Search Count: 9
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Fragment-Based Discovery Of A Novel Bruton'S Tyrosine Kinase Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.25 Å Release Date: 2021-09-08 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: IMD, PGO, 0BQ, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-08
Ligands: IMD, PGO, 0BQ, EDO
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Fragment-Based Discovery Of A Novel Bruton'S Tyrosine Kinase Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2021-09-08 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: IMD, EDO, DMS, 0UW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-08
Ligands: IMD, EDO, DMS, 0UW
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Fragment-Based Discovery Of A Novel Bruton'S Tyrosine Kinase Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2021-09-08 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: IMD, PGO, DMS, 0GW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-08
Ligands: IMD, PGO, DMS, 0GW
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Fragment-Based Drug Design Of A Novel, Covalent Bruton'S Tyrosine Kinase Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2021-09-08 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: IMD, 0CI, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-08
Ligands: IMD, 0CI, DMS
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Discovery Of Tak-659, An Orally Available Investigational Inhibitor Of Spleen Tyrosine Kinase (Syk)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.93 Å Release Date: 2016-11-30 Classification: Transferase/Transferase Inhibitor Ligands: 7KG, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-30
Ligands: 7KG, EDO
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Discovery Of Tak-659, An Orally Available Investigational Inhibitor Of Spleen Tyrosine Kinase (Syk)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.77 Å Release Date: 2016-11-30 Classification: Transferase/Transferase Inhibitor Ligands: 7KF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-30
Ligands: 7KF
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Fragment-Based Discovery Of A Small Molecule Reversible Inhibitor Of Bruton'S Tyrosine Kinase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2015-07-01 Classification: TRANSFERASE Ligands: IMD, IPA, EDO, 4L6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-07-01
Ligands: IMD, IPA, EDO, 4L6
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Crystal Structure Of Bruton'S Tyrosine Kinase Bound To A Cinnoline Fragment
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2015-07-01 Classification: Transferase/Transferase Inhibitor Ligands: IMD, IPA, DMS, 4RU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-07-01
Ligands: IMD, IPA, DMS, 4RU
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Crystal Structure Of Bruton'S Tyrosine Kinase In Complex With A Substituted Cinnoline
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2015-07-01 Classification: Transferase/Transferase Inhibitor Ligands: IMD, IPA, DMS, 4RV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-07-01
Ligands: IMD, IPA, DMS, 4RV