Search Count: 12
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A Check On Rational Drug Design. Crystal Structure Of A Complex Of Hiv-1 Protease With A Novel Gamma-Turn Mimetic
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 1995-07-10 Classification: HYDROLASE (ACID PROTEASE) Ligands: GAN |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 1995-07-10
Ligands: GAN
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An Orally-Bioavailable Hiv-1 Protease Inhibitor Containing An Imidazole-Derived Peptide Bond Replacement. Crystallographic And Pharmacokinetic Analysis
Organism: Human immunodeficiency virus type 1 bh10
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 1994-10-15 Classification: HYDROLASE(ACID PROTEASE) Ligands: IM1 |
Organism: Human immunodeficiency virus type 1 bh10
Method: X-RAY DIFFRACTION
Release Date: 1994-10-15
Ligands: IM1
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Rational Design, Synthesis And Crystallographic Analysis Of A Hydroxyethylene-Based Hiv-1 Protease Inhibitor Containing A Heterocyclic P1'-P2' Amide Bond Isostere
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 1994-08-31 Classification: HYDROLASE(ACID PROTEINASE) Ligands: RUN |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 1994-08-31
Ligands: RUN
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The Crystal Structures At 2.2 Angstroms Resolution Of Hydroxyethylene-Based Inhibitors Bound To Human Immunodeficiency Virus Type 1 Protease Show That The Inhibitors Are Present In Two Distinct Orientations
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 1994-05-31 Classification: HYDROLASE/HYDROLASE INHIBITOR |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 1994-05-31
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The Crystal Structures At 2.2 Angstroms Resolution Of Hydroxyethylene-Based Inhibitors Bound To Human Immunodeficiency Virus Type 1 Protease Show That The Inhibitors Are Present In Two Distinct Orientations
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 1994-05-31 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: PSI |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 1994-05-31
Ligands: PSI
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Three-Dimensional Structure Of A Siv Protease(Slash)Inhibitor Complex. Implications For The Design Of Hiv-1 And Hiv-2 Protease Inhibitors
Organism: Simian immunodeficiency virus
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 1994-01-31 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: PSI |
Organism: Simian immunodeficiency virus
Method: X-RAY DIFFRACTION
Release Date: 1994-01-31
Ligands: PSI
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Inhibition Of Human Immunodeficiency Virus-1 Protease By A C2-Symmetric Phosphinate Synthesis And Crystallographic Analysis
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 1993-10-31 Classification: HYDROLASE(ACID PROTEINASE) Ligands: PHP |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 1993-10-31
Ligands: PHP
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A Metal-Mediated Hydride Shift Mechanism For Xylose Isomerase Based On The 1.6 Angstroms Streptomyces Rubiginosus Structures With Xylitol And D-Xylose
Organism: Streptomyces rubiginosus
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 1992-07-15 Classification: ISOMERASE(INTRAMOLECULAR OXIDOREDUCTASE) Ligands: MN |
Organism: Streptomyces rubiginosus
Method: X-RAY DIFFRACTION
Release Date: 1992-07-15
Ligands: MN
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A Metal-Mediated Hydride Shift Mechanism For Xylose Isomerase Based On The 1.6 Angstroms Streptomyces Rubiginosus Structures With Xylitol And D-Xylose
Organism: Streptomyces rubiginosus
Method: X-RAY DIFFRACTION Resolution:1.71 Å Release Date: 1992-07-15 Classification: ISOMERASE(INTRAMOLECULAR OXIDOREDUCTASE) Ligands: XYL, MG |
Organism: Streptomyces rubiginosus
Method: X-RAY DIFFRACTION
Release Date: 1992-07-15
Ligands: XYL, MG
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A Metal-Mediated Hydride Shift Mechanism For Xylose Isomerase Based On The 1.6 Angstroms Streptomyces Rubiginosus Structures With Xylitol And D-Xylose
Organism: Streptomyces rubiginosus
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 1992-07-15 Classification: ISOMERASE(INTRAMOLECULAR OXIDOREDUCTASE) Ligands: XYS, XLS, MG |
Organism: Streptomyces rubiginosus
Method: X-RAY DIFFRACTION
Release Date: 1992-07-15
Ligands: XYS, XLS, MG
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A Metal-Mediated Hydride Shift Mechanism For Xylose Isomerase Based On The 1.6 Angstroms Streptomyces Rubiginosus Structures With Xylitol And D-Xylose
Organism: Streptomyces rubiginosus
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 1992-07-15 Classification: ISOMERASE(INTRAMOLECULAR OXIDOREDUCTASE) Ligands: XLS, XYS, MN |
Organism: Streptomyces rubiginosus
Method: X-RAY DIFFRACTION
Release Date: 1992-07-15
Ligands: XLS, XYS, MN
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The Three-Dimensional Structure Of Recombinant Bovine Chymosin At 2.3 Angstroms Resolution
Organism: Bos taurus
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 1990-01-15 Classification: HYDROLASE(ACID PROTEINASE) |
Organism: Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 1990-01-15