Search Count: 17
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Crystal Structure Of Dpp9 In Complex With A 4-Oxo-B-Lactam Based Inhibitor, A295
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.81 Å Release Date: 2022-09-28 Classification: HYDROLASE Ligands: KBO, EDO, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-09-28
Ligands: KBO, EDO, PEG
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Crystal Structure Of Compound 10 In Complex With The Bromodomain Of Human Smarca2 And Pvhl:Elonginc:Elonginb
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.32 Å Release Date: 2022-09-14 Classification: LIGASE Ligands: IOD, IFJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-09-14
Ligands: IOD, IFJ
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Crystal Structure Of Compound 6 In Complex With The Bromodomain Of Human Smarca2 And Pvhl:Elonginc:Elonginb
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2022-09-14 Classification: LIGASE Ligands: IFF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-09-14
Ligands: IFF
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Crystal Structure Of Compound 4 In Complex With The Bromodomain Of Human Smarca2 And Pvhl:Elonginc:Elonginb
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.32 Å Release Date: 2022-09-14 Classification: LIGASE Ligands: IF8, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-09-14
Ligands: IF8, ZN
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Crystal Structure Of Protac 5 In Complex With The Bromodomain Of Human Smarca2 And Pvhl:Elonginc:Elonginb
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.24 Å Release Date: 2022-09-07 Classification: LIGASE Ligands: IEI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-09-07
Ligands: IEI
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Crystal Structure Of Dpp8 In Complex With A 4-Oxo-B-Lactam Based Inhibitor, L84
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2021-07-14 Classification: HYDROLASE Ligands: MQ2, TMO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-14
Ligands: MQ2, TMO
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Crystal Structure Of Dpp8 In Complex With A 4-Oxo-B-Lactam Based Inhibitor, B142
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.44 Å Release Date: 2021-07-07 Classification: HYDROLASE Ligands: TMO, 2YI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-07
Ligands: TMO, 2YI
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Crystal Structure Of Dpp8 In Complex With A 4-Oxo-B-Lactam Based Inhibitor, 91
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2021-06-30 Classification: HYDROLASE Ligands: TMO, QXQ, GOL, PO4, QXT, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-06-30
Ligands: TMO, QXQ, GOL, PO4, QXT, CL
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Crystal Structure Of Dpp8 In Complex With A 4-Oxo-B-Lactam Based Inhibitor, A272
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2021-06-30 Classification: HYDROLASE Ligands: QXK, TMO, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-06-30
Ligands: QXK, TMO, CL
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Crystal Structure Of Dpp8 In Complex With A 4-Oxo-B-Lactam Based Inhibitor, A241
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2021-06-30 Classification: HYDROLASE Ligands: QXN, GOL, TMO, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-06-30
Ligands: QXN, GOL, TMO, CL
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Crystal Structure Of Dpp8 In Complex With A 4-Oxo-B-Lactam Based Inhibitor, B114
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2021-06-30 Classification: HYDROLASE Ligands: TMO, PO4, GOL, S9Z |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-06-30
Ligands: TMO, PO4, GOL, S9Z
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Crystal Structure Of Dpp8 In Complex With A 4-Oxo-B-Lactam Based Inhibitor, B115
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.69 Å Release Date: 2021-06-30 Classification: HYDROLASE Ligands: TMO, PO4, S9W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-06-30
Ligands: TMO, PO4, S9W
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Beta-Catenin In Complex With Compound 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.81 Å Release Date: 2020-12-16 Classification: ONCOPROTEIN Ligands: R9Q |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-16
Ligands: R9Q
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Crystal Structure Of Protac 2 In Complex With The Bromodomain Of Human Smarca2 And Pvhl:Elonginc:Elonginb
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2019-06-12 Classification: GENE REGULATION Ligands: EDO, FWZ, EPE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-12
Ligands: EDO, FWZ, EPE
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Crystal Structure Of Protac 1 In Complex With The Bromodomain Of Human Smarca2 And Pvhl:Elonginc:Elonginb
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.24 Å Release Date: 2019-06-12 Classification: GENE REGULATION Ligands: FX8, EDO, FMT, EPE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-12
Ligands: FX8, EDO, FMT, EPE
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Crystal Structure Of The Bromodomain Of Human Smarca2 In Complex With Smarca-Bd Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.31 Å Release Date: 2019-06-12 Classification: GENE REGULATION Ligands: FX5, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-12
Ligands: FX5, ZN
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Crystal Structure Of Protac 2 In Complex With The Bromodomain Of Human Smarca4 And Pvhl:Elonginc:Elonginb
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.76 Å Release Date: 2019-06-12 Classification: TRANSCRIPTION Ligands: FWZ, DMS, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-12
Ligands: FWZ, DMS, EDO
