Search Count: 14
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Crystal Structure Of Human Akt2 In Complex With Gsk690693
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2008-10-21 Classification: TRANSFERASE INHIBITOR Ligands: G93 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-10-21
Ligands: G93
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Crystal Structure Of Cathepsin K Complexed With 7-Methyl-Substituted Azepan-3-One Compound
Organism: Macaca mulatta
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2007-01-30 Classification: HYDROLASE Ligands: ILI |
Organism: Macaca mulatta
Method: X-RAY DIFFRACTION
Release Date: 2007-01-30
Ligands: ILI
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Crystal Structure Of The Cysteine Protease Human Cathepsin K In Complex With A Covalent Azepanone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2003-01-14 Classification: HYDROLASE Ligands: 750 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2003-01-14
Ligands: 750
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Crystal Structure Of The Cysteine Protease Human Cathepsin K In Complex With A Covalent Azepanone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2003-01-14 Classification: HYDROLASE Ligands: 2CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2003-01-14
Ligands: 2CA
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Use Of Papain As A Model For The Structure-Based Design Of Cathepsin K Inhibitors. Crystal Structures Of Two Papain Inhibitor Complexes Demonstrate Binding To S'-Subsites.
Organism: Carica papaya
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 1999-08-16 Classification: HYDROLASE Ligands: SBA |
Organism: Carica papaya
Method: X-RAY DIFFRACTION
Release Date: 1999-08-16
Ligands: SBA
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Use Of Papain As A Model For The Structure-Based Design Of Cathepsin K Inhibitors. Crystal Structures Of Two Papain Inhibitor Complexes Demonstrate Binding To S'-Subsites.
Organism: Carica papaya
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 1999-08-12 Classification: HYDROLASE Ligands: ALD |
Organism: Carica papaya
Method: X-RAY DIFFRACTION
Release Date: 1999-08-12
Ligands: ALD
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Crystal Structure Of Cysteine Protease Human Cathepsin K In Complex With A Covalent Peptidomimetic Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 1999-06-08 Classification: HYDROLASE Ligands: I10 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 1999-06-08
Ligands: I10
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Crystal Structure Of The Cysteine Protease Human Cathepsin K In Complex With A Covalent Symmetric Diacylaminomethyl Ketone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 1998-10-14 Classification: HYDROLASE Ligands: SDK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 1998-10-14
Ligands: SDK
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Crystal Structure Of The Cysteine Protease Human Cathepsin K In Complex With A Covalent Propanone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 1998-10-14 Classification: HYDROLASE Ligands: POS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 1998-10-14
Ligands: POS
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Crystal Structure Of The Cysteine Protease Human Cathepsin K In Complex With A Covalent Pyrrolidinone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 1998-10-14 Classification: HYDROLASE Ligands: PCM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 1998-10-14
Ligands: PCM
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Crystal Structure Of The Cysteine Protease Human Cathepsin K In Complex With A Covalent Pyrrolidinone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 1998-10-14 Classification: HYDROLASE Ligands: INP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 1998-10-14
Ligands: INP
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Design, Synthesis, And Kinetic Evaluation Of High-Affinity Fkbp Ligands, And The X-Ray Crystal Structures Of Their Complexes With Fkbp12
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 1994-01-31 Classification: CIS-TRANS ISOMERASE Ligands: SB3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 1994-01-31
Ligands: SB3
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Design, Synthesis, And Kinetic Evaluation Of High-Affinity Fkbp Ligands, And The X-Ray Crystal Structures Of Their Complexes With Fkbp12
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 1994-01-31 Classification: CIS-TRANS ISOMERASE Ligands: SBX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 1994-01-31
Ligands: SBX
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Design, Synthesis, And Kinetic Evaluation Of High-Affinity Fkbp Ligands, And The X-Ray Crystal Structures Of Their Complexes With Fkbp12
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 1994-01-31 Classification: CIS-TRANS ISOMERASE Ligands: SB1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 1994-01-31
Ligands: SB1
