7H2, GLY
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Crystal Structure Of Nicotinamide Phosphoribosyltransferase (Nampt) In Complex With Inhibitors 37
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2016-08-31 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6TA, PO4, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-08-31
Ligands: 6TA, PO4, EDO
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Structure Of The Human Glun1/Glun2A Lbd In Complex With Gne0723
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.44 Å Release Date: 2016-07-13 Classification: TRANSPORT PROTEIN Ligands: ACT, GLU, 6RV, GLY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-07-13
Ligands: ACT, GLU, 6RV, GLY
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Structure Of The Human Glun1/Glun2A Lbd In Complex With 7-{[Ethyl(4-Fluorophenyl)Amino]Methyl}-N,2-Dimethyl-5-Oxo-5H-[1,3]Thiazolo[3,2-A]Pyrimidine-3-Carboxamide (Compound 19)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.86 Å Release Date: 2016-03-16 Classification: TRANSPORT PROTEIN Ligands: GLU, GLY, 67H |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-03-16
Ligands: GLU, GLY, 67H
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Structure Of The Human Glun1/Glun2A Lbd In Complex With N-Ethyl-7-{[2-Fluoro-3-(Trifluoromethyl)Phenyl]Methyl}-2-Methyl-5-Oxo-5H-[1,3]Thiazolo[3,2-A]Pyrimidine-3-Carboxamide (Compound 29)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.12 Å Release Date: 2016-03-16 Classification: TRANSPORT PROTEIN Ligands: CA, GLU, 67J, EPE, GLY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-03-16
Ligands: CA, GLU, 67J, EPE, GLY
 |
Itk Kinase Domain In Complex With Compound 1 N-{1-[(1,1-Dioxo-1-Thian-2-Yl)(Phenyl)Methyl]-1H- Pyrazol-4-Yl}-5,5-Difluoro-5A-Methyl-1H,4H,4Ah,5H,5Ah,6H-Cyclopropa[F]Indazole-3-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2015-04-29 Classification: TRANSFERASE/INHIBITOR Ligands: 3P6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-29
Ligands: 3P6
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The Crystal Structure Of Human Nicotinamide Phosphoribosyltransferase (Nampt) In Complex With N-(4-{(S)-[1-(2-Methylpropyl)Piperidin-4-Yl]Sulfinyl}Benzyl)Furo[2,3-C]Pyridine-2-Carboxamide Inhibitor (Compound 21)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2015-02-11 Classification: Transferase/Transferase inhibitor Ligands: 3TQ, PO4, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-02-11
Ligands: 3TQ, PO4, EDO
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Itk Kinase Domain With Compound Gne-9822
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.71 Å Release Date: 2014-07-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 2W6, P4G |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-02
Ligands: 2W6, P4G
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Aurora A Kinase Domain With Compound 2 (N-[1-(3-Cyanobenzyl)-1H-Pyrazol-4-Yl]-6-(1H-Pyrazol-4-Yl)-1H-Indazole-3-Carboxamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2014-07-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 2VU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-02
Ligands: 2VU