Search Count: 30
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Crystal Structure Of Kat6A In Complex With Inhibitor Ctx-648 (Pf-9363)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.58 Å Release Date: 2023-07-05 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: R7L, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-07-05
Ligands: R7L, ZN
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Crystal Structure Of Bovine Heart Cytochrome C Oxidase, Apo Structure With Dmso
Organism: Bos taurus
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2022-12-21 Classification: OXIDOREDUCTASE Ligands: HEA, CU, MG, NA, PER, PGV, TGL, CUA, CDL, CHD, PEK, PSC, ZN, DMU |
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Crystal Structure Of Bovine Heart Cytochrome C Oxidase, The Structure Complexed With An Allosteric Inhibitor T113
Organism: Bos taurus
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2022-12-21 Classification: OXIDOREDUCTASE Ligands: HEA, CU, MG, NA, PER, TGL, J6X, CUA, CHD, PSC, PEK, PGV, CDL, DMU, ZN |
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Cryo-Em Structure Of Cytochrome Bo3 From Escherichia Coli, Apo Structure With Dmso
Organism: Escherichia coli
Method: ELECTRON MICROSCOPY Release Date: 2022-12-21 Classification: OXIDOREDUCTASE Ligands: HEO, HEM, CU, PEE, UNX |
Organism: Escherichia coli
Method: ELECTRON MICROSCOPY
Release Date: 2022-12-21
Ligands: HEO, HEM, CU, PEE, UNX
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Cryo-Em Structure Of Cytochrome Bo3 From Escherichia Coli, The Structure Complexed With An Allosteric Inhibitor N4
Organism: Escherichia coli
Method: ELECTRON MICROSCOPY Release Date: 2022-12-21 Classification: OXIDOREDUCTASE Ligands: HEO, HEM, CU, PEE, JYR, UNX |
Organism: Escherichia coli
Method: ELECTRON MICROSCOPY
Release Date: 2022-12-21
Ligands: HEO, HEM, CU, PEE, JYR, UNX
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Prmt5:Mep50 Complexed With Inhibitor Pf-06939999
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.49 Å Release Date: 2021-11-17 Classification: TRANSFERASE/Transcription Ligands: ZR1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-11-17
Ligands: ZR1
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Prmt5:Mep50 Complexed With Inhibitor Pf-06855800
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.71 Å Release Date: 2021-11-17 Classification: Transferase/Transcription Ligands: ZR4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-11-17
Ligands: ZR4
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Prmt5:Mep50 Complexed With Adenosine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.41 Å Release Date: 2021-11-17 Classification: TRANSFERASE/Transcription Ligands: ADN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-11-17
Ligands: ADN
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Prmt5(M420T Mutant):Mep50 Complexed With Inhibitor Pf-06855800
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2021-11-17 Classification: TRANSFERASE/Transcription Ligands: ZR4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-11-17
Ligands: ZR4
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Prmt5(M420T Mutant):Mep50 Complexed With Inhibitor Pf-06939999
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2021-11-17 Classification: transferase/Transcription Ligands: ZR1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-11-17
Ligands: ZR1
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Structure Of Hs/Acprc2 In Complex With 5,8-Dichloro-2-[(4-Methoxy-6-Methyl-2-Oxo-1,2-Dihydropyridin-3-Yl)Methyl]-7-[(R)-Methoxy(Oxetan-3-Yl)Methyl]-3,4-Dihydroisoquinolin-1(2H)-One
Organism: Anolis carolinensis, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.81 Å Release Date: 2017-12-27 Classification: Transferase/Transferase Inhibitor Ligands: ZN, CJD |
Organism: Anolis carolinensis, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-27
Ligands: ZN, CJD
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Structure Of Hs/Acprc2 In Complex With 5,8-Dichloro-7-(3,5-Dimethyl-1,2-Oxazol-4-Yl)-2-[(4,6-Dimethyl-2-Oxo-1,2-Dihydropyridin-3-Yl)Methyl]-3,4-Dihydroisoquinolin-1(2H)-One
Organism: Anolis carolinensis, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.05 Å Release Date: 2017-12-27 Classification: METAL BINDING PROTEIN Ligands: ZN, CJG |
Organism: Anolis carolinensis, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-27
Ligands: ZN, CJG
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X-Ray Structure Of C-Met Kinase In Complex With Inhibitor 6-((6-(4- Fluorophenyl)-(1,2,4)Triazolo(4,3-B)(1,2,4)Triazin-3-Yl)Methyl) Quinoline.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2013-11-27 Classification: TRANSFERASE Ligands: 6XE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-11-27
Ligands: 6XE
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X-Ray Structure Of C-Met Kinase In Complex With Inhibitor (S)-6-(1-(6- (1-Methyl-1H-Pyrazol-4-Yl)-(1,2,4)Triazolo(4,3-B)Pyridazin-3-Yl)Ethyl) Quinoline.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2013-11-27 Classification: TRANSFERASE Ligands: W9Z |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-11-27
Ligands: W9Z
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X-Ray Structure Of C-Met Kinase In Complex With Inhibitor (S)-3-(1-(1H-Pyrrolo(2,3-B)Pyridin-3-Yl)Ethyl)-N-Isopropyl-(1,2,4)Triazolo(4,3- B)Pyridazin-6-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2013-11-27 Classification: TRANSFERASE Ligands: 5TF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-11-27
Ligands: 5TF
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Crystal Structure Of C-Met Kinase Domain In Complex With 4-(3-((1H- Pyrrolo(2,3-B)Pyridin-3-Yl)Methyl)-(1,2,4)Triazolo(4,3-B)(1,2,4) Triazin-6-Yl)Benzonitrile
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2012-09-26 Classification: TRANSFERASE Ligands: 4K0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-09-26
Ligands: 4K0
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Crystal Structure Of C-Met Kinase Domain In Complex With 4-((6-(4- Fluorophenyl)-(1,2,4)Triazolo(4,3-B)(1,2,4)Triazin-3-Yl)Methyl)Phenol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2012-09-26 Classification: TRANSFERASE Ligands: F47 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-09-26
Ligands: F47
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Crystal Structure Of C-Met Kinase Domain In Complex With N'-((3Z)-4- Chloro-7-Methyl-2-Oxo-1,2-Dihydro-3H-Indol-3-Ylidene)-2-(4- Hydroxyphenyl)Propanohydrazide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.87 Å Release Date: 2011-09-14 Classification: TRANSFERASE Ligands: 6XP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-09-14
Ligands: 6XP
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X-Ray Structure Of Pf-04217903 Bound To The Kinase Domain Of C-Met
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2011-08-31 Classification: TRANSFERASE Ligands: KRW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-08-31
Ligands: KRW
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Optimization Of Potent, Selective, And Orally Bioavailable Pyrrolodinopyrimidine-Containing Inhibitors Of Heat Shock Protein 90. Identification Of Development Candidate 2-Amino-4-{4-Chloro-2-[2-(4-Fluoro-1H-Pyrazol-1-Yl)Ethoxy]-6-Methylphenyl}-N-(2,2-Difluoropropyl)-5,7-Dihydro-6H-Pyrrolo[3,4-D]Pyrimidine-6-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2011-04-27 Classification: Chaperone/Chaperone inhibitor Ligands: WOE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-04-27
Ligands: WOE
